Compile Data Set for Download or QSAR
maximum 50k data
Found 15 Enz. Inhib. hit(s) with all data for entry = 50034414
TargetAutoinducer 2-binding periplasmic protein LuxP(Vibrio harveyi)
Instituto De Tecnologia Qu£Mica E Biol£Gica

Curated by ChEMBL
LigandPNGBDBM50362021(CHEMBL1939887 | CHEMBL1939889)
Affinity DataIC50:  5.75E+4nMAssay Description:Antagonist activity at Vibrio harveyi MM32 LuxP receptor assessed as decrease in receptor agonist DPD-induced bioluminescence after 5 hrs 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAutoinducer 2-binding periplasmic protein LuxP(Vibrio harveyi)
Instituto De Tecnologia Qu£Mica E Biol£Gica

Curated by ChEMBL
LigandPNGBDBM50362022(CHEMBL1939888 | CHEMBL1939890)
Affinity DataIC50:  1.60E+5nMAssay Description:Antagonist activity at Vibrio harveyi MM32 LuxP receptor assessed as decrease in receptor agonist DPD-induced bioluminescence after 5 hrs 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAutoinducer 2-binding periplasmic protein LuxP(Vibrio harveyi)
Instituto De Tecnologia Qu£Mica E Biol£Gica

Curated by ChEMBL
LigandPNGBDBM50362021(CHEMBL1939887 | CHEMBL1939889)
Affinity DataIC50:  1.69E+5nMAssay Description:Antagonist activity at Vibrio harveyi MM32 LuxP receptor assessed as decrease in receptor agonist DPD-induced bioluminescence after 5 hrs 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAutoinducer 2-binding periplasmic protein LuxP(Vibrio harveyi)
Instituto De Tecnologia Qu£Mica E Biol£Gica

Curated by ChEMBL
LigandPNGBDBM50362021(CHEMBL1939887 | CHEMBL1939889)
Affinity DataEC50:  140nMAssay Description:Binding affinity to Vibrio harveyi CFP/YFP-tagged LuxP receptor assessed as decrease in FRET ratioMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAutoinducer 2-binding periplasmic protein LuxP(Vibrio harveyi)
Instituto De Tecnologia Qu£Mica E Biol£Gica

Curated by ChEMBL
LigandPNGBDBM50362022(CHEMBL1939888 | CHEMBL1939890)
Affinity DataEC50:  1.16E+4nMAssay Description:Binding affinity to Vibrio harveyi CFP/YFP-tagged LuxP receptor assessed as decrease in FRET ratioMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAutoinducer 2-binding periplasmic protein LuxP(Vibrio harveyi)
Instituto De Tecnologia Qu£Mica E Biol£Gica

Curated by ChEMBL
LigandPNGBDBM50165862((4S)-4,5-dihydroxypentane-2,3-dione | (S)-4,5-dihy...)
Affinity DataEC50:  76nMAssay Description:Agonist activity at Vibrio harveyi MM32 LuxP receptor assessed as induction of bioluminescence after 5 hrs 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAutoinducer 2-binding periplasmic protein LuxP(Vibrio harveyi)
Instituto De Tecnologia Qu£Mica E Biol£Gica

Curated by ChEMBL
LigandPNGBDBM50362021(CHEMBL1939887 | CHEMBL1939889)
Affinity DataEC50:  6.21E+3nMAssay Description:Agonist activity at Vibrio harveyi MM32 LuxP receptor assessed as induction of bioluminescence after 5 hrs 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAutoinducer 2-binding periplasmic protein LuxP(Vibrio harveyi)
Instituto De Tecnologia Qu£Mica E Biol£Gica

Curated by ChEMBL
LigandPNGBDBM50362022(CHEMBL1939888 | CHEMBL1939890)
Affinity DataEC50:  2.65E+4nMAssay Description:Agonist activity at Vibrio harveyi MM32 LuxP receptor assessed as induction of bioluminescence after 5 hrs 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAutoinducer 2-binding periplasmic protein LuxP(Vibrio harveyi)
Instituto De Tecnologia Qu£Mica E Biol£Gica

Curated by ChEMBL
LigandPNGBDBM50362021(CHEMBL1939887 | CHEMBL1939889)
Affinity DataEC50:  650nMAssay Description:Agonist activity at Vibrio harveyi MM32 LuxP receptor assessed as induction of bioluminescence after 5 hrs 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAutoinducer 2-binding periplasmic protein LuxP(Vibrio harveyi)
Instituto De Tecnologia Qu£Mica E Biol£Gica

Curated by ChEMBL
LigandPNGBDBM50362022(CHEMBL1939888 | CHEMBL1939890)
Affinity DataEC50:  1.95E+4nMAssay Description:Agonist activity at Vibrio harveyi MM32 LuxP receptor assessed as induction of bioluminescence after 5 hrs 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAutoinducer 2-binding periplasmic protein LuxP(Vibrio harveyi)
Instituto De Tecnologia Qu£Mica E Biol£Gica

Curated by ChEMBL
LigandPNGBDBM50362025(CHEMBL1939886)
Affinity DataEC50:  3.00E+4nMAssay Description:Agonist activity at Vibrio harveyi LuxP receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAutoinducer 2-binding periplasmic protein LuxP(Vibrio harveyi)
Instituto De Tecnologia Qu£Mica E Biol£Gica

Curated by ChEMBL
LigandPNGBDBM50362022(CHEMBL1939888 | CHEMBL1939890)
Affinity DataEC50:  1.00E+4nMAssay Description:Binding affinity to Vibrio harveyi CFP/YFP-tagged LuxP receptor assessed as decrease in FRET ratioMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAutoinducer 2-binding periplasmic protein LuxP(Vibrio harveyi)
Instituto De Tecnologia Qu£Mica E Biol£Gica

Curated by ChEMBL
LigandPNGBDBM50165862((4S)-4,5-dihydroxypentane-2,3-dione | (S)-4,5-dihy...)
Affinity DataEC50:  3.00E+4nMAssay Description:Agonist activity at Vibrio harveyi LuxP receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAutoinducer 2-binding periplasmic protein LuxP(Vibrio harveyi)
Instituto De Tecnologia Qu£Mica E Biol£Gica

Curated by ChEMBL
LigandPNGBDBM50165862((4S)-4,5-dihydroxypentane-2,3-dione | (S)-4,5-dihy...)
Affinity DataEC50:  32nMAssay Description:Binding affinity to Vibrio harveyi CFP/YFP-tagged LuxP receptor assessed as decrease in FRET ratioMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAutoinducer 2-binding periplasmic protein LuxP(Vibrio harveyi)
Instituto De Tecnologia Qu£Mica E Biol£Gica

Curated by ChEMBL
LigandPNGBDBM50362021(CHEMBL1939887 | CHEMBL1939889)
Affinity DataEC50:  1.87E+3nMAssay Description:Binding affinity to Vibrio harveyi CFP/YFP-tagged LuxP receptor assessed as decrease in FRET ratioMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed