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Found 16 Enz. Inhib. hit(s) with all data for entry = 50038263
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universita degli Studi di Bari

Curated by ChEMBL
LigandPNGBDBM50373901(CHEMBL271987)
Affinity DataKi:  0.0300nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor expressed in HEK293 cells after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universita degli Studi di Bari

Curated by ChEMBL
LigandPNGBDBM50329675(6-methoxy-N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)...)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor expressed in HEK293 cells after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universita degli Studi di Bari

Curated by ChEMBL
LigandPNGBDBM50373895(CHEMBL259686)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor expressed in HEK293 cells after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universita degli Studi di Bari

Curated by ChEMBL
LigandPNGBDBM50373891(CHEMBL410515)
Affinity DataKi:  0.380nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor expressed in HEK293 cells after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universita degli Studi di Bari

Curated by ChEMBL
LigandPNGBDBM50373893(CHEMBL261383)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor expressed in HEK293 cells after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universita degli Studi di Bari

Curated by ChEMBL
LigandPNGBDBM50373892(CHEMBL261600)
Affinity DataKi:  0.540nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor expressed in HEK293 cells after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universita degli Studi di Bari

Curated by ChEMBL
LigandPNGBDBM50373897(CHEMBL270750)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor expressed in HEK293 cells after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universita degli Studi di Bari

Curated by ChEMBL
LigandPNGBDBM50373898(CHEMBL261824)
Affinity DataKi:  2.60nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor expressed in HEK293 cells after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universita degli Studi di Bari

Curated by ChEMBL
LigandPNGBDBM50373894(CHEMBL270736)
Affinity DataKi:  4.60nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor expressed in HEK293 cells after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universita degli Studi di Bari

Curated by ChEMBL
LigandPNGBDBM21393(7-(dipropylamino)-5,6,7,8-tetrahydronaphthalen-1-o...)
Affinity DataKi:  5.10nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor expressed in HEK293 cells after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universita degli Studi di Bari

Curated by ChEMBL
LigandPNGBDBM50373902(CHEMBL405228)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor expressed in HEK293 cells after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universita degli Studi di Bari

Curated by ChEMBL
LigandPNGBDBM50373896(CHEMBL259889)
Affinity DataKi:  14.2nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor expressed in HEK293 cells after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universita degli Studi di Bari

Curated by ChEMBL
LigandPNGBDBM50373899(CHEMBL258600)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor expressed in HEK293 cells after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universita degli Studi di Bari

Curated by ChEMBL
LigandPNGBDBM50373900(CHEMBL258602)
Affinity DataKi:  28nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor expressed in HEK293 cells after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universita degli Studi di Bari

Curated by ChEMBL
LigandPNGBDBM50373903(CHEMBL259887)
Affinity DataKi:  33nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor expressed in HEK293 cells after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universita degli Studi di Bari

Curated by ChEMBL
LigandPNGBDBM50325743(CHEMBL271989 | N-(4-(4-(2-methoxyphenyl)piperazin-...)
Affinity DataKi:  97nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor expressed in HEK293 cells after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed