Compile Data Set for Download or QSAR
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Found 28 Enz. Inhib. hit(s) with all data for entry = 50012517
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50119864(2-{2-[4-(2-Chloro-benzyl)-piperazin-1-yl]-ethylsul...)
Affinity DataKi:  4.30nMAssay Description:Affinity for 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50119871(5-(3-Methoxy-benzyl)-2-{2-[4-(3-trifluoromethyl-be...)
Affinity DataKi:  4.90nMAssay Description:Affinity for 5-hydroxytryptamine 2C receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50119867(5-(2-Methoxy-benzyl)-2-{2-[4-(3-trifluoromethyl-be...)
Affinity DataKi:  5.5nMAssay Description:Affinity for 5-hydroxytryptamine 2C receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50119875(2-(4,6-Diamino-2-{2-[4-(2-chloro-benzyl)-piperazin...)
Affinity DataKi:  5.5nMAssay Description:Affinity for 5-hydroxytryptamine 2C receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50119870(2-{2-[4-(2-Chloro-benzyl)-piperazin-1-yl]-ethylsul...)
Affinity DataKi:  5.70nMAssay Description:Affinity for 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50119873(2-(4,6-Diamino-2-{2-[4-(3-trifluoromethyl-benzyl)-...)
Affinity DataKi:  6.20nMAssay Description:Affinity for 5-hydroxytryptamine 2C receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50119874(5-(2-Methoxy-benzyl)-2-{2-[4-(2-trifluoromethyl-be...)
Affinity DataKi:  7.70nMAssay Description:Affinity for 5-hydroxytryptamine 2C receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50119866(5-(2-Isopropoxy-benzyl)-2-{2-[4-(3-trifluoromethyl...)
Affinity DataKi:  8.60nMAssay Description:Affinity for 5-hydroxytryptamine 2C receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50119863(5-(2-Chloro-benzyl)-2-{2-[4-(2-chloro-benzyl)-pipe...)
Affinity DataKi:  8.70nMAssay Description:Affinity for 5-hydroxytryptamine 2C receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50119865(5-(2-Ethoxy-benzyl)-2-{2-[4-(3-trifluoromethyl-ben...)
Affinity DataKi:  9.10nMAssay Description:Affinity for 5-hydroxytryptamine 2C receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50119870(2-{2-[4-(2-Chloro-benzyl)-piperazin-1-yl]-ethylsul...)
Affinity DataKi:  10nMAssay Description:Affinity for 5-hydroxytryptamine 2C receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50119869(5-Benzyl-2-{2-[4-(2-chloro-benzyl)-piperazin-1-yl]...)
Affinity DataKi:  12nMAssay Description:Affinity for 5-hydroxytryptamine 2C receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50119868(5-(4-Methoxy-benzyl)-2-{2-[4-(2-methyl-benzyl)-pip...)
Affinity DataKi:  12nMAssay Description:Affinity for 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50119863(5-(2-Chloro-benzyl)-2-{2-[4-(2-chloro-benzyl)-pipe...)
Affinity DataKi:  12nMAssay Description:Affinity for 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50119862(5-(4-Methoxy-benzyl)-2-{2-[4-(4-methyl-benzyl)-pip...)
Affinity DataKi:  13nMAssay Description:Affinity for 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50119868(5-(4-Methoxy-benzyl)-2-{2-[4-(2-methyl-benzyl)-pip...)
Affinity DataKi:  16nMAssay Description:Affinity for 5-hydroxytryptamine 2C receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50119864(2-{2-[4-(2-Chloro-benzyl)-piperazin-1-yl]-ethylsul...)
Affinity DataKi:  18nMAssay Description:Affinity for 5-hydroxytryptamine 2C receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50119869(5-Benzyl-2-{2-[4-(2-chloro-benzyl)-piperazin-1-yl]...)
Affinity DataKi:  18nMAssay Description:Affinity for 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50119872(5-Benzyl-2-{2-[4-(2-trifluoromethyl-benzyl)-pipera...)
Affinity DataKi:  21nMAssay Description:Affinity for 5-hydroxytryptamine 2C receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50119875(2-(4,6-Diamino-2-{2-[4-(2-chloro-benzyl)-piperazin...)
Affinity DataKi:  23nMAssay Description:Affinity for 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50119871(5-(3-Methoxy-benzyl)-2-{2-[4-(3-trifluoromethyl-be...)
Affinity DataKi:  45nMAssay Description:Affinity for 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50119874(5-(2-Methoxy-benzyl)-2-{2-[4-(2-trifluoromethyl-be...)
Affinity DataKi:  48nMAssay Description:Affinity for 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50119867(5-(2-Methoxy-benzyl)-2-{2-[4-(3-trifluoromethyl-be...)
Affinity DataKi:  60nMAssay Description:Affinity for 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50119872(5-Benzyl-2-{2-[4-(2-trifluoromethyl-benzyl)-pipera...)
Affinity DataKi:  61nMAssay Description:Affinity for 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50119865(5-(2-Ethoxy-benzyl)-2-{2-[4-(3-trifluoromethyl-ben...)
Affinity DataKi:  70nMAssay Description:Affinity for 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50119873(2-(4,6-Diamino-2-{2-[4-(3-trifluoromethyl-benzyl)-...)
Affinity DataKi:  93nMAssay Description:Affinity for 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50119866(5-(2-Isopropoxy-benzyl)-2-{2-[4-(3-trifluoromethyl...)
Affinity DataKi:  121nMAssay Description:Affinity for 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Egis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50119862(5-(4-Methoxy-benzyl)-2-{2-[4-(4-methyl-benzyl)-pip...)
Affinity DataKi:  300nMAssay Description:Affinity for 5-hydroxytryptamine 2C receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed