Compile Data Set for Download or QSAR
maximum 50k data
Found 17 Enz. Inhib. hit(s) with all data for entry = 5853
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Eisai

US Patent
LigandPNGBDBM97558(US8470825, 4d)
Affinity DataIC50:  20nMpH: 8.0 T: 2°CAssay Description:PARP assay using purified recombinant human PARP from Trevigan.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Eisai

US Patent
LigandPNGBDBM97556(US8470825, 4b)
Affinity DataIC50:  20nMpH: 8.0 T: 2°CAssay Description:PARP assay using purified recombinant human PARP from Trevigan.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Eisai

US Patent
LigandPNGBDBM97557(US8470825, 4c)
Affinity DataIC50:  30nMpH: 8.0 T: 2°CAssay Description:PARP assay using purified recombinant human PARP from Trevigan.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Eisai

US Patent
LigandPNGBDBM97555(US8470825, 4a)
Affinity DataIC50:  30nMpH: 8.0 T: 2°CAssay Description:PARP assay using purified recombinant human PARP from Trevigan.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Eisai

US Patent
LigandPNGBDBM97572(US8470825, 4r)
Affinity DataIC50:  30nMpH: 8.0 T: 2°CAssay Description:PARP assay using purified recombinant human PARP from Trevigan.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Eisai

US Patent
LigandPNGBDBM97570(US8470825, 4p)
Affinity DataIC50:  30nMpH: 8.0 T: 2°CAssay Description:PARP assay using purified recombinant human PARP from Trevigan.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Eisai

US Patent
LigandPNGBDBM97563(US8470825, 4i)
Affinity DataIC50:  40nMpH: 8.0 T: 2°CAssay Description:PARP assay using purified recombinant human PARP from Trevigan.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Eisai

US Patent
LigandPNGBDBM97569(US8470825, 4o)
Affinity DataIC50:  50nMpH: 8.0 T: 2°CAssay Description:PARP assay using purified recombinant human PARP from Trevigan.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Eisai

US Patent
LigandPNGBDBM97571(US8470825, 4q)
Affinity DataIC50:  50nMpH: 8.0 T: 2°CAssay Description:PARP assay using purified recombinant human PARP from Trevigan.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Eisai

US Patent
LigandPNGBDBM97567(US8470825, 4m)
Affinity DataIC50:  100nMpH: 8.0 T: 2°CAssay Description:PARP assay using purified recombinant human PARP from Trevigan.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Eisai

US Patent
LigandPNGBDBM97566(US8470825, 4l)
Affinity DataIC50:  100nMpH: 8.0 T: 2°CAssay Description:PARP assay using purified recombinant human PARP from Trevigan.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Eisai

US Patent
LigandPNGBDBM97564(US8470825, 4j)
Affinity DataIC50:  100nMpH: 8.0 T: 2°CAssay Description:PARP assay using purified recombinant human PARP from Trevigan.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Eisai

US Patent
LigandPNGBDBM97568(US8470825, 4n)
Affinity DataIC50:  100nMpH: 8.0 T: 2°CAssay Description:PARP assay using purified recombinant human PARP from Trevigan.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Eisai

US Patent
LigandPNGBDBM97562(US8470825, 4h)
Affinity DataIC50:  100nMpH: 8.0 T: 2°CAssay Description:PARP assay using purified recombinant human PARP from Trevigan.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Eisai

US Patent
LigandPNGBDBM97573(US8470825, 4s)
Affinity DataIC50:  120nMpH: 8.0 T: 2°CAssay Description:PARP assay using purified recombinant human PARP from Trevigan.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Eisai

US Patent
LigandPNGBDBM97565(US8470825, 4k)
Affinity DataIC50:  300nMpH: 8.0 T: 2°CAssay Description:PARP assay using purified recombinant human PARP from Trevigan.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Eisai

US Patent
LigandPNGBDBM97561(US8470825, 4g)
Affinity DataIC50:  500nMpH: 8.0 T: 2°CAssay Description:PARP assay using purified recombinant human PARP from Trevigan.More data for this Ligand-Target Pair
In DepthDetails US Patent