TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Jiangxi University Of Traditional Chinese Medicine
Curated by ChEMBL
Jiangxi University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataEC50: 78nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as increase in cAMP stimulation measured after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Jiangxi University Of Traditional Chinese Medicine
Curated by ChEMBL
Jiangxi University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as increase in cAMP stimulation measured after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Jiangxi University Of Traditional Chinese Medicine
Curated by ChEMBL
Jiangxi University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataEC50: 236nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as increase in cAMP stimulation measured after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Jiangxi University Of Traditional Chinese Medicine
Curated by ChEMBL
Jiangxi University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataEC50: 4.90nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as increase in cAMP stimulation measured after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Jiangxi University Of Traditional Chinese Medicine
Curated by ChEMBL
Jiangxi University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as increase in cAMP stimulation measured after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Jiangxi University Of Traditional Chinese Medicine
Curated by ChEMBL
Jiangxi University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataEC50: 1.20nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as increase in cAMP stimulation measured after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Jiangxi University Of Traditional Chinese Medicine
Curated by ChEMBL
Jiangxi University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataEC50: 5.30nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as increase in cAMP stimulation measured after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Jiangxi University Of Traditional Chinese Medicine
Curated by ChEMBL
Jiangxi University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataEC50: 1.80nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as increase in cAMP stimulation measured after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Jiangxi University Of Traditional Chinese Medicine
Curated by ChEMBL
Jiangxi University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataEC50: 2.20E+3nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as increase in cAMP stimulation measured after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Jiangxi University Of Traditional Chinese Medicine
Curated by ChEMBL
Jiangxi University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataEC50: 110nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as increase in cAMP stimulation measured after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Jiangxi University Of Traditional Chinese Medicine
Curated by ChEMBL
Jiangxi University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as increase in cAMP stimulation measured after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Jiangxi University Of Traditional Chinese Medicine
Curated by ChEMBL
Jiangxi University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataEC50: 48nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as increase in cAMP stimulation measured after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Jiangxi University Of Traditional Chinese Medicine
Curated by ChEMBL
Jiangxi University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as increase in cAMP stimulation measured after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Jiangxi University Of Traditional Chinese Medicine
Curated by ChEMBL
Jiangxi University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataEC50: 3.10nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as increase in cAMP stimulation measured after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Jiangxi University Of Traditional Chinese Medicine
Curated by ChEMBL
Jiangxi University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataEC50: 6.40nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as increase in cAMP stimulation measured after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Jiangxi University Of Traditional Chinese Medicine
Curated by ChEMBL
Jiangxi University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataEC50: 5.60nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as increase in cAMP stimulation measured after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Jiangxi University Of Traditional Chinese Medicine
Curated by ChEMBL
Jiangxi University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataEC50: 53nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as increase in cAMP stimulation measured after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Jiangxi University Of Traditional Chinese Medicine
Curated by ChEMBL
Jiangxi University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as increase in cAMP stimulation measured after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Jiangxi University Of Traditional Chinese Medicine
Curated by ChEMBL
Jiangxi University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataEC50: 315nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as increase in cAMP stimulation measured after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Jiangxi University Of Traditional Chinese Medicine
Curated by ChEMBL
Jiangxi University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as increase in cAMP stimulation measured after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Jiangxi University Of Traditional Chinese Medicine
Curated by ChEMBL
Jiangxi University Of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataEC50: 5.60nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as increase in cAMP stimulation measured after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair