Compile Data Set for Download or QSAR
maximum 50k data
Found 38 Enz. Inhib. hit(s) with all data for entry = 50044666
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM86757(CAS_0 | NSC_11603174 | [11C]MMP)
Affinity DataKi:  0.150nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50024574(CHEMBL3330616)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50024567(CHEMBL3330623)
Affinity DataKi:  0.440nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50024643(CHEMBL3329234)
Affinity DataKi:  0.460nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50024647(CHEMBL3330599)
Affinity DataKi:  0.660nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50024646(CHEMBL3330600)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50024595(CHEMBL3330605)
Affinity DataKi:  0.835nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50024580(CHEMBL3330612)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50024577(CHEMBL3330614)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50024573(CHEMBL3330617 | US9290463, A)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50024584(CHEMBL3330609)
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50024582(CHEMBL3330611)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50024566(CHEMBL3330624)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50024605(CHEMBL3330603 | US9290463, E)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50024583(CHEMBL3330610)
Affinity DataKi:  2.80nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50024587(CHEMBL3330606)
Affinity DataKi:  4.80nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50024575(CHEMBL3330615)
Affinity DataKi:  8nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50024585(CHEMBL3330608)
Affinity DataKi:  28nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50024603(CHEMBL3330604 | US9290463, C)
Affinity DataKi:  59nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50024578(CHEMBL3330613)
Affinity DataKi:  68nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50024568(CHEMBL3330622)
Affinity DataKi:  150nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50024564(CHEMBL3330626)
Affinity DataKi:  175nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50024576(Eptapirone)
Affinity DataKi:  175nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50024645(CHEMBL3330601)
Affinity DataKi:  180nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50024571(CHEMBL3330619)
Affinity DataKi:  180nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50024648(CHEMBL3330598)
Affinity DataKi:  190nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50024586(CHEMBL3330607)
Affinity DataKi:  215nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50024644(CHEMBL3330602)
Affinity DataKi:  220nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50024572(CHEMBL3330618)
Affinity DataKi:  240nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50024565(CHEMBL3330625)
Affinity DataKi:  240nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50024569(CHEMBL3330621)
Affinity DataKi:  250nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50024570(CHEMBL3330620)
Affinity DataKi:  350nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50024650(CHEMBL3330597)
Affinity DataKi:  414nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1AR (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50024574(CHEMBL3330616)
Affinity DataEC50:  0.200nMAssay Description:Agonist activity at human 5HT1AR expressed in CHO cells assessed as increase in [35S]GTPgammaS binding by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM86757(CAS_0 | NSC_11603174 | [11C]MMP)
Affinity DataEC50:  0.100nMAssay Description:Agonist activity at human 5HT1AR expressed in CHO cells assessed as increase in [35S]GTPgammaS binding by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50024605(CHEMBL3330603 | US9290463, E)
Affinity DataEC50:  0.300nMAssay Description:Agonist activity at human 5HT1AR expressed in CHO cells assessed as increase in [35S]GTPgammaS binding by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50024580(CHEMBL3330612)
Affinity DataEC50:  0.0800nMAssay Description:Agonist activity at human 5HT1AR expressed in CHO cells assessed as increase in [35S]GTPgammaS binding by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Stony Brook University

Curated by ChEMBL
LigandPNGBDBM50024577(CHEMBL3330614)
Affinity DataEC50:  0.800nMAssay Description:Agonist activity at human 5HT1AR expressed in CHO cells assessed as increase in [35S]GTPgammaS binding by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed