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Found 12 Enz. Inhib. hit(s) with all data for entry = 50048355
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50052880(CHEMBL49137 | Imidazolidin-2-ylidene-(5-methyl-qui...)
Affinity DataKi:  1.30nMAssay Description:Binding affinity towards Alpha-2 adrenergic receptor in HT-29 cellsMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM34572(BRIMONIDINE | CHEMBL844 | MLS000069370 | SMR000058...)
Affinity DataKi:  2.40nMAssay Description:Binding affinity towards Alpha-2 adrenergic receptor of HT-29 cellsMore data for this Ligand-Target Pair
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213028(CHEMBL74283)
Affinity DataKi:  6nMAssay Description:Binding affinity towards Alpha-2 adrenergic receptor in HT-29 cellsMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50052881(AGN-192172 | CHEMBL49284 | Imidazolidin-2-ylidene-...)
Affinity DataKi:  6.80nMAssay Description:Binding affinity towards Alpha-2 adrenergic receptor in HT-29 cellsMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213027(CHEMBL342029)
Affinity DataKi:  46nMAssay Description:Binding affinity towards Alpha-2 adrenergic receptor in HT-29 cellsMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213029(CHEMBL49395)
Affinity DataKi:  64nMAssay Description:Binding affinity towards Alpha-2 adrenergic receptor in HT-29 cellsMore data for this Ligand-Target Pair
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TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213028(CHEMBL74283)
Affinity DataKi:  1.10E+3nMAssay Description:Binding affinity towards Alpha-1 adrenergic receptor in human brainMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50052880(CHEMBL49137 | Imidazolidin-2-ylidene-(5-methyl-qui...)
Affinity DataKi:  1.40E+3nMAssay Description:Binding affinity towards Alpha-1 adrenergic receptor in human brainMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM34572(BRIMONIDINE | CHEMBL844 | MLS000069370 | SMR000058...)
Affinity DataKi:  1.90E+3nMAssay Description:Binding affinity towards Alpha-1 adrenergic receptor of human brainMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213027(CHEMBL342029)
Affinity DataKi:  5.10E+3nMAssay Description:Binding affinity towards Alpha-1 adrenergic receptor in human brainMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50052881(AGN-192172 | CHEMBL49284 | Imidazolidin-2-ylidene-...)
Affinity DataKi:  8.70E+3nMAssay Description:Binding affinity towards Alpha-1 adrenergic receptor in human brainMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213029(CHEMBL49395)
Affinity DataKi:  1.10E+4nMAssay Description:Binding affinity towards Alpha-1 adrenergic receptor in human brainMore data for this Ligand-Target Pair
In DepthDetails