TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Affinity DataIC50: 0.190nMAssay Description:Displacement of [3H]prazosin from adrenergic alpha1B receptor in Wistar rat liver membrane after 60 minsMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Affinity DataIC50: 0.254nMAssay Description:Displacement of [3H]prazosin from adrenergic alpha1A receptor in Wistar rat submaxillary gland after 60 minsMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Affinity DataIC50: 3.67nMAssay Description:Displacement of [3H]MK9112 from human recombinant adrenergic alpha2A receptor expressed in insect Sf9 cells after 60 minsMore data for this Ligand-Target Pair
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Affinity DataIC50: 27.1nMAssay Description:Displacement of radioligand from human adrenergic alpha2C receptor after 60 minsMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Affinity DataIC50: 56nMAssay Description:Displacement of [3H]prazosin from adrenergic alpha1A receptor in Wistar rat submaxillary gland after 60 minsMore data for this Ligand-Target Pair
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Affinity DataIC50: 102nMAssay Description:Displacement of [3H]prazosin from adrenergic alpha1B receptor in Wistar rat liver membrane after 60 minsMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Affinity DataIC50: 320nMAssay Description:Displacement of [3H]MK9112 from human recombinant adrenergic alpha2A receptor expressed in insect Sf9 cells after 60 minsMore data for this Ligand-Target Pair