TargetProstaglandin E2 receptor EP3 subtype(Homo sapiens (Human))
Merck Frosst Canada
Curated by ChEMBL
Merck Frosst Canada
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Antagonistic activity at Prostanoid EP3 receptor in human was determinedMore data for this Ligand-Target Pair
TargetProstaglandin E2 receptor EP3 subtype(Homo sapiens (Human))
Merck Frosst Canada
Curated by ChEMBL
Merck Frosst Canada
Curated by ChEMBL
Affinity DataKi: 32nMAssay Description:Antagonistic activity at Prostanoid EP3 receptor in human was determinedMore data for this Ligand-Target Pair
TargetProstaglandin E2 receptor EP3 subtype(Homo sapiens (Human))
Merck Frosst Canada
Curated by ChEMBL
Merck Frosst Canada
Curated by ChEMBL
Affinity DataKi: 80nMAssay Description:Antagonistic activity at Prostanoid EP3 receptor in human was determinedMore data for this Ligand-Target Pair
TargetProstaglandin E2 receptor EP3 subtype(Homo sapiens (Human))
Merck Frosst Canada
Curated by ChEMBL
Merck Frosst Canada
Curated by ChEMBL
Affinity DataKi: 110nMAssay Description:Antagonistic activity at Prostanoid EP3 receptor in human was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 520nMAssay Description:Antagonistic activity at Thromboxane A2 receptor in human was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 530nMAssay Description:Antagonistic activity at Prostanoid DP receptor in human was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 900nMAssay Description:Antagonistic activity at Thromboxane A2 receptor in human was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 2.40E+3nMAssay Description:Antagonistic activity at Prostanoid DP receptor in human was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 2.50E+3nMAssay Description:Antagonistic activity at Prostanoid DP receptor in human was determinedMore data for this Ligand-Target Pair
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Merck Frosst Canada
Curated by ChEMBL
Merck Frosst Canada
Curated by ChEMBL
Affinity DataKi: 3.10E+3nMAssay Description:Antagonistic activity at Prostanoid EP4 receptor in human was determinedMore data for this Ligand-Target Pair
TargetProstaglandin E2 receptor EP2 subtype(Homo sapiens (Human))
Merck Frosst Canada
Curated by ChEMBL
Merck Frosst Canada
Curated by ChEMBL
Affinity DataKi: 4.10E+3nMAssay Description:Antagonistic activity at Prostanoid EP2 receptor in human was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 4.10E+3nMAssay Description:Antagonistic activity at Prostanoid DP receptor in human was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 4.60E+3nMAssay Description:Antagonistic activity at Thromboxane A2 receptor in human was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+4nMAssay Description:Antagonistic activity at Thromboxane A2 receptor in human was determinedMore data for this Ligand-Target Pair
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Merck Frosst Canada
Curated by ChEMBL
Merck Frosst Canada
Curated by ChEMBL
Affinity DataKi: 1.00E+4nMAssay Description:Antagonistic activity at Prostanoid EP4 receptor in human was determinedMore data for this Ligand-Target Pair
TargetProstaglandin E2 receptor EP2 subtype(Homo sapiens (Human))
Merck Frosst Canada
Curated by ChEMBL
Merck Frosst Canada
Curated by ChEMBL
Affinity DataKi: 1.20E+4nMAssay Description:Antagonistic activity at Prostanoid EP2 receptor in human was determinedMore data for this Ligand-Target Pair
TargetProstaglandin E2 receptor EP2 subtype(Homo sapiens (Human))
Merck Frosst Canada
Curated by ChEMBL
Merck Frosst Canada
Curated by ChEMBL
Affinity DataKi: 1.30E+4nMAssay Description:Antagonistic activity at Prostanoid EP2 receptor in human was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 3.10E+4nMAssay Description:Antagonistic activity at Prostanoid IP receptor in human was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 3.70E+4nMAssay Description:Antagonistic activity at Prostanoid IP receptor in human was determinedMore data for this Ligand-Target Pair
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Merck Frosst Canada
Curated by ChEMBL
Merck Frosst Canada
Curated by ChEMBL
Affinity DataKi: >4.00E+4nMAssay Description:Antagonistic activity at Prostanoid EP4 receptor in human was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 4.10E+4nMAssay Description:Antagonistic activity at Prostanoid FP receptor in human was determinedMore data for this Ligand-Target Pair
TargetProstaglandin E2 receptor EP2 subtype(Homo sapiens (Human))
Merck Frosst Canada
Curated by ChEMBL
Merck Frosst Canada
Curated by ChEMBL
Affinity DataKi: 4.30E+4nMAssay Description:Antagonistic activity at Prostanoid EP2 receptor in human was determinedMore data for this Ligand-Target Pair
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Merck Frosst Canada
Curated by ChEMBL
Merck Frosst Canada
Curated by ChEMBL
Affinity DataKi: >5.00E+4nMAssay Description:Antagonistic activity at Prostanoid EP4 receptor in human was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 6.30E+4nMAssay Description:Antagonistic activity at Prostanoid FP receptor in human was determinedMore data for this Ligand-Target Pair
TargetProstaglandin E2 receptor EP1 subtype(Homo sapiens (Human))
Merck Frosst Canada
Curated by ChEMBL
Merck Frosst Canada
Curated by ChEMBL
Affinity DataKi: 6.30E+4nMAssay Description:Antagonistic activity at Prostanoid EP1 receptor in human was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 6.90E+4nMAssay Description:Antagonistic activity at Prostanoid FP receptor in human was determinedMore data for this Ligand-Target Pair
Affinity DataKi: >7.60E+4nMAssay Description:Antagonistic activity at Prostanoid IP receptor in human was determinedMore data for this Ligand-Target Pair
Affinity DataKi: >8.30E+4nMAssay Description:Antagonistic activity at Prostanoid FP receptor in human was determinedMore data for this Ligand-Target Pair
TargetProstaglandin E2 receptor EP1 subtype(Homo sapiens (Human))
Merck Frosst Canada
Curated by ChEMBL
Merck Frosst Canada
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Antagonistic activity at Prostanoid EP1 receptor in human was determinedMore data for this Ligand-Target Pair
TargetProstaglandin E2 receptor EP1 subtype(Homo sapiens (Human))
Merck Frosst Canada
Curated by ChEMBL
Merck Frosst Canada
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Antagonistic activity at Prostanoid EP1 receptor in human was determinedMore data for this Ligand-Target Pair
TargetProstaglandin E2 receptor EP1 subtype(Homo sapiens (Human))
Merck Frosst Canada
Curated by ChEMBL
Merck Frosst Canada
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Antagonistic activity at Prostanoid EP1 receptor in human was determinedMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Antagonistic activity at Prostanoid IP receptor in human was determinedMore data for this Ligand-Target Pair