Compile Data Set for Download or QSAR
maximum 50k data
Found 12 Enz. Inhib. hit(s) with all data for entry = 50026245
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50244177(1'-[(3-methyl-1-phenyl-1H-pyrazol-4-yl)methyl]-3H-...)
Affinity DataIC50:  740nMAssay Description:Displacement of [35S]MK499 from human ERG in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50244177(1'-[(3-methyl-1-phenyl-1H-pyrazol-4-yl)methyl]-3H-...)
Affinity DataIC50:  3.20E+3nMAssay Description:Displacement of [3H]diprenorphin from human cloned mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50244275(1'-{[3-methyl-1-(3-methylpyridin-2-yl)-1H-pyrazol-...)
Affinity DataIC50:  4.40E+3nMAssay Description:Displacement of [3H]diprenorphin from human cloned mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50244247(1'-{[1-(3-chloropyridin-2-yl)-3-methyl-1H-pyrazol-...)
Affinity DataIC50:  7.40E+3nMAssay Description:Displacement of [3H]diprenorphin from human cloned mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50244247(1'-{[1-(3-chloropyridin-2-yl)-3-methyl-1H-pyrazol-...)
Affinity DataIC50:  7.80E+3nMAssay Description:Displacement of [35S]MK499 from human ERG in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50244177(1'-[(3-methyl-1-phenyl-1H-pyrazol-4-yl)methyl]-3H-...)
Affinity DataIC50:  9.70E+3nMAssay Description:Displacement of [3H]U69593 from human cloned kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50244247(1'-{[1-(3-chloropyridin-2-yl)-3-methyl-1H-pyrazol-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]U69593 from human cloned kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50244313(1'-{[1-(3-chloropyridin-2-yl)-1H-pyrazol-4-yl]meth...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]diprenorphin from human cloned mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50244313(1'-{[1-(3-chloropyridin-2-yl)-1H-pyrazol-4-yl]meth...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]U69593 from human cloned kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50244275(1'-{[3-methyl-1-(3-methylpyridin-2-yl)-1H-pyrazol-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]U69593 from human cloned kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50244275(1'-{[3-methyl-1-(3-methylpyridin-2-yl)-1H-pyrazol-...)
Affinity DataIC50:  1.30E+4nMAssay Description:Displacement of [35S]MK499 from human ERG in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50244313(1'-{[1-(3-chloropyridin-2-yl)-1H-pyrazol-4-yl]meth...)
Affinity DataIC50:  1.70E+4nMAssay Description:Displacement of [35S]MK499 from human ERG in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed