Compile Data Set for Download or QSAR
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Found 28 Enz. Inhib. hit(s) with all data for entry = 7749
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Georg-August-University Of Goettingen

LigandPNGBDBM213831(SLRFLYEG)
Affinity DataKi:  147nM ΔG°:  -36.3kJ/moleT: 2°CAssay Description:All assays were performed in TB supplemented with 0.2% Tween 20. For inhibition assays, recombinant DPP9 (25 nM) purified from insect cells was incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Georg-August-University Of Goettingen

LigandPNGBDBM213830(SLRFLYDG)
Affinity DataKi:  167nM ΔG°:  -36.0kJ/moleT: 2°CAssay Description:All assays were performed in TB supplemented with 0.2% Tween 20. For inhibition assays, recombinant DPP9 (25 nM) purified from insect cells was incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Georg-August-University Of Goettingen

LigandPNGBDBM213831(SLRFLYEG)
Affinity DataKi:  170nM ΔG°:  -35.9kJ/moleT: 2°CAssay Description:All assays were performed in TB supplemented with 0.2% Tween 20. For inhibition assays, recombinant DPP9 (25 nM) purified from insect cells was incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Georg-August-University Of Goettingen

LigandPNGBDBM213830(SLRFLYDG)
Affinity DataKi:  179nM ΔG°:  -35.8kJ/moleT: 2°CAssay Description:All assays were performed in TB supplemented with 0.2% Tween 20. For inhibition assays, recombinant DPP9 (25 nM) purified from insect cells was incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Georg-August-University Of Goettingen

LigandPNGBDBM213832(SLRFLYAG)
Affinity DataKi:  200nM ΔG°:  -35.5kJ/moleT: 2°CAssay Description:All assays were performed in TB supplemented with 0.2% Tween 20. For inhibition assays, recombinant DPP9 (25 nM) purified from insect cells was incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Georg-August-University Of Goettingen

LigandPNGBDBM213829(SLRFLWEG)
Affinity DataKi:  256nM ΔG°:  -35.0kJ/moleT: 2°CAssay Description:All assays were performed in TB supplemented with 0.2% Tween 20. For inhibition assays, recombinant DPP9 (25 nM) purified from insect cells was incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Georg-August-University Of Goettingen

LigandPNGBDBM213832(SLRFLYAG)
Affinity DataKi:  740nM ΔG°:  -32.5kJ/moleT: 2°CAssay Description:All assays were performed in TB supplemented with 0.2% Tween 20. For inhibition assays, recombinant DPP9 (25 nM) purified from insect cells was incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Georg-August-University Of Goettingen

LigandPNGBDBM213829(SLRFLWEG)
Affinity DataKi:  1.12E+3nM ΔG°:  -31.6kJ/moleT: 2°CAssay Description:All assays were performed in TB supplemented with 0.2% Tween 20. For inhibition assays, recombinant DPP9 (25 nM) purified from insect cells was incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Georg-August-University Of Goettingen

LigandPNGBDBM213828(SLRFLFEG)
Affinity DataKi:  1.34E+3nM ΔG°:  -31.2kJ/moleT: 2°CAssay Description:All assays were performed in TB supplemented with 0.2% Tween 20. For inhibition assays, recombinant DPP9 (25 nM) purified from insect cells was incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9 [H289A](Homo sapiens (Human))
Georg-August-University Of Goettingen

LigandPNGBDBM213827(E67 interacting loop (EIL) | SLRFLFEGQRIADNH)
Affinity DataKi:  3.90E+3nM ΔG°:  -28.7kJ/moleT: 2°CAssay Description:All assays were performed in TB supplemented with 0.2% Tween 20. For inhibition assays, recombinant DPP9 (25 nM) purified from insect cells was incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9 [V290A](Homo sapiens (Human))
Georg-August-University Of Goettingen

LigandPNGBDBM213827(E67 interacting loop (EIL) | SLRFLFEGQRIADNH)
Affinity DataKi:  4.00E+3nM ΔG°:  -28.6kJ/moleT: 2°CAssay Description:All assays were performed in TB supplemented with 0.2% Tween 20. For inhibition assays, recombinant DPP9 (25 nM) purified from insect cells was incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Georg-August-University Of Goettingen

LigandPNGBDBM213828(SLRFLFEG)
Affinity DataKi:  4.07E+3nM ΔG°:  -28.6kJ/moleT: 2°CAssay Description:All assays were performed in TB supplemented with 0.2% Tween 20. For inhibition assays, recombinant DPP9 (25 nM) purified from insect cells was incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9 [I288A](Homo sapiens (Human))
Georg-August-University Of Goettingen

LigandPNGBDBM213827(E67 interacting loop (EIL) | SLRFLFEGQRIADNH)
Affinity DataKi:  4.10E+3nM ΔG°:  -28.6kJ/moleT: 2°CAssay Description:All assays were performed in TB supplemented with 0.2% Tween 20. For inhibition assays, recombinant DPP9 (25 nM) purified from insect cells was incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Georg-August-University Of Goettingen

LigandPNGBDBM213827(E67 interacting loop (EIL) | SLRFLFEGQRIADNH)
Affinity DataKi:  4.20E+3nM ΔG°:  -28.5kJ/moleT: 2°CAssay Description:All assays were performed in TB supplemented with 0.2% Tween 20. For inhibition assays, recombinant DPP9 (25 nM) purified from insect cells was incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9 [Y277A](Homo sapiens (Human))
Georg-August-University Of Goettingen

LigandPNGBDBM213827(E67 interacting loop (EIL) | SLRFLFEGQRIADNH)
Affinity DataKi:  4.40E+3nM ΔG°:  -28.4kJ/moleT: 2°CAssay Description:All assays were performed in TB supplemented with 0.2% Tween 20. For inhibition assays, recombinant DPP9 (25 nM) purified from insect cells was incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9 [E286A](Homo sapiens (Human))
Georg-August-University Of Goettingen

LigandPNGBDBM213827(E67 interacting loop (EIL) | SLRFLFEGQRIADNH)
Affinity DataKi:  4.50E+3nM ΔG°:  -28.4kJ/moleT: 2°CAssay Description:All assays were performed in TB supplemented with 0.2% Tween 20. For inhibition assays, recombinant DPP9 (25 nM) purified from insect cells was incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9 [E286A,E297A](Homo sapiens (Human))
Georg-August-University Of Goettingen

LigandPNGBDBM213827(E67 interacting loop (EIL) | SLRFLFEGQRIADNH)
Affinity DataKi:  4.50E+3nM ΔG°:  -28.4kJ/moleT: 2°CAssay Description:All assays were performed in TB supplemented with 0.2% Tween 20. For inhibition assays, recombinant DPP9 (25 nM) purified from insect cells was incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9 [S292A](Homo sapiens (Human))
Georg-August-University Of Goettingen

LigandPNGBDBM213827(E67 interacting loop (EIL) | SLRFLFEGQRIADNH)
Affinity DataKi:  4.50E+3nM ΔG°:  -28.4kJ/moleT: 2°CAssay Description:All assays were performed in TB supplemented with 0.2% Tween 20. For inhibition assays, recombinant DPP9 (25 nM) purified from insect cells was incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9 [K299A](Homo sapiens (Human))
Georg-August-University Of Goettingen

LigandPNGBDBM213827(E67 interacting loop (EIL) | SLRFLFEGQRIADNH)
Affinity DataKi:  4.80E+3nM ΔG°:  -28.2kJ/moleT: 2°CAssay Description:All assays were performed in TB supplemented with 0.2% Tween 20. For inhibition assays, recombinant DPP9 (25 nM) purified from insect cells was incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9 [R298A](Homo sapiens (Human))
Georg-August-University Of Goettingen

LigandPNGBDBM213827(E67 interacting loop (EIL) | SLRFLFEGQRIADNH)
Affinity DataKi:  6.30E+3nM ΔG°:  -27.6kJ/moleT: 2°CAssay Description:All assays were performed in TB supplemented with 0.2% Tween 20. For inhibition assays, recombinant DPP9 (25 nM) purified from insect cells was incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9 [L295A](Homo sapiens (Human))
Georg-August-University Of Goettingen

LigandPNGBDBM213827(E67 interacting loop (EIL) | SLRFLFEGQRIADNH)
Affinity DataKi:  6.50E+3nM ΔG°:  -27.5kJ/moleT: 2°CAssay Description:All assays were performed in TB supplemented with 0.2% Tween 20. For inhibition assays, recombinant DPP9 (25 nM) purified from insect cells was incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9 [Y303D](Homo sapiens (Human))
Georg-August-University Of Goettingen

LigandPNGBDBM213827(E67 interacting loop (EIL) | SLRFLFEGQRIADNH)
Affinity DataKi:  9.30E+3nM ΔG°:  -26.7kJ/moleT: 2°CAssay Description:All assays were performed in TB supplemented with 0.2% Tween 20. For inhibition assays, recombinant DPP9 (25 nM) purified from insect cells was incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9 [V285A](Homo sapiens (Human))
Georg-August-University Of Goettingen

LigandPNGBDBM213827(E67 interacting loop (EIL) | SLRFLFEGQRIADNH)
Affinity DataKi:  1.04E+4nM ΔG°:  -26.4kJ/moleT: 2°CAssay Description:All assays were performed in TB supplemented with 0.2% Tween 20. For inhibition assays, recombinant DPP9 (25 nM) purified from insect cells was incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9 [D301A](Homo sapiens (Human))
Georg-August-University Of Goettingen

LigandPNGBDBM213827(E67 interacting loop (EIL) | SLRFLFEGQRIADNH)
Affinity DataKi:  1.39E+4nM ΔG°:  -25.8kJ/moleT: 2°CAssay Description:All assays were performed in TB supplemented with 0.2% Tween 20. For inhibition assays, recombinant DPP9 (25 nM) purified from insect cells was incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Georg-August-University Of Goettingen

LigandPNGBDBM213833(SLRYLYEG)
Affinity DataKi:  2.31E+4nM ΔG°:  -24.6kJ/moleT: 2°CAssay Description:All assays were performed in TB supplemented with 0.2% Tween 20. For inhibition assays, recombinant DPP9 (25 nM) purified from insect cells was incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Georg-August-University Of Goettingen

LigandPNGBDBM213833(SLRYLYEG)
Affinity DataKi:  3.52E+4nM ΔG°:  -23.6kJ/moleT: 2°CAssay Description:All assays were performed in TB supplemented with 0.2% Tween 20. For inhibition assays, recombinant DPP9 (25 nM) purified from insect cells was incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9 [Y305D](Homo sapiens (Human))
Georg-August-University Of Goettingen

LigandPNGBDBM213827(E67 interacting loop (EIL) | SLRFLFEGQRIADNH)
Affinity DataKi:  4.00E+4nM ΔG°:  -23.3kJ/moleT: 2°CAssay Description:All assays were performed in TB supplemented with 0.2% Tween 20. For inhibition assays, recombinant DPP9 (25 nM) purified from insect cells was incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9 [Y305A](Homo sapiens (Human))
Georg-August-University Of Goettingen

LigandPNGBDBM213827(E67 interacting loop (EIL) | SLRFLFEGQRIADNH)
Affinity DataKi:  4.55E+4nM ΔG°:  -23.0kJ/moleT: 2°CAssay Description:All assays were performed in TB supplemented with 0.2% Tween 20. For inhibition assays, recombinant DPP9 (25 nM) purified from insect cells was incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed