Compile Data Set for Download or QSAR
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Found 7 Enz. Inhib. hit(s) with all data for entry = 50000798
TargetB-cell lymphoma 6 protein(Homo sapiens)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50260529(CHEMBL4077626)
Affinity DataIC50:  1nMAssay Description:Inhibition of C-terminal biotin-labelled BCoR (Arg498 to 514Pro residues) binding to recombinant FLAG-tagged BCL6 BTB (5 to 129 residues) (unknown or...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB-cell lymphoma 6 protein(Homo sapiens)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50260534(CHEMBL4066375)
Affinity DataIC50:  2.12E+5nMAssay Description:Inhibition of C-terminal biotin-labelled BCoR/wild-type BCL6 BTB domain (unknown origin) protein-protein interaction by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB-cell lymphoma 6 protein(Homo sapiens)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50260529(CHEMBL4077626)
Affinity DataKd:  0.570nMAssay Description:Inhibition of recombinant human BCoR (112 to 753 residues) protein interaction with recombinant GAL4-fused BCL6 (5 to 129 residues) expressed in HEK2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB-cell lymphoma 6 protein(Homo sapiens)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50260534(CHEMBL4066375)
Affinity DataKd:  1.29E+5nMAssay Description:Inhibition of recombinant human BCoR (112 to 753 residues) protein interaction with recombinant GAL4-fused BCL6 (5 to 129 residues) expressed in HEK2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB-cell lymphoma 6 protein(Homo sapiens)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50260528(CHEMBL4063725)
Affinity DataKd:  5.00E+3nMAssay Description:Binding affinity to wild-type avi-tagged BCL6 BTB domain (unknown origin) by SPR analysisMore data for this Ligand-Target Pair
TargetB-cell lymphoma 6 protein(Homo sapiens)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50260527(CHEMBL4096591)
Affinity DataKd:  2.40E+4nMAssay Description:Binding affinity to wild-type avi-tagged BCL6 BTB domain (unknown origin) by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB-cell lymphoma 6 protein(Homo sapiens)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50239395(CHEMBL4061302)
Affinity DataKd:  7.00E+3nMAssay Description:Binding affinity to recombinant RED-NHS labelled BCL6 BTB domain (1 to 129 residues) (unknown origin) after 10 mins by microscale thermophoresis meth...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed