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Found 4 Enz. Inhib. hit(s) with all data for entry = 50012246
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Alma Mater Studiorum-Universit£

Curated by ChEMBL
LigandPNGBDBM50555892(CHEMBL4745205)
Affinity DataIC50:  2.66E+4nMAssay Description:Inhibition of human DNA topoisomerase 2alpha assessed as suppression of decatenation using catenated kinetoplast DNA as substrate measured after 30 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Alma Mater Studiorum-Universit£

Curated by ChEMBL
LigandPNGBDBM50127140((-)-etoposide | (5S,5aR,8aR,9R)-9-(4-hydroxy-3,5-d...)
Affinity DataIC50:  6.83E+4nMAssay Description:Inhibition of human DNA topoisomerase 2alpha assessed as suppression of decatenation using catenated kinetoplast DNA as substrate measured after 30 m...More data for this Ligand-Target Pair
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Alma Mater Studiorum-Universit£

Curated by ChEMBL
LigandPNGBDBM50555891(CHEMBL4756707)
Affinity DataIC50:  1.14E+5nMAssay Description:Inhibition of human DNA topoisomerase 2alpha assessed as suppression of decatenation using catenated kinetoplast DNA as substrate measured after 30 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Alma Mater Studiorum-Universit£

Curated by ChEMBL
LigandPNGBDBM50555893(CHEMBL4747945)
Affinity DataIC50:  1.38E+5nMAssay Description:Inhibition of human DNA topoisomerase 2alpha assessed as suppression of decatenation using catenated kinetoplast DNA as substrate measured after 30 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed