Found 46 Enz. Inhib. hit(s) with all data for entry = 50049307 
Affinity DataKi: 0.130nMAssay Description:Displacement of [3H]estradiol from full-length human ERalpha receptor by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.180nMAssay Description:Displacement of [3H]estradiol from full-length human ERalpha receptor by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.270nMAssay Description:Displacement of [3H]estradiol from full-length human ERalpha receptor by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.320nMAssay Description:Displacement of [3H]estradiol from full-length human ERalpha receptor by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.350nMAssay Description:Displacement of [3H]estradiol from full-length human ERalpha receptor by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.360nMAssay Description:Displacement of [3H]estradiol from full-length human ERalpha receptor by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.370nMAssay Description:Displacement of [3H]estradiol from full-length human ERalpha receptor by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.370nMAssay Description:Displacement of [3H]estradiol from full-length human ERalpha receptor by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.370nMAssay Description:Inhibition constant was evaluated against Histamine N-methyl-transferaseMore data for this Ligand-Target Pair
Affinity DataKi: 0.380nMAssay Description:Displacement of [3H]estradiol from full-length human ERalpha receptor by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Displacement of [3H]estradiol from full-length human ERalpha receptor by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.430nMAssay Description:Displacement of [3H]estradiol from full-length human ERalpha receptor by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.430nMAssay Description:Displacement of [3H]estradiol from full-length human ERalpha receptor by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.450nMAssay Description:Displacement of [3H]estradiol from full-length human ERalpha receptor by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.570nMAssay Description:Displacement of [3H]estradiol from full-length human ERalpha receptor by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.650nMAssay Description:Displacement of [3H]estradiol from full-length human ERalpha receptor by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.710nMAssay Description:Displacement of [3H]estradiol from full-length human ERalpha receptor by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.710nMAssay Description:Displacement of [3H]estradiol from full-length human ERalpha receptor by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.710nMAssay Description:Displacement of [3H]estradiol from full-length human ERalpha receptor by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.740nMAssay Description:Displacement of [3H]estradiol from full-length human ERalpha receptor by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Displacement of [3H]estradiol from full-length human ERalpha receptor by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Displacement of [3H]estradiol from full-length human ERalpha receptor by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Displacement of [3H]estradiol from full-length human ERalpha receptor by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Displacement of [3H]estradiol from full-length human ERalpha receptor by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Displacement of [3H]estradiol from full-length human ERalpha receptor by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Displacement of [3H]estradiol from full-length human ERalpha receptor by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 3.30nMAssay Description:Displacement of [3H]estradiol from full-length human ERalpha receptor by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 7.10nMAssay Description:Displacement of [3H]estradiol from full-length human ERalpha receptor by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Downregulation of human ERalpha in human MCF-7 cells after 24 hrs by in-cell Western immunoassay methodMore data for this Ligand-Target Pair
Affinity DataIC50: 0.530nMAssay Description:Downregulation of human ERalpha in human MCF-7 cells after 24 hrs by in-cell Western immunoassay methodMore data for this Ligand-Target Pair
Affinity DataIC50: 2.10nMAssay Description:Downregulation of human ERalpha in human MCF-7 cells after 24 hrs by in-cell Western immunoassay methodMore data for this Ligand-Target Pair
Affinity DataIC50: 2.90nMAssay Description:Downregulation of human ERalpha in human MCF-7 cells after 24 hrs by in-cell Western immunoassay methodMore data for this Ligand-Target Pair
Affinity DataIC50: 4.30nMAssay Description:Downregulation of human ERalpha in human MCF-7 cells after 24 hrs by in-cell Western immunoassay methodMore data for this Ligand-Target Pair
Affinity DataIC50: 5.40nMAssay Description:Downregulation of human ERalpha in human MCF-7 cells after 24 hrs by in-cell Western immunoassay methodMore data for this Ligand-Target Pair
Affinity DataIC50: 5.60nMAssay Description:Downregulation of human ERalpha in human MCF-7 cells after 24 hrs by in-cell Western immunoassay methodMore data for this Ligand-Target Pair
Affinity DataIC50: 9.10nMAssay Description:Downregulation of human ERalpha in human MCF-7 cells after 24 hrs by in-cell Western immunoassay methodMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Downregulation of human ERalpha in human MCF-7 cells after 24 hrs by in-cell Western immunoassay methodMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Downregulation of human ERalpha in human MCF-7 cells after 24 hrs by in-cell Western immunoassay methodMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Downregulation of human ERalpha in human MCF-7 cells after 24 hrs by in-cell Western immunoassay methodMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Downregulation of human ERalpha in human MCF-7 cells after 24 hrs by in-cell Western immunoassay methodMore data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Downregulation of ERalpha in human MCF-7 cells assessed as reduction of estradiol-induced GREB1 mRNA levels after 24 hrs by RT-PCR methodMore data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Downregulation of ERalpha in human MCF-7 cells assessed as reduction of estradiol-induced pS2 mRNA levels after 24 hrs by RT-PCR methodMore data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Downregulation of ERalpha in human MCF-7 cells assessed as reduction of estradiol-induced PgR mRNA levels after 24 hrs by RT-PCR methodMore data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Downregulation of ERalpha in human MCF-7 cells assessed as reduction of estradiol-induced pS2 mRNA levels after 24 hrs by RT-PCR methodMore data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Downregulation of ERalpha in human MCF-7 cells assessed as reduction of estradiol-induced PgR mRNA levels after 24 hrs by RT-PCR methodMore data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Downregulation of ERalpha in human MCF-7 cells assessed as reduction of estradiol-induced GREB1 mRNA levels after 24 hrs by RT-PCR methodMore data for this Ligand-Target Pair
