Compile Data Set for Download or QSAR
maximum 50k data
Found 98 Enz. Inhib. hit(s) with all data for entry = 50049077
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50200526(CHEMBL1234118)
Affinity DataKi:  50nMAssay Description:Displacement of [3H]kainate from human GluK1 expressed in HEK293 cell membranes after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 1(RAT)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50234094(CHEMBL4089715)
Affinity DataKi:  2.27E+3nMAssay Description:Displacement of [3H]-(2S,4R)-4-Methylglutamic acid from rat eGFP-fused GluK1 receptor LBD expressed in HEK293T/17 cells by liquid scintillation count...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50234102(CHEMBL4090052)
Affinity DataKi:  3.50E+3nMAssay Description:Displacement of [3H]NF608 from eGFP-fused recombinant rat full length GluK1 receptor expressed in HEK293T/17 cells by liquid scintillation counting m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50234102(CHEMBL4090052)
Affinity DataKi:  3.51E+3nMAssay Description:Displacement of [3H]NF608 from eGFP-fused recombinant rat full length GluK1 receptor expressed in HEK293T/17 cells by liquid scintillation counting m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50234094(CHEMBL4089715)
Affinity DataKi:  3.98E+3nMAssay Description:Displacement of [3H]NF608 from eGFP-fused recombinant rat full length GluK1 receptor expressed in HEK293T/17 cells by liquid scintillation counting m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50234094(CHEMBL4089715)
Affinity DataKi:  4.00E+3nMAssay Description:Displacement of [3H]NF608 from eGFP-fused recombinant rat full length GluK1 receptor expressed in HEK293T/17 cells by liquid scintillation counting m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50234109(CHEMBL4067910)
Affinity DataKi:  4.47E+3nMAssay Description:Displacement of [3H]NF608 from eGFP-fused recombinant rat full length GluK1 receptor expressed in HEK293T/17 cells by liquid scintillation counting m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50234109(CHEMBL4067910)
Affinity DataKi:  4.50E+3nMAssay Description:Displacement of [3H]NF608 from eGFP-fused recombinant rat full length GluK1 receptor expressed in HEK293T/17 cells by liquid scintillation counting m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50234110(CHEMBL4090961)
Affinity DataKi:  4.68E+3nMAssay Description:Displacement of [3H]NF608 from eGFP-fused recombinant rat full length GluK1 receptor expressed in HEK293T/17 cells by liquid scintillation counting m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50234110(CHEMBL4090961)
Affinity DataKi:  4.70E+3nMAssay Description:Displacement of [3H]NF608 from eGFP-fused recombinant rat full length GluK1 receptor expressed in HEK293T/17 cells by liquid scintillation counting m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50234111(CHEMBL4063058)
Affinity DataKi:  5.37E+3nMAssay Description:Displacement of [3H]NF608 from eGFP-fused recombinant rat full length GluK1 receptor expressed in HEK293T/17 cells by liquid scintillation counting m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50234111(CHEMBL4063058)
Affinity DataKi:  5.40E+3nMAssay Description:Displacement of [3H]NF608 from eGFP-fused recombinant rat full length GluK1 receptor expressed in HEK293T/17 cells by liquid scintillation counting m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50234096(CHEMBL4084004)
Affinity DataKi:  7.94E+3nMAssay Description:Displacement of [3H]NF608 from eGFP-fused recombinant rat full length GluK1 receptor expressed in HEK293T/17 cells by liquid scintillation counting m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50234096(CHEMBL4084004)
Affinity DataKi:  8.40E+3nMAssay Description:Displacement of [3H]NF608 from eGFP-fused recombinant rat full length GluK1 receptor expressed in HEK293T/17 cells by liquid scintillation counting m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 3(Homo sapiens (Human))
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50200526(CHEMBL1234118)
Affinity DataKi:  8.90E+3nMAssay Description:Inhibition of GluK3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50234096(CHEMBL4084004)
Affinity DataKi:  2.19E+4nMAssay Description:Displacement of [3H]kainic acid from eGFP-fused recombinant rat full length GluK3 receptor expressed in HEK293T/17 cells by liquid scintillation coun...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50234096(CHEMBL4084004)
Affinity DataKi:  2.20E+4nMAssay Description:Displacement of [3H]kainic acid from eGFP-fused recombinant rat full length GluK3 receptor expressed in HEK293T/17 cells by liquid scintillation coun...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50234104(CHEMBL4105498)
Affinity DataKi:  2.34E+4nMAssay Description:Displacement of [3H]NF608 from eGFP-fused recombinant rat full length GluK1 receptor expressed in HEK293T/17 cells by liquid scintillation counting m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50234100(CHEMBL4097766)
Affinity DataKi:  2.40E+4nMAssay Description:Displacement of [3H]NF608 from eGFP-fused recombinant rat full length GluK1 receptor expressed in HEK293T/17 cells by liquid scintillation counting m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50234104(CHEMBL4105498)
Affinity DataKi:  2.40E+4nMAssay Description:Displacement of [3H]NF608 from eGFP-fused recombinant rat full length GluK1 receptor expressed in HEK293T/17 cells by liquid scintillation counting m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50234100(CHEMBL4097766)
Affinity DataKi:  2.40E+4nMAssay Description:Displacement of [3H]NF608 from eGFP-fused recombinant rat full length GluK1 receptor expressed in HEK293T/17 cells by liquid scintillation counting m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50234110(CHEMBL4090961)
Affinity DataKi:  2.95E+4nMAssay Description:Displacement of [3H]kainic acid from eGFP-fused recombinant rat full length GluK3 receptor expressed in HEK293T/17 cells by liquid scintillation coun...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50234110(CHEMBL4090961)
Affinity DataKi:  3.00E+4nMAssay Description:Displacement of [3H]kainic acid from eGFP-fused recombinant rat full length GluK3 receptor expressed in HEK293T/17 cells by liquid scintillation coun...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50234092(CHEMBL4073637)
Affinity DataKi:  3.31E+4nMAssay Description:Displacement of [3H]NF608 from eGFP-fused recombinant rat full length GluK1 receptor expressed in HEK293T/17 cells by liquid scintillation counting m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50234092(CHEMBL4073637)
Affinity DataKi:  3.60E+4nMAssay Description:Displacement of [3H]NF608 from eGFP-fused recombinant rat full length GluK1 receptor expressed in HEK293T/17 cells by liquid scintillation counting m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50234101(CHEMBL4068976)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]kainic acid from eGFP-fused recombinant rat full length GluK3 receptor expressed in HEK293T/17 cells by liquid scintillation coun...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50234098(CHEMBL4065054)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]kainic acid from eGFP-fused recombinant rat full length GluK3 receptor expressed in HEK293T/17 cells by liquid scintillation coun...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50234091(CHEMBL4084974)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]kainic acid from eGFP-fused recombinant rat full length GluK3 receptor expressed in HEK293T/17 cells by liquid scintillation coun...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50234093(CHEMBL4068592)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]NF608 from eGFP-fused recombinant rat full length GluK1 receptor expressed in HEK293T/17 cells by liquid scintillation counting m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50234095(CHEMBL4100460)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]NF608 from eGFP-fused recombinant rat full length GluK1 receptor expressed in HEK293T/17 cells by liquid scintillation counting m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50234097(CHEMBL4102927)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]NF608 from eGFP-fused recombinant rat full length GluK1 receptor expressed in HEK293T/17 cells by liquid scintillation counting m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50234091(CHEMBL4084974)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]NF608 from eGFP-fused recombinant rat full length GluK1 receptor expressed in HEK293T/17 cells by liquid scintillation counting m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50234098(CHEMBL4065054)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]NF608 from eGFP-fused recombinant rat full length GluK1 receptor expressed in HEK293T/17 cells by liquid scintillation counting m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50234099(CHEMBL4087475)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]NF608 from eGFP-fused recombinant rat full length GluK1 receptor expressed in HEK293T/17 cells by liquid scintillation counting m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50234101(CHEMBL4068976)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]NF608 from eGFP-fused recombinant rat full length GluK1 receptor expressed in HEK293T/17 cells by liquid scintillation counting m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50234107(CHEMBL4087617)
Affinity DataKi:  1.00E+5nMAssay Description:Displacement of [3H]NF608 from eGFP-fused recombinant rat full length GluK1 receptor expressed in HEK293T/17 cells by liquid scintillation counting m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50234108(CHEMBL4062289)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]kainic acid from eGFP-fused recombinant rat full length GluK2 receptor expressed in HEK293T/17 cells by liquid scintillation coun...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50234099(CHEMBL4087475)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]kainic acid from eGFP-fused recombinant rat full length GluK2 receptor expressed in HEK293T/17 cells by liquid scintillation coun...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50234105(CHEMBL4095318)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]kainic acid from eGFP-fused recombinant rat full length GluK3 receptor expressed in HEK293T/17 cells by liquid scintillation coun...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50234092(CHEMBL4073637)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]kainic acid from eGFP-fused recombinant rat full length GluK2 receptor expressed in HEK293T/17 cells by liquid scintillation coun...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50234097(CHEMBL4102927)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]kainic acid from eGFP-fused recombinant rat full length GluK3 receptor expressed in HEK293T/17 cells by liquid scintillation coun...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Rattus norvegicus)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50234104(CHEMBL4105498)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of (RS)-[3H]AMPA from eGFP-fused recombinant rat full length GluA2 receptor expressed in HEK293T/17 cells by liquid scintillation counti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50234109(CHEMBL4067910)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]kainic acid from eGFP-fused recombinant rat full length GluK2 receptor expressed in HEK293T/17 cells by liquid scintillation coun...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50234104(CHEMBL4105498)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]kainic acid from eGFP-fused recombinant rat full length GluK2 receptor expressed in HEK293T/17 cells by liquid scintillation coun...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50234091(CHEMBL4084974)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]kainic acid from eGFP-fused recombinant rat full length GluK2 receptor expressed in HEK293T/17 cells by liquid scintillation coun...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Rattus norvegicus)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50234102(CHEMBL4090052)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of (RS)-[3H]AMPA from eGFP-fused recombinant rat full length GluA2 receptor expressed in HEK293T/17 cells by liquid scintillation counti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50234095(CHEMBL4100460)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]kainic acid from eGFP-fused recombinant rat full length GluK3 receptor expressed in HEK293T/17 cells by liquid scintillation coun...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Rattus norvegicus)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50234110(CHEMBL4090961)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of (RS)-[3H]AMPA from eGFP-fused recombinant rat full length GluA2 receptor expressed in HEK293T/17 cells by liquid scintillation counti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Rattus norvegicus)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50234101(CHEMBL4068976)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of (RS)-[3H]AMPA from eGFP-fused recombinant rat full length GluA2 receptor expressed in HEK293T/17 cells by liquid scintillation counti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
Mcgill University

Curated by ChEMBL
LigandPNGBDBM50234106(CHEMBL4092735)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]kainic acid from eGFP-fused recombinant rat full length GluK2 receptor expressed in HEK293T/17 cells by liquid scintillation coun...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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