Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with all data for entry = 50040968
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Hebei Medical University

Curated by ChEMBL
LigandPNGBDBM50403019(CHEMBL2208193)
Affinity DataEC50:  3.10E+3nMAssay Description:Agonist activity at PPARgamma-LBD expressed in human L02 cells co-expressing pGL3-SV40-GAL4 after 24 hrs by luciferase reporter gene based transactiv...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Hebei Medical University

Curated by ChEMBL
LigandPNGBDBM28681(5-[(4-{2-[methyl(pyridin-2-yl)amino]ethoxy}phenyl)...)
Affinity DataEC50:  900nMAssay Description:Agonist activity at PPARgamma-LBD expressed in human L02 cells co-expressing pGL3-SV40-GAL4 after 24 hrs by luciferase reporter gene based transactiv...More data for this Ligand-Target Pair