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Found 23 Enz. Inhib. hit(s) with all data for entry = 50048413
TargetHistamine H3 receptor(Rattus norvegicus (rat))TBA
LigandPNGBDBM50214615(CHEBI:64177 | Clobenpropit)
Affinity DataKi:  0.158nMAssay Description:Binding affinity against H3 receptor in rat cerebral cortex membranes was evaluated using [3H]N-methyl-histamine as radioligandMore data for this Ligand-Target Pair
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TargetHistamine H3 receptor(Rattus norvegicus (rat))TBA
LigandPNGBDBM22914(CHEMBL260374 | N-cyclohexyl-4-(1H-imidazol-5-yl)pi...)
Affinity DataKi:  2nMAssay Description:Binding affinity against H3 receptor in rat cerebral cortex membranes was evaluated using [3H]N-methyl-histamine as radioligandMore data for this Ligand-Target Pair
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TargetHistamine H3 receptor(Rattus norvegicus (rat))TBA
LigandPNGBDBM50214616(CHEMBL168960)
Affinity DataKi:  3.20nMAssay Description:Binding affinity against H3 receptor in rat cerebral cortex membranes was evaluated using [3H]N-methyl-histamine as radioligandMore data for this Ligand-Target Pair
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TargetHistamine H3 receptor(Rattus norvegicus (rat))TBA
LigandPNGBDBM50214519(CHEMBL169994)
Affinity DataKi:  6.30nMAssay Description:Binding affinity against H3 receptor in rat cerebral cortex membranes was evaluated using [3H]N-methyl-histamine as radioligandMore data for this Ligand-Target Pair
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TargetHistamine H3 receptor(Rattus norvegicus (rat))TBA
LigandPNGBDBM50070213(3-(4-Chloro-benzyl)-5-[2-(1H-imidazol-4-yl)-ethyl]...)
Affinity DataKi:  6.30nMAssay Description:Binding affinity against H3 receptor in rat cerebral cortex membranes was evaluated using [3H]N-methyl-histamine as radioligandMore data for this Ligand-Target Pair
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TargetHistamine H3 receptor(Rattus norvegicus (rat))TBA
LigandPNGBDBM50214619(CHEMBL169426)
Affinity DataKi:  7.90nMAssay Description:Binding affinity against H3 receptor in rat cerebral cortex membranes was evaluated using [3H]N-methyl-histamine as radioligandMore data for this Ligand-Target Pair
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TargetHistamine H3 receptor(Rattus norvegicus (rat))TBA
LigandPNGBDBM50214524(CHEMBL169348)
Affinity DataKi:  10nMAssay Description:Binding affinity against H3 receptor in rat cerebral cortex membranes was evaluated using [3H]N-methyl-histamine as radioligandMore data for this Ligand-Target Pair
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TargetHistamine H3 receptor(Rattus norvegicus (rat))TBA
LigandPNGBDBM50214614(CHEMBL423445)
Affinity DataKi:  13nMAssay Description:Binding affinity against H3 receptor in rat cerebral cortex membranes was evaluated using [3H]N-methyl-histamine as radioligandMore data for this Ligand-Target Pair
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TargetHistamine H3 receptor(Rattus norvegicus (rat))TBA
LigandPNGBDBM50214620(CHEMBL353939)
Affinity DataKi:  20nMAssay Description:Binding affinity against H3 receptor in rat cerebral cortex membranes was evaluated using [3H]N-methyl-histamine as radioligandMore data for this Ligand-Target Pair
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TargetHistamine H3 receptor(Rattus norvegicus (rat))TBA
LigandPNGBDBM50214617(CHEMBL168196)
Affinity DataKi:  20nMAssay Description:Binding affinity against H3 receptor in rat cerebral cortex membranes was evaluated using [3H]N-methyl-histamine as radioligandMore data for this Ligand-Target Pair
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TargetHistamine H3 receptor(Rattus norvegicus (rat))TBA
LigandPNGBDBM50214623(CHEMBL354348)
Affinity DataKi:  25nMAssay Description:Binding affinity against H3 receptor in rat cerebral cortex membranes was evaluated using [3H]N-methyl-histamine as radioligandMore data for this Ligand-Target Pair
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TargetHistamine H3 receptor(Rattus norvegicus (rat))TBA
LigandPNGBDBM50409217(CHEMBL45056)
Affinity DataKi:  25nMAssay Description:Binding affinity against H3 receptor in rat cerebral cortex membranes was evaluated using [3H]N-methyl-histamine as radioligandMore data for this Ligand-Target Pair
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TargetHistamine H3 receptor(Rattus norvegicus (rat))TBA
LigandPNGBDBM50214622(CHEMBL166603)
Affinity DataKi:  25nMAssay Description:Binding affinity against H3 receptor in rat cerebral cortex membranes was evaluated using [3H]N-methyl-histamine as radioligandMore data for this Ligand-Target Pair
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TargetHistamine H3 receptor(Rattus norvegicus (rat))TBA
LigandPNGBDBM50214626(CHEMBL424010)
Affinity DataKi:  40nMAssay Description:Binding affinity against H3 receptor in rat cerebral cortex membranes was evaluated using [3H]N-methyl-histamine as radioligandMore data for this Ligand-Target Pair
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TargetHistamine H3 receptor(Rattus norvegicus (rat))TBA
LigandPNGBDBM50214526(CHEMBL168973)
Affinity DataKi:  63nMAssay Description:Binding affinity against H3 receptor in rat cerebral cortex membranes was evaluated using [3H]N-methyl-histamine as radioligandMore data for this Ligand-Target Pair
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TargetHistamine H3 receptor(Rattus norvegicus (rat))TBA
LigandPNGBDBM50214625(CHEMBL354711)
Affinity DataKi:  100nMAssay Description:Binding affinity against H3 receptor in rat cerebral cortex membranes was evaluated using [3H]N-methyl-histamine as radioligandMore data for this Ligand-Target Pair
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TargetHistamine H3 receptor(Rattus norvegicus (rat))TBA
LigandPNGBDBM50214613(CHEMBL166761)
Affinity DataKi:  126nMAssay Description:Binding affinity against H3 receptor in rat cerebral cortex membranes was evaluated using [3H]N-methyl-histamine as radioligandMore data for this Ligand-Target Pair
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TargetHistamine H3 receptor(Rattus norvegicus (rat))TBA
LigandPNGBDBM50214621(CHEMBL169026)
Affinity DataKi:  200nMAssay Description:Binding affinity against H3 receptor in rat cerebral cortex membranes was evaluated using [3H]N-methyl-histamine as radioligandMore data for this Ligand-Target Pair
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TargetHistamine H3 receptor(Rattus norvegicus (rat))TBA
LigandPNGBDBM50214618(CHEMBL166802)
Affinity DataKi:  200nMAssay Description:Binding affinity against H3 receptor in rat cerebral cortex membranes was evaluated using [3H]N-methyl-histamine as radioligandMore data for this Ligand-Target Pair
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TargetHistamine H3 receptor(Rattus norvegicus (rat))TBA
LigandPNGBDBM50214525(CHEMBL353915)
Affinity DataKi:  251nMAssay Description:Binding affinity against H3 receptor in rat cerebral cortex membranes was evaluated using [3H]N-methyl-histamine as radioligandMore data for this Ligand-Target Pair
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TargetHistamine H3 receptor(Rattus norvegicus (rat))TBA
LigandPNGBDBM50214624(CHEMBL352869)
Affinity DataKi:  316nMAssay Description:Binding affinity against H3 receptor in rat cerebral cortex membranes was evaluated using [3H]N-methyl-histamine as radioligandMore data for this Ligand-Target Pair
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TargetHistamine H3 receptor(Rattus norvegicus (rat))TBA
LigandPNGBDBM50214609(CHEMBL165537)
Affinity DataKi:  1.26E+3nMAssay Description:Binding affinity against H3 receptor in rat cerebral cortex membranes was evaluated using [3H]N-methyl-histamine as radioligandMore data for this Ligand-Target Pair
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TargetHistamine H3 receptor(Rattus norvegicus (rat))TBA
LigandPNGBDBM50214518(CHEMBL168889)
Affinity DataKi:  2.51E+3nMAssay Description:Binding affinity against H3 receptor in rat cerebral cortex membranes was evaluated using [3H]N-methyl-histamine as radioligandMore data for this Ligand-Target Pair
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