Compile Data Set for Download or QSAR
maximum 50k data
Found 8 Enz. Inhib. hit(s) with all data for entry = 50010217
TargetInsulin receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50092148(2-Benzo[b]thiophen-3-yl-3,6-dihydroxy-5-phenyl-[1,...)
Affinity DataEC50:  1.00E+3nMAssay Description:Activation of human insulin receptor tyrosine kinase (IRTK)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50092149(2-[2-(1,1-Dimethyl-allyl)-1H-indol-3-yl]-3,6-dihyd...)
Affinity DataEC50:  5.00E+3nMAssay Description:Activation of human insulin receptor tyrosine kinase (IRTK)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50092146(2-Benzofuran-3-yl-3,6-dihydroxy-5-phenyl-[1,4]benz...)
Affinity DataEC50:  1.50E+3nMAssay Description:Activation of human insulin receptor tyrosine kinase (IRTK)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50092150(2,5-Dihydroxy-3-(1-methyl-1H-indol-3-yl)-6-phenyl-...)
Affinity DataEC50:  300nMAssay Description:Activation of human insulin receptor tyrosine kinase (IRTK)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50092143(2,5-Dihydroxy-3-(1H-indol-3-yl)-6-phenyl-[1,4]benz...)
Affinity DataEC50:  300nMAssay Description:Activation of human insulin receptor tyrosine kinase (IRTK)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50092145(2,5-Dihydroxy-3-naphthalen-2-yl-6-phenyl-[1,4]benz...)
Affinity DataEC50:  3.00E+4nMAssay Description:Activation of human insulin receptor tyrosine kinase (IRTK)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50092144(2,5-Dihydroxy-3-(1H-indol-3-yl)-6-(7-methyl-1H-ind...)
Affinity DataEC50:  7.00E+3nMAssay Description:Activation of human insulin receptor tyrosine kinase (IRTK)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50092147(2,5-Dihydroxy-3-naphthalen-1-yl-6-phenyl-[1,4]benz...)
Affinity DataEC50:  6.00E+3nMAssay Description:Activation of human insulin receptor tyrosine kinase (IRTK)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed