Compile Data Set for Download or QSAR
maximum 50k data
Found 49 Enz. Inhib. hit(s) with all data for entry = 50030478
TargetNeutrophil elastase(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50296807(5-ethyl-2-(2-(4-methylpiperazin-1-yl)pyridin-3-yl)...)
Affinity DataIC50:  8.10nMAssay Description:Inhibition of human sputum neutrophil elastase by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50296805(5-ethyl-2-(2-(4-(1-methylpiperidin-4-yl)piperazin-...)
Affinity DataIC50:  8.5nMAssay Description:Inhibition of human sputum neutrophil elastase by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50296806(1-(3-(5-ethyl-4-oxo-4H-benzo[d][1,3]oxazin-2-yl)py...)
Affinity DataIC50:  8.60nMAssay Description:Inhibition of human sputum neutrophil elastase by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50296826(5-ethyl-2-(2-(4-(2-hydroxyethyl)piperazin-1-yl)pyr...)
Affinity DataIC50:  16nMAssay Description:Inhibition of human sputum neutrophil elastase by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50296830(5-ethyl-7-methoxy-2-(2-(4-(2-methoxyethyl)piperazi...)
Affinity DataIC50:  16nMAssay Description:Inhibition of human sputum neutrophil elastase by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50296834((R)-1-(3-(5-ethyl-7-methoxy-4-oxo-4H-benzo[d][1,3]...)
Affinity DataIC50:  19nMAssay Description:Inhibition of human sputum neutrophil elastase by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50296804(5-ethyl-7-methoxy-2-(2-(4-methylpiperazin-1-yl)pyr...)
Affinity DataIC50:  20nMAssay Description:Inhibition of human sputum neutrophil elastase by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50296824(2-(2-(4-(2-(dimethylamino)ethyl)piperazin-1-yl)pyr...)
Affinity DataIC50:  21nMAssay Description:Inhibition of human sputum neutrophil elastase by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50296828(5-ethyl-2-(2-(4-isobutylpiperazin-1-yl)pyridin-3-y...)
Affinity DataIC50:  21nMAssay Description:Inhibition of human sputum neutrophil elastase by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50296827(5-ethyl-7-methoxy-2-(2-(4-(2-morpholinoethyl)piper...)
Affinity DataIC50:  22nMAssay Description:Inhibition of human sputum neutrophil elastase by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50296835(2-(4-(3-(5-ethyl-7-methoxy-4-oxo-4H-benzo[d][1,3]o...)
Affinity DataIC50:  23nMAssay Description:Inhibition of human sputum neutrophil elastase by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50296825(3-(4-(3-(5-ethyl-7-methoxy-4-oxo-4H-benzo[d][1,3]o...)
Affinity DataIC50:  24nMAssay Description:Inhibition of human sputum neutrophil elastase by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50296833((S)-1-(3-(5-ethyl-7-methoxy-4-oxo-4H-benzo[d][1,3]...)
Affinity DataIC50:  25nMAssay Description:Inhibition of human sputum neutrophil elastase by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50296829(2-(2-(4-butylpiperazin-1-yl)pyridin-3-yl)-5-ethyl-...)
Affinity DataIC50:  27nMAssay Description:Inhibition of human sputum neutrophil elastase by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50296831(2-(2-(4-(cyclopropylmethyl)piperazin-1-yl)pyridin-...)
Affinity DataIC50:  28nMAssay Description:Inhibition of human sputum neutrophil elastase by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50296802(5-ethyl-7-methoxy-2-(2-(4-(1-methylpiperidin-4-yl)...)
Affinity DataIC50:  28nMAssay Description:Inhibition of human sputum neutrophil elastase by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50296803(1-(3-(5-ethyl-7-methoxy-4-oxo-4H-benzo[d][1,3]oxaz...)
Affinity DataIC50:  28nMAssay Description:Inhibition of human sputum neutrophil elastase by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50296832(2-(2-(4-cyclopentylpiperazin-1-yl)pyridin-3-yl)-5-...)
Affinity DataIC50:  34nMAssay Description:Inhibition of human sputum neutrophil elastase by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50296823(5-methyl-2-(2-phenoxypyridin-3-yl)-4H-benzo[d][1,3...)
Affinity DataIC50:  61nMAssay Description:Inhibition of human sputum neutrophil elastase by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50296811(2-(2-(1H-imidazol-1-yl)pyridin-3-yl)-5-methyl-4H-b...)
Affinity DataIC50:  64nMAssay Description:Inhibition of human sputum neutrophil elastase by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50296797(7-methoxy-2-(2-(4-(1-methylpiperidin-4-yl)piperazi...)
Affinity DataIC50:  71nMAssay Description:Inhibition of human sputum neutrophil elastase by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50296808(5-methyl-2-(2-(4-(1-methylpiperidin-4-yl)piperazin...)
Affinity DataIC50:  74nMAssay Description:Inhibition of human sputum neutrophil elastase by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50296809(1-(3-(5-methyl-4-oxo-4H-benzo[d][1,3]oxazin-2-yl)p...)
Affinity DataIC50:  79nMAssay Description:Inhibition of human sputum neutrophil elastase by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50296819(2-(2-methoxypyridin-3-yl)-5-methyl-4H-benzo[d][1,3...)
Affinity DataIC50:  85nMAssay Description:Inhibition of human sputum neutrophil elastase by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50296818(5-methyl-2-(2-methylpyridin-3-yl)-4H-benzo[d][1,3]...)
Affinity DataIC50:  87nMAssay Description:Inhibition of human sputum neutrophil elastase by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50296810(5-methyl-2-(2-(4-methylpiperazin-1-yl)pyridin-3-yl...)
Affinity DataIC50:  93nMAssay Description:Inhibition of human sputum neutrophil elastase by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50296812(2-(2-((2-(dimethylamino)ethyl)(methyl)amino)pyridi...)
Affinity DataIC50:  110nMAssay Description:Inhibition of human sputum neutrophil elastase by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50296840(5-cyclopropyl-7-methoxy-2-(2-(4-(1-methylpiperidin...)
Affinity DataIC50:  110nMAssay Description:Inhibition of human sputum neutrophil elastase by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50296793(5-cyclopropyl-7-methoxy-2-(2-(4-methylpiperazin-1-...)
Affinity DataIC50:  120nMAssay Description:Inhibition of human sputum neutrophil elastase by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50296792(1-(3-(5-cyclopropyl-7-methoxy-4-oxo-4H-benzo[d][1,...)
Affinity DataIC50:  140nMAssay Description:Inhibition of human sputum neutrophil elastase by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50296794(5-isopropyl-7-methoxy-2-(2-(4-(1-methylpiperidin-4...)
Affinity DataIC50:  140nMAssay Description:Inhibition of human sputum neutrophil elastase by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50296839(5-cyclobutyl-7-methoxy-2-(2-(4-methylpiperazin-1-y...)
Affinity DataIC50:  150nMAssay Description:Inhibition of human sputum neutrophil elastase by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50296816(5-chloro-2-(2-phenoxypyridin-3-yl)-4H-benzo[d][1,3...)
Affinity DataIC50:  160nMAssay Description:Inhibition of human sputum neutrophil elastase by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50296822(5-methyl-2-(2-phenoxyphenyl)-4H-benzo[d][1,3]oxazi...)
Affinity DataIC50:  170nMAssay Description:Inhibition of human sputum neutrophil elastase by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50296798(1-(3-(7-methoxy-4-oxo-5-propyl-4H-benzo[d][1,3]oxa...)
Affinity DataIC50:  180nMAssay Description:Inhibition of human sputum neutrophil elastase by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50296796(5-isopropyl-7-methoxy-2-(2-(4-methylpiperazin-1-yl...)
Affinity DataIC50:  210nMAssay Description:Inhibition of human sputum neutrophil elastase by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50296799(7-methoxy-2-(2-(4-methylpiperazin-1-yl)pyridin-3-y...)
Affinity DataIC50:  250nMAssay Description:Inhibition of human sputum neutrophil elastase by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50296795(1-(3-(5-isopropyl-7-methoxy-4-oxo-4H-benzo[d][1,3]...)
Affinity DataIC50:  330nMAssay Description:Inhibition of human sputum neutrophil elastase by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50296815(5-methoxy-2-(2-phenoxypyridin-3-yl)-4H-benzo[d][1,...)
Affinity DataIC50:  390nMAssay Description:Inhibition of human sputum neutrophil elastase by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50296817(5-methyl-2-(6-methylpyridin-3-yl)-4H-benzo[d][1,3]...)
Affinity DataIC50:  710nMAssay Description:Inhibition of human sputum neutrophil elastase by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50296837(5-cyclobutyl-7-methoxy-2-(2-(4-(1-methylpiperidin-...)
Affinity DataIC50:  850nMAssay Description:Inhibition of human sputum neutrophil elastase by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50296820(5-methyl-2-(pyridin-3-yl)-4H-benzo[d][1,3]oxazin-4...)
Affinity DataIC50:  900nMAssay Description:Inhibition of human sputum neutrophil elastase by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50296838(1-(3-(5-cyclobutyl-7-methoxy-4-oxo-4H-benzo[d][1,3...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of human sputum neutrophil elastase by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50296800(7-(dimethylamino)-5-ethyl-2-(2-(4-(1-methylpiperid...)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of human sputum neutrophil elastase by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50296801(7-(dimethylamino)-5-ethyl-2-(2-(4-methylpiperazin-...)
Affinity DataIC50:  5.30E+3nMAssay Description:Inhibition of human sputum neutrophil elastase by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50296814(5-methyl-2-(2-(2-morpholinoethylamino)pyridin-3-yl...)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of human sputum neutrophil elastase by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50296813(2-(2-(2-(dimethylamino)ethylamino)pyridin-3-yl)-5-...)
Affinity DataIC50:  8.10E+3nMAssay Description:Inhibition of human sputum neutrophil elastase by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50296821(2-(2-phenoxypyridin-3-yl)-4H-benzo[d][1,3]oxazin-4...)
Affinity DataIC50:  9.30E+3nMAssay Description:Inhibition of human sputum neutrophil elastase by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50296836(5-tert-butyl-7-methoxy-2-(2-(4-methylpiperazin-1-y...)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of human sputum neutrophil elastase by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed