Compile Data Set for Download or QSAR
maximum 50k data
Found 134 Enz. Inhib. hit(s) with all data for entry = 50014564
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Lycera

Curated by ChEMBL
LigandPNGBDBM50280398(CHEMBL4162171)
Affinity DataEC50:  223nMAssay Description:Agonist activity at human His-tagged RORgamma-LBD expressed in Sf9 cells assessed as inhibition of N-terminal biotinylated co-activator SRC1 recruitm...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Lycera

Curated by ChEMBL
LigandPNGBDBM50577411(CHEMBL4865225)
Affinity DataEC50:  105nMAssay Description:Agonist activity at human His-tagged RORgamma-LBD expressed in Sf9 cells assessed as inhibition of N-terminal biotinylated co-activator SRC1 recruitm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Lycera

Curated by ChEMBL
LigandPNGBDBM50577412(CHEMBL4848784)
Affinity DataEC50:  195nMAssay Description:Agonist activity at human His-tagged RORgamma-LBD expressed in Sf9 cells assessed as inhibition of N-terminal biotinylated co-activator SRC1 recruitm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Lycera

Curated by ChEMBL
LigandPNGBDBM50577413(CHEMBL4874944)
Affinity DataEC50:  85nMAssay Description:Agonist activity at human His-tagged RORgamma-LBD expressed in Sf9 cells assessed as inhibition of N-terminal biotinylated co-activator SRC1 recruitm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Lycera

Curated by ChEMBL
LigandPNGBDBM50577414(CHEMBL4873783)
Affinity DataEC50:  269nMAssay Description:Agonist activity at human His-tagged RORgamma-LBD expressed in Sf9 cells assessed as inhibition of N-terminal biotinylated co-activator SRC1 recruitm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Lycera

Curated by ChEMBL
LigandPNGBDBM50577415(CHEMBL4868679)
Affinity DataEC50:  36nMAssay Description:Agonist activity at human His-tagged RORgamma-LBD expressed in Sf9 cells assessed as inhibition of N-terminal biotinylated co-activator SRC1 recruitm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Lycera

Curated by ChEMBL
LigandPNGBDBM50280399(CHEMBL4172843)
Affinity DataEC50:  68nMAssay Description:Agonist activity at human His-tagged RORgamma-LBD expressed in Sf9 cells assessed as inhibition of N-terminal biotinylated co-activator SRC1 recruitm...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Lycera

Curated by ChEMBL
LigandPNGBDBM50577416(CHEMBL4878616)
Affinity DataEC50:  95nMAssay Description:Agonist activity at human His-tagged RORgamma-LBD expressed in Sf9 cells assessed as inhibition of N-terminal biotinylated co-activator SRC1 recruitm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Lycera

Curated by ChEMBL
LigandPNGBDBM50577417(CHEMBL4866161)
Affinity DataEC50:  112nMAssay Description:Agonist activity at human His-tagged RORgamma-LBD expressed in Sf9 cells assessed as inhibition of N-terminal biotinylated co-activator SRC1 recruitm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Lycera

Curated by ChEMBL
LigandPNGBDBM50577418(CHEMBL4847760)
Affinity DataEC50:  108nMAssay Description:Agonist activity at human His-tagged RORgamma-LBD expressed in Sf9 cells assessed as inhibition of N-terminal biotinylated co-activator SRC1 recruitm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Lycera

Curated by ChEMBL
LigandPNGBDBM50577419(CHEMBL4879241)
Affinity DataEC50:  46nMAssay Description:Agonist activity at human His-tagged RORgamma-LBD expressed in Sf9 cells assessed as inhibition of N-terminal biotinylated co-activator SRC1 recruitm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Lycera

Curated by ChEMBL
LigandPNGBDBM50577420(CHEMBL4846685)
Affinity DataEC50:  435nMAssay Description:Agonist activity at human His-tagged RORgamma-LBD expressed in Sf9 cells assessed as inhibition of N-terminal biotinylated co-activator SRC1 recruitm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Lycera

Curated by ChEMBL
LigandPNGBDBM50577421(CHEMBL4868432)
Affinity DataEC50:  33nMAssay Description:Agonist activity at human His-tagged RORgamma-LBD expressed in Sf9 cells assessed as inhibition of N-terminal biotinylated co-activator SRC1 recruitm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Lycera

Curated by ChEMBL
LigandPNGBDBM50577422(CHEMBL4846389)
Affinity DataEC50:  342nMAssay Description:Agonist activity at human His-tagged RORgamma-LBD expressed in Sf9 cells assessed as inhibition of N-terminal biotinylated co-activator SRC1 recruitm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Lycera

Curated by ChEMBL
LigandPNGBDBM50577423(CHEMBL4865235)
Affinity DataEC50:  1.08E+3nMAssay Description:Agonist activity at human His-tagged RORgamma-LBD expressed in Sf9 cells assessed as inhibition of N-terminal biotinylated co-activator SRC1 recruitm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Lycera

Curated by ChEMBL
LigandPNGBDBM50577424(CHEMBL4874524)
Affinity DataEC50:  9nMAssay Description:Agonist activity at human His-tagged RORgamma-LBD expressed in Sf9 cells assessed as inhibition of N-terminal biotinylated co-activator SRC1 recruitm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Lycera

Curated by ChEMBL
LigandPNGBDBM50577425(CHEMBL4851214)
Affinity DataEC50:  3nMAssay Description:Agonist activity at human His-tagged RORgamma-LBD expressed in Sf9 cells assessed as inhibition of N-terminal biotinylated co-activator SRC1 recruitm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Lycera

Curated by ChEMBL
LigandPNGBDBM50577426(CHEMBL4861757)
Affinity DataEC50:  27nMAssay Description:Agonist activity at human His-tagged RORgamma-LBD expressed in Sf9 cells assessed as inhibition of N-terminal biotinylated co-activator SRC1 recruitm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Lycera

Curated by ChEMBL
LigandPNGBDBM50577427(CHEMBL4849989)
Affinity DataEC50:  6nMAssay Description:Agonist activity at human His-tagged RORgamma-LBD expressed in Sf9 cells assessed as inhibition of N-terminal biotinylated co-activator SRC1 recruitm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Lycera

Curated by ChEMBL
LigandPNGBDBM50577428(CHEMBL4860324)
Affinity DataEC50:  8nMAssay Description:Agonist activity at human His-tagged RORgamma-LBD expressed in Sf9 cells assessed as inhibition of N-terminal biotinylated co-activator SRC1 recruitm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Lycera

Curated by ChEMBL
LigandPNGBDBM50577429(CHEMBL4859796)
Affinity DataEC50:  10nMAssay Description:Agonist activity at human His-tagged RORgamma-LBD expressed in Sf9 cells assessed as inhibition of N-terminal biotinylated co-activator SRC1 recruitm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Lycera

Curated by ChEMBL
LigandPNGBDBM50577430(CHEMBL4869479)
Affinity DataEC50:  42nMAssay Description:Agonist activity at human His-tagged RORgamma-LBD expressed in Sf9 cells assessed as inhibition of N-terminal biotinylated co-activator SRC1 recruitm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Lycera

Curated by ChEMBL
LigandPNGBDBM50577431(CHEMBL4873257)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human His-tagged RORgamma-LBD expressed in Sf9 cells assessed as inhibition of N-terminal biotinylated co-activator SRC1 recruitm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Lycera

Curated by ChEMBL
LigandPNGBDBM50577432(CHEMBL4874647)
Affinity DataEC50:  262nMAssay Description:Agonist activity at human His-tagged RORgamma-LBD expressed in Sf9 cells assessed as inhibition of N-terminal biotinylated co-activator SRC1 recruitm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Lycera

Curated by ChEMBL
LigandPNGBDBM50577433(CHEMBL4861064)
Affinity DataEC50:  145nMAssay Description:Agonist activity at human His-tagged RORgamma-LBD expressed in Sf9 cells assessed as inhibition of N-terminal biotinylated co-activator SRC1 recruitm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Lycera

Curated by ChEMBL
LigandPNGBDBM50577434(CHEMBL4875312)
Affinity DataEC50:  22nMAssay Description:Agonist activity at human His-tagged RORgamma-LBD expressed in Sf9 cells assessed as inhibition of N-terminal biotinylated co-activator SRC1 recruitm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Lycera

Curated by ChEMBL
LigandPNGBDBM50577435(CHEMBL4864871)
Affinity DataEC50:  8nMAssay Description:Agonist activity at human His-tagged RORgamma-LBD expressed in Sf9 cells assessed as inhibition of N-terminal biotinylated co-activator SRC1 recruitm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Lycera

Curated by ChEMBL
LigandPNGBDBM50577436(CHEMBL4846130)
Affinity DataEC50:  14nMAssay Description:Agonist activity at human His-tagged RORgamma-LBD expressed in Sf9 cells assessed as inhibition of N-terminal biotinylated co-activator SRC1 recruitm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Lycera

Curated by ChEMBL
LigandPNGBDBM50577437(CHEMBL4862004)
Affinity DataEC50:  6nMAssay Description:Agonist activity at human His-tagged RORgamma-LBD expressed in Sf9 cells assessed as inhibition of N-terminal biotinylated co-activator SRC1 recruitm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Lycera

Curated by ChEMBL
LigandPNGBDBM50577438(CHEMBL4846510)
Affinity DataEC50:  24nMAssay Description:Agonist activity at human His-tagged RORgamma-LBD expressed in Sf9 cells assessed as inhibition of N-terminal biotinylated co-activator SRC1 recruitm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Lycera

Curated by ChEMBL
LigandPNGBDBM50577439(CHEMBL4859771)
Affinity DataEC50:  4nMAssay Description:Agonist activity at human His-tagged RORgamma-LBD expressed in Sf9 cells assessed as inhibition of N-terminal biotinylated co-activator SRC1 recruitm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Lycera

Curated by ChEMBL
LigandPNGBDBM50577440(CHEMBL4870074)
Affinity DataEC50:  3nMAssay Description:Agonist activity at human His-tagged RORgamma-LBD expressed in Sf9 cells assessed as inhibition of N-terminal biotinylated co-activator SRC1 recruitm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Lycera

Curated by ChEMBL
LigandPNGBDBM50577441(CHEMBL4865657)
Affinity DataEC50:  13nMAssay Description:Agonist activity at human His-tagged RORgamma-LBD expressed in Sf9 cells assessed as inhibition of N-terminal biotinylated co-activator SRC1 recruitm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Lycera

Curated by ChEMBL
LigandPNGBDBM50577442(CHEMBL4847229)
Affinity DataEC50:  10nMAssay Description:Agonist activity at human His-tagged RORgamma-LBD expressed in Sf9 cells assessed as inhibition of N-terminal biotinylated co-activator SRC1 recruitm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Lycera

Curated by ChEMBL
LigandPNGBDBM50515653(CHEMBL4472508)
Affinity DataEC50:  13nMAssay Description:Agonist activity at human His-tagged RORgamma-LBD expressed in Sf9 cells assessed as inhibition of N-terminal biotinylated co-activator SRC1 recruitm...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Lycera

Curated by ChEMBL
LigandPNGBDBM50577443(CHEMBL4854926)
Affinity DataEC50:  159nMAssay Description:Agonist activity at human His-tagged RORgamma-LBD expressed in Sf9 cells assessed as inhibition of N-terminal biotinylated co-activator SRC1 recruitm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Lycera

Curated by ChEMBL
LigandPNGBDBM50577444(CHEMBL4856642)
Affinity DataEC50:  6nMAssay Description:Agonist activity at human His-tagged RORgamma-LBD expressed in Sf9 cells assessed as inhibition of N-terminal biotinylated co-activator SRC1 recruitm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Lycera

Curated by ChEMBL
LigandPNGBDBM50577445(CHEMBL4846575)
Affinity DataEC50:  10nMAssay Description:Agonist activity at human His-tagged RORgamma-LBD expressed in Sf9 cells assessed as inhibition of N-terminal biotinylated co-activator SRC1 recruitm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Lycera

Curated by ChEMBL
LigandPNGBDBM50577446(CHEMBL4868437)
Affinity DataEC50:  5nMAssay Description:Agonist activity at human His-tagged RORgamma-LBD expressed in Sf9 cells assessed as inhibition of N-terminal biotinylated co-activator SRC1 recruitm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Lycera

Curated by ChEMBL
LigandPNGBDBM50577447(CHEMBL4869567)
Affinity DataEC50:  8nMAssay Description:Agonist activity at human His-tagged RORgamma-LBD expressed in Sf9 cells assessed as inhibition of N-terminal biotinylated co-activator SRC1 recruitm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Lycera

Curated by ChEMBL
LigandPNGBDBM50577448(CHEMBL4849995)
Affinity DataEC50:  24nMAssay Description:Agonist activity at human His-tagged RORgamma-LBD expressed in Sf9 cells assessed as inhibition of N-terminal biotinylated co-activator SRC1 recruitm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Lycera

Curated by ChEMBL
LigandPNGBDBM50577449(CHEMBL4875777)
Affinity DataEC50:  120nMAssay Description:Agonist activity at human His-tagged RORgamma-LBD expressed in Sf9 cells assessed as inhibition of N-terminal biotinylated co-activator SRC1 recruitm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Lycera

Curated by ChEMBL
LigandPNGBDBM50577450(CHEMBL4858971)
Affinity DataEC50:  13nMAssay Description:Agonist activity at human His-tagged RORgamma-LBD expressed in Sf9 cells assessed as inhibition of N-terminal biotinylated co-activator SRC1 recruitm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Lycera

Curated by ChEMBL
LigandPNGBDBM50515653(CHEMBL4472508)
Affinity DataEC50:  120nMAssay Description:Agonist activity at RORgamma in human whole blood assessed as increase in IL-17A productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Lycera

Curated by ChEMBL
LigandPNGBDBM50280398(CHEMBL4162171)
Affinity DataEC50:  324nMAssay Description:Agonist activity at human ROR-gamma LBD expressed in HEK293 cells assessed as transcriptional activity in presence of ursolic acid by Gal4-luciferase...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Lycera

Curated by ChEMBL
LigandPNGBDBM50577411(CHEMBL4865225)
Affinity DataEC50:  520nMAssay Description:Agonist activity at human ROR-gamma LBD expressed in HEK293 cells assessed as transcriptional activity in presence of ursolic acid by Gal4-luciferase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Lycera

Curated by ChEMBL
LigandPNGBDBM50577412(CHEMBL4848784)
Affinity DataEC50:  280nMAssay Description:Agonist activity at human ROR-gamma LBD expressed in HEK293 cells assessed as transcriptional activity in presence of ursolic acid by Gal4-luciferase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Lycera

Curated by ChEMBL
LigandPNGBDBM50577413(CHEMBL4874944)
Affinity DataEC50:  411nMAssay Description:Agonist activity at human ROR-gamma LBD expressed in HEK293 cells assessed as transcriptional activity in presence of ursolic acid by Gal4-luciferase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Lycera

Curated by ChEMBL
LigandPNGBDBM50577414(CHEMBL4873783)
Affinity DataEC50:  495nMAssay Description:Agonist activity at human ROR-gamma LBD expressed in HEK293 cells assessed as transcriptional activity in presence of ursolic acid by Gal4-luciferase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Lycera

Curated by ChEMBL
LigandPNGBDBM50577451(CHEMBL4855415)
Affinity DataEC50:  199nMAssay Description:Agonist activity at human ROR-gamma LBD expressed in HEK293 cells assessed as transcriptional activity in presence of ursolic acid by Gal4-luciferase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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