Found 32 Enz. Inhib. hit(s) with all data for entry = 50011825 TargetProteasome subunit beta type-5(Homo sapiens (Human))
Peking University Health Science Center
Curated by ChEMBL
Peking University Health Science Center
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta5 subunit using Suc-LLVY-Glo as substrate incubated for 2 hrs followed by substr...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Peking University Health Science Center
Curated by ChEMBL
Peking University Health Science Center
Curated by ChEMBL
Affinity DataIC50: 180nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta5 subunit using Suc-LLVY-Glo as substrate incubated for 2 hrs followed by substr...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Peking University Health Science Center
Curated by ChEMBL
Peking University Health Science Center
Curated by ChEMBL
Affinity DataIC50: 540nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta5 subunit using Suc-LLVY-Glo as substrate incubated for 2 hrs followed by substr...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Peking University Health Science Center
Curated by ChEMBL
Peking University Health Science Center
Curated by ChEMBL
Affinity DataIC50: 680nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta5 subunit using Suc-LLVY-Glo as substrate incubated for 2 hrs followed by substr...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Peking University Health Science Center
Curated by ChEMBL
Peking University Health Science Center
Curated by ChEMBL
Affinity DataIC50: 1.64E+3nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta 5 subunit using Suc-LLVY-aminoluciferin as substrate preincubated for 15 mins f...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Peking University Health Science Center
Curated by ChEMBL
Peking University Health Science Center
Curated by ChEMBL
Affinity DataIC50: 2.33E+3nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta5 subunit using Suc-LLVY-Glo as substrate incubated for 2 hrs followed by substr...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Peking University Health Science Center
Curated by ChEMBL
Peking University Health Science Center
Curated by ChEMBL
Affinity DataIC50: 3.12E+3nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta5 subunit using Suc-LLVY-Glo as substrate incubated for 2 hrs followed by substr...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Peking University Health Science Center
Curated by ChEMBL
Peking University Health Science Center
Curated by ChEMBL
Affinity DataIC50: 3.19E+3nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta5 subunit using Suc-LLVY-Glo as substrate incubated for 2 hrs followed by substr...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Peking University Health Science Center
Curated by ChEMBL
Peking University Health Science Center
Curated by ChEMBL
Affinity DataIC50: 4.16E+3nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta5 subunit using Suc-LLVY-Glo as substrate incubated for 2 hrs followed by substr...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Peking University Health Science Center
Curated by ChEMBL
Peking University Health Science Center
Curated by ChEMBL
Affinity DataIC50: 4.56E+3nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta5 subunit using Suc-LLVY-Glo as substrate incubated for 2 hrs followed by substr...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Peking University Health Science Center
Curated by ChEMBL
Peking University Health Science Center
Curated by ChEMBL
Affinity DataIC50: 5.63E+3nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta5 subunit using Suc-LLVY-Glo as substrate incubated for 2 hrs followed by substr...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Peking University Health Science Center
Curated by ChEMBL
Peking University Health Science Center
Curated by ChEMBL
Affinity DataIC50: 5.86E+3nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta5 subunit using Suc-LLVY-Glo as substrate incubated for 2 hrs followed by substr...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Peking University Health Science Center
Curated by ChEMBL
Peking University Health Science Center
Curated by ChEMBL
Affinity DataIC50: 6.30E+3nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta5 subunit using Suc-LLVY-Glo as substrate incubated for 2 hrs followed by substr...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Peking University Health Science Center
Curated by ChEMBL
Peking University Health Science Center
Curated by ChEMBL
Affinity DataIC50: 7.26E+3nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta5 subunit using Suc-LLVY-Glo as substrate incubated for 2 hrs followed by substr...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Peking University Health Science Center
Curated by ChEMBL
Peking University Health Science Center
Curated by ChEMBL
Affinity DataIC50: 7.26E+3nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta5 subunit using Suc-LLVY-Glo as substrate incubated for 2 hrs followed by substr...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Peking University Health Science Center
Curated by ChEMBL
Peking University Health Science Center
Curated by ChEMBL
Affinity DataIC50: 8.15E+3nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta 5 subunit using Suc-LLVY-aminoluciferin as substrate preincubated for 15 mins f...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Peking University Health Science Center
Curated by ChEMBL
Peking University Health Science Center
Curated by ChEMBL
Affinity DataIC50: 8.25E+3nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta5 subunit using Suc-LLVY-Glo as substrate incubated for 2 hrs followed by substr...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Peking University Health Science Center
Curated by ChEMBL
Peking University Health Science Center
Curated by ChEMBL
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta5 subunit using Suc-LLVY-Glo as substrate incubated for 2 hrs followed by substr...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Peking University Health Science Center
Curated by ChEMBL
Peking University Health Science Center
Curated by ChEMBL
Affinity DataIC50: 1.23E+4nMAssay Description:Inhibition of caspase-like activity of human 20S proteasome beta 1 subunit using Z-nLPnLD-Glo as substrate incubated for 2 hrs followed by substrate ...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Peking University Health Science Center
Curated by ChEMBL
Peking University Health Science Center
Curated by ChEMBL
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta5 subunit using Suc-LLVY-Glo as substrate incubated for 2 hrs followed by substr...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Peking University Health Science Center
Curated by ChEMBL
Peking University Health Science Center
Curated by ChEMBL
Affinity DataIC50: 1.43E+4nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta5 subunit using Suc-LLVY-Glo as substrate incubated for 2 hrs followed by substr...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Peking University Health Science Center
Curated by ChEMBL
Peking University Health Science Center
Curated by ChEMBL
Affinity DataIC50: 1.63E+4nMAssay Description:Inhibition of trypsin-like activity of human 20S proteasome beta 2 subunit using Z-LRR-Glo as substrate incubated for 2 hrs followed by substrate add...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Peking University Health Science Center
Curated by ChEMBL
Peking University Health Science Center
Curated by ChEMBL
Affinity DataIC50: 4.56E+4nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta5 subunit using Suc-LLVY-Glo as substrate incubated for 2 hrs followed by substr...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Peking University Health Science Center
Curated by ChEMBL
Peking University Health Science Center
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta5 subunit using Suc-LLVY-Glo as substrate incubated for 2 hrs followed by substr...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Peking University Health Science Center
Curated by ChEMBL
Peking University Health Science Center
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta5 subunit using Suc-LLVY-Glo as substrate incubated for 2 hrs followed by substr...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Peking University Health Science Center
Curated by ChEMBL
Peking University Health Science Center
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta5 subunit using Suc-LLVY-Glo as substrate incubated for 2 hrs followed by substr...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Peking University Health Science Center
Curated by ChEMBL
Peking University Health Science Center
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta5 subunit using Suc-LLVY-Glo as substrate incubated for 2 hrs followed by substr...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Peking University Health Science Center
Curated by ChEMBL
Peking University Health Science Center
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta5 subunit using Suc-LLVY-Glo as substrate incubated for 2 hrs followed by substr...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Peking University Health Science Center
Curated by ChEMBL
Peking University Health Science Center
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta5 subunit using Suc-LLVY-Glo as substrate incubated for 2 hrs followed by substr...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Peking University Health Science Center
Curated by ChEMBL
Peking University Health Science Center
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta5 subunit using Suc-LLVY-Glo as substrate incubated for 2 hrs followed by substr...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Peking University Health Science Center
Curated by ChEMBL
Peking University Health Science Center
Curated by ChEMBL
Affinity DataKd: 4.80E+3nMAssay Description:Binding affinity to immobilized human 20S proteasome beta 5 subunit by SPR analysisMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Peking University Health Science Center
Curated by ChEMBL
Peking University Health Science Center
Curated by ChEMBL
Affinity DataKd: 1.70E+4nMAssay Description:Binding affinity to immobilized human 20S proteasome beta 5 subunit by SPR analysisMore data for this Ligand-Target Pair
