Compile Data Set for Download or QSAR
maximum 50k data
Found 18 Enz. Inhib. hit(s) with all data for entry = 50049074
TargetMicrotubule-associated protein 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50234032(CHEMBL4060668)
Affinity DataIC50:  38nMAssay Description:Inhibition of recombinant human N-terminal His tagged MetAP-2 using tripeptide Met-Ala-Ser as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMicrotubule-associated protein 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50234031(CHEMBL4082542)
Affinity DataIC50:  110nMAssay Description:Inhibition of recombinant human N-terminal His tagged MetAP-2 using tripeptide Met-Ala-Ser as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMicrotubule-associated protein 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50234025(CHEMBL4093791)
Affinity DataIC50:  230nMAssay Description:Inhibition of recombinant human N-terminal His tagged MetAP-2 using tripeptide Met-Ala-Ser as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMicrotubule-associated protein 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50234035(CHEMBL4070008)
Affinity DataIC50:  450nMAssay Description:Inhibition of recombinant human N-terminal His tagged MetAP-2 using tripeptide Met-Ala-Ser as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMicrotubule-associated protein 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50234037(CHEMBL4083510)
Affinity DataIC50:  560nMAssay Description:Inhibition of recombinant human N-terminal His tagged MetAP-2 using tripeptide Met-Ala-Ser as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMicrotubule-associated protein 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50234024(CHEMBL4097198)
Affinity DataIC50:  700nMAssay Description:Inhibition of recombinant human N-terminal His tagged MetAP-2 using tripeptide Met-Ala-Ser as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMicrotubule-associated protein 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50234033(CHEMBL4078213)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of recombinant human N-terminal His tagged MetAP-2 using tripeptide Met-Ala-Ser as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMicrotubule-associated protein 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50234022(CHEMBL4066295)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of recombinant human N-terminal His tagged MetAP-2 using tripeptide Met-Ala-Ser as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMicrotubule-associated protein 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50234020(CHEMBL4101592)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of recombinant human N-terminal His tagged MetAP-2 using tripeptide Met-Ala-Ser as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMicrotubule-associated protein 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50234030(CHEMBL4101510)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of recombinant human N-terminal His tagged MetAP-2 using tripeptide Met-Ala-Ser as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMicrotubule-associated protein 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50234021(CHEMBL4074903)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of recombinant human N-terminal His tagged MetAP-2 using tripeptide Met-Ala-Ser as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMicrotubule-associated protein 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50234027(CHEMBL4086033)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of recombinant human N-terminal His tagged MetAP-2 using tripeptide Met-Ala-Ser as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMicrotubule-associated protein 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50234028(CHEMBL4063448)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of recombinant human N-terminal His tagged MetAP-2 using tripeptide Met-Ala-Ser as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMicrotubule-associated protein 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50234034(CHEMBL4093860)
Affinity DataIC50:  3.80E+3nMAssay Description:Inhibition of recombinant human N-terminal His tagged MetAP-2 using tripeptide Met-Ala-Ser as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMicrotubule-associated protein 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50234036(CHEMBL4064507)
Affinity DataIC50:  8.60E+3nMAssay Description:Inhibition of recombinant human N-terminal His tagged MetAP-2 using tripeptide Met-Ala-Ser as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMicrotubule-associated protein 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50234026(CHEMBL4073089)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant human N-terminal His tagged MetAP-2 using tripeptide Met-Ala-Ser as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMicrotubule-associated protein 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50234019(CHEMBL4096268)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant human N-terminal His tagged MetAP-2 using tripeptide Met-Ala-Ser as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMicrotubule-associated protein 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50234029(CHEMBL4091303)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant human N-terminal His tagged MetAP-2 using tripeptide Met-Ala-Ser as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed