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Found 21 Enz. Inhib. hit(s) with all data for entry = 50000091
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Jiangxi University Of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50240377(CHEMBL4095373)
Affinity DataEC50:  78nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as increase in cAMP stimulation measured after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Jiangxi University Of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50240392(CHEMBL4063625)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as increase in cAMP stimulation measured after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Jiangxi University Of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50240381(CHEMBL4078851)
Affinity DataEC50:  236nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as increase in cAMP stimulation measured after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Jiangxi University Of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50240384(CHEMBL4065265)
Affinity DataEC50:  4.90nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as increase in cAMP stimulation measured after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Jiangxi University Of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50240384(CHEMBL4065265)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as increase in cAMP stimulation measured after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Jiangxi University Of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50240387(CHEMBL4098760)
Affinity DataEC50:  1.20nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as increase in cAMP stimulation measured after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Jiangxi University Of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50240388(CHEMBL4078300)
Affinity DataEC50:  5.30nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as increase in cAMP stimulation measured after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Jiangxi University Of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50240388(CHEMBL4078300)
Affinity DataEC50:  1.80nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as increase in cAMP stimulation measured after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Jiangxi University Of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM29080(CHEMBL280065 | N-oleoylethanolamine | Oleamide MEA...)
Affinity DataEC50:  2.20E+3nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as increase in cAMP stimulation measured after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Jiangxi University Of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50240389(CHEMBL4080761)
Affinity DataEC50:  110nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as increase in cAMP stimulation measured after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Jiangxi University Of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50240390(CHEMBL4088637)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as increase in cAMP stimulation measured after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Jiangxi University Of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50240391(CHEMBL4067384)
Affinity DataEC50:  48nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as increase in cAMP stimulation measured after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Jiangxi University Of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50240391(CHEMBL4067384)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as increase in cAMP stimulation measured after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Jiangxi University Of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50240392(CHEMBL4063625)
Affinity DataEC50:  3.10nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as increase in cAMP stimulation measured after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Jiangxi University Of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50240394(CHEMBL4062726)
Affinity DataEC50:  6.40nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as increase in cAMP stimulation measured after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Jiangxi University Of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50240394(CHEMBL4062726)
Affinity DataEC50:  5.60nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as increase in cAMP stimulation measured after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Jiangxi University Of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50240381(CHEMBL4078851)
Affinity DataEC50:  53nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as increase in cAMP stimulation measured after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Jiangxi University Of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50240395(CHEMBL4071750)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as increase in cAMP stimulation measured after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Jiangxi University Of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50240396(CHEMBL4086187)
Affinity DataEC50:  315nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as increase in cAMP stimulation measured after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Jiangxi University Of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50240390(CHEMBL4088637)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as increase in cAMP stimulation measured after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Jiangxi University Of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50240378(CHEMBL4067982)
Affinity DataEC50:  5.60nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as increase in cAMP stimulation measured after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed