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Found 4 Enz. Inhib. hit(s) with all data for entry = 50043716
TargetHistone acetyltransferase KAT2B(Homo sapiens (Human))
Utrecht University

Curated by ChEMBL
LigandPNGBDBM50445037(CHEMBL3098704)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of PCAF (unknown origin) using histone H3 derived peptide as substrate after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT2B(Homo sapiens (Human))
Utrecht University

Curated by ChEMBL
LigandPNGBDBM50445038(CHEMBL3098705)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of PCAF (unknown origin) using histone H3 derived peptide as substrate after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT2B(Homo sapiens (Human))
Utrecht University

Curated by ChEMBL
LigandPNGBDBM50445037(CHEMBL3098704)
Affinity DataIC50:  3.30E+4nMAssay Description:Competitive inhibition of PCAF (unknown origin) using histone H3 derived peptide as substrate after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT2B(Homo sapiens (Human))
Utrecht University

Curated by ChEMBL
LigandPNGBDBM50445038(CHEMBL3098705)
Affinity DataIC50:  1.17E+5nMAssay Description:Competitive inhibition of PCAF (unknown origin) using histone H3 derived peptide as substrate after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed