Compile Data Set for Download or QSAR
maximum 50k data
Found 22 Enz. Inhib. hit(s) with all data for entry = 50020553
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50215029((2S)-6-amino-N-benzyl-2-[(4R)-3-oxo-4-[(phenylacet...)
Affinity DataIC50:  1.20nMAssay Description:Agonist activity at human SST5 receptor expressed in CHOK1 cells assessed as effect on forskolin-induced cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50215029((2S)-6-amino-N-benzyl-2-[(4R)-3-oxo-4-[(phenylacet...)
Affinity DataIC50:  1.20nMAssay Description:Displacement of [125I][Leu8-D-Trp22, Tyr25]-SRIF28 from human SST5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50215029((2S)-6-amino-N-benzyl-2-[(4R)-3-oxo-4-[(phenylacet...)
Affinity DataIC50:  3.30nMAssay Description:Displacement of [125I][Leu8-D-Trp22, Tyr25]-SRIF28 from human SST4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50215026((2S)-6-amino-N-benzyl-2-[(4R)-4-[(3,3-diphenylprop...)
Affinity DataIC50:  8nMAssay Description:Displacement of [125I][Leu8-D-Trp22, Tyr25]-SRIF28 from human SST5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50215026((2S)-6-amino-N-benzyl-2-[(4R)-4-[(3,3-diphenylprop...)
Affinity DataIC50:  73nMAssay Description:Displacement of [125I][Leu8-D-Trp22, Tyr25]-SRIF28 from human SST4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50215027(5-[(4R)-3-oxo-4-[(phenylacetyl)amino]-3,4,5,10-tet...)
Affinity DataIC50:  75nMAssay Description:Displacement of [125I][Leu8-D-Trp22, Tyr25]-SRIF28 from human SST4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50215029((2S)-6-amino-N-benzyl-2-[(4R)-3-oxo-4-[(phenylacet...)
Affinity DataIC50:  83nMAssay Description:Displacement of [125I][Leu8-D-Trp22, Tyr25]-SRIF28 from human SST2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50215026((2S)-6-amino-N-benzyl-2-[(4R)-4-[(3,3-diphenylprop...)
Affinity DataIC50:  89nMAssay Description:Displacement of [125I][Leu8-D-Trp22, Tyr25]-SRIF28 from human SST1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50215026((2S)-6-amino-N-benzyl-2-[(4R)-4-[(3,3-diphenylprop...)
Affinity DataIC50:  103nMAssay Description:Displacement of [125I][Leu8-D-Trp22, Tyr25]-SRIF28 from human SST2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50215028(CHEMBL227211 | N-[(4R)-2-(5-aminopentyl)-3-oxo-1,2...)
Affinity DataIC50:  129nMAssay Description:Displacement of [125I][Leu8-D-Trp22, Tyr25]-SRIF28 from human SST4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50215029((2S)-6-amino-N-benzyl-2-[(4R)-3-oxo-4-[(phenylacet...)
Affinity DataIC50:  233nMAssay Description:Displacement of [125I][Leu8-D-Trp22, Tyr25]-SRIF28 from human SST1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50215027(5-[(4R)-3-oxo-4-[(phenylacetyl)amino]-3,4,5,10-tet...)
Affinity DataIC50:  245nMAssay Description:Displacement of [125I][Leu8-D-Trp22, Tyr25]-SRIF28 from human SST5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50215029((2S)-6-amino-N-benzyl-2-[(4R)-3-oxo-4-[(phenylacet...)
Affinity DataIC50:  251nMAssay Description:Displacement of [125I][Leu8-D-Trp22, Tyr25]-SRIF28 from human SST3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50215028(CHEMBL227211 | N-[(4R)-2-(5-aminopentyl)-3-oxo-1,2...)
Affinity DataIC50:  318nMAssay Description:Displacement of [125I][Leu8-D-Trp22, Tyr25]-SRIF28 from human SST5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50215028(CHEMBL227211 | N-[(4R)-2-(5-aminopentyl)-3-oxo-1,2...)
Affinity DataIC50:  357nMAssay Description:Displacement of [125I][Leu8-D-Trp22, Tyr25]-SRIF28 from human SST2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50215026((2S)-6-amino-N-benzyl-2-[(4R)-4-[(3,3-diphenylprop...)
Affinity DataIC50:  694nMAssay Description:Displacement of [125I][Leu8-D-Trp22, Tyr25]-SRIF28 from human SST3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50215027(5-[(4R)-3-oxo-4-[(phenylacetyl)amino]-3,4,5,10-tet...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [125I][Leu8-D-Trp22, Tyr25]-SRIF28 from human SST2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50215027(5-[(4R)-3-oxo-4-[(phenylacetyl)amino]-3,4,5,10-tet...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [125I][Leu8-D-Trp22, Tyr25]-SRIF28 from human SST3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50215028(CHEMBL227211 | N-[(4R)-2-(5-aminopentyl)-3-oxo-1,2...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [125I][Leu8-D-Trp22, Tyr25]-SRIF28 from human SST3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50215027(5-[(4R)-3-oxo-4-[(phenylacetyl)amino]-3,4,5,10-tet...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [125I][Leu8-D-Trp22, Tyr25]-SRIF28 from human SST1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50215028(CHEMBL227211 | N-[(4R)-2-(5-aminopentyl)-3-oxo-1,2...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [125I][Leu8-D-Trp22, Tyr25]-SRIF28 from human SST1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50215029((2S)-6-amino-N-benzyl-2-[(4R)-3-oxo-4-[(phenylacet...)
Affinity DataEC50:  13nMAssay Description:Agonist activity at human SST5 receptor expressed in CHOK1 cells assessed as effect on forskolin-induced cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed