Compile Data Set for Download or QSAR
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Found 10 Enz. Inhib. hit(s) with all data for entry = 50020446
TargetTranscription factor Jun(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50213931(CHEMBL250854 | tylophorinidine)
Affinity DataIC50:  65nMAssay Description:Inhibition of AP1-mediated gene transcription in HepG2 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription factor Jun(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50213932(CHEMBL250474 | [(R)-(+)-deoxytylophorinidine)
Affinity DataIC50:  68nMAssay Description:Inhibition of AP1-mediated gene transcription in HepG2 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription factor Jun(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50213934(CHEMBL398325 | tylophorinine)
Affinity DataIC50:  110nMAssay Description:Inhibition of AP1-mediated gene transcription in HepG2 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription factor Jun(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50213935((12aS,13R)-2,3,6,7-tetramethoxy-9,10,11,12,12a,13-...)
Affinity DataIC50: >300nMAssay Description:Inhibition of AP1-mediated gene transcription in HepG2 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription factor Jun(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50213936((S)-2,3,6,7-tetramethoxy-8b,9,10,11,12,12a-hexahyd...)
Affinity DataIC50: >300nMAssay Description:Inhibition of AP1-mediated gene transcription in HepG2 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription factor Jun(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50213937((12aS,13S)-2,6,7-trimethoxy-9,10,11,12,12a,13-hexa...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of AP1-mediated gene transcription in HepG2 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription factor Jun(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50213933((12aS,13S)-2,3,6,7-tetramethoxy-9,10,11,12,12a,13-...)
Affinity DataIC50:  1.07E+3nMAssay Description:Inhibition of AP1-mediated gene transcription in HepG2 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription factor Jun(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50213930(6,7-Dimethoxy-12a-methyl-9,10,11,12,12a,13-hexahyd...)
Affinity DataIC50: >3.00E+3nMAssay Description:Inhibition of AP1-mediated gene transcription in HepG2 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription factor Jun(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50213929(CHEMBL401479 | tylophoridicine F)
Affinity DataIC50: >3.00E+3nMAssay Description:Inhibition of AP1-mediated gene transcription in HepG2 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription factor Jun(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50213938(CHEMBL249029 | tylophoridicine C)
Affinity DataIC50: >3.00E+3nMAssay Description:Inhibition of AP1-mediated gene transcription in HepG2 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed