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Found 38 Enz. Inhib. hit(s) with all data for entry = 50003495
TargetSodium/hydrogen exchanger 3(Oryctolagus cuniculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50058715(CHEMBL64360 | EMD-96785 | ENIPORIDE | N-(5-Methane...)
Affinity DataIC50:  8nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/hydrogen exchanger 3(Oryctolagus cuniculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50471819(CHEMBL332433)
Affinity DataIC50:  13nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium/hydrogen exchanger 3(Oryctolagus cuniculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50471814(CHEMBL126367)
Affinity DataIC50:  14nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium/hydrogen exchanger 3(Oryctolagus cuniculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50471802(CHEMBL124274)
Affinity DataIC50:  16nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium/hydrogen exchanger 3(Oryctolagus cuniculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50471801(CHEMBL331794)
Affinity DataIC50:  17nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium/hydrogen exchanger 3(Oryctolagus cuniculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50471791(CHEMBL439605)
Affinity DataIC50:  19nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium/hydrogen exchanger 3(Oryctolagus cuniculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50471796(CHEMBL124547)
Affinity DataIC50:  21nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium/hydrogen exchanger 3(Oryctolagus cuniculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50471794(CHEMBL124044)
Affinity DataIC50:  24nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium/hydrogen exchanger 3(Oryctolagus cuniculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50234609(Cariporide | HOE-642)
Affinity DataIC50:  26nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/hydrogen exchanger 3(Oryctolagus cuniculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50471811(CHEMBL126060)
Affinity DataIC50:  27nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium/hydrogen exchanger 3(Oryctolagus cuniculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50471823(CHEMBL341296)
Affinity DataIC50:  28nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium/hydrogen exchanger 3(Oryctolagus cuniculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50471812(CHEMBL331630)
Affinity DataIC50:  28nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium/hydrogen exchanger 3(Oryctolagus cuniculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50471815(CHEMBL123578)
Affinity DataIC50:  29nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium/hydrogen exchanger 3(Oryctolagus cuniculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50471805(CHEMBL122142)
Affinity DataIC50:  30nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium/hydrogen exchanger 3(Oryctolagus cuniculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50471808(CHEMBL333059)
Affinity DataIC50:  34nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium/hydrogen exchanger 3(Oryctolagus cuniculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50471803(CHEMBL123859)
Affinity DataIC50:  36nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium/hydrogen exchanger 3(Oryctolagus cuniculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50471804(CHEMBL421240)
Affinity DataIC50:  38nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium/hydrogen exchanger 3(Oryctolagus cuniculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50471813(CHEMBL331457)
Affinity DataIC50:  40nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium/hydrogen exchanger 3(Oryctolagus cuniculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50471807(CHEMBL125283)
Affinity DataIC50:  43nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium/hydrogen exchanger 3(Oryctolagus cuniculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50471818(CHEMBL273539)
Affinity DataIC50:  44nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium/hydrogen exchanger 3(Oryctolagus cuniculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50471795(CHEMBL123160)
Affinity DataIC50:  45nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium/hydrogen exchanger 3(Oryctolagus cuniculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50471816(CHEMBL125952)
Affinity DataIC50:  45nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium/hydrogen exchanger 3(Oryctolagus cuniculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50471790(CHEMBL333480)
Affinity DataIC50:  54nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium/hydrogen exchanger 3(Oryctolagus cuniculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50471820(CHEMBL330935)
Affinity DataIC50:  56nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium/hydrogen exchanger 3(Oryctolagus cuniculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50471799(CHEMBL124884)
Affinity DataIC50:  60nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium/hydrogen exchanger 3(Oryctolagus cuniculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50471797(CHEMBL124762)
Affinity DataIC50:  60nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium/hydrogen exchanger 3(Oryctolagus cuniculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50471809(CHEMBL333804)
Affinity DataIC50:  70nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium/hydrogen exchanger 3(Oryctolagus cuniculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50471817(CHEMBL122853)
Affinity DataIC50:  93nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium/hydrogen exchanger 3(Oryctolagus cuniculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50471792(CHEMBL340249)
Affinity DataIC50:  95nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium/hydrogen exchanger 3(Oryctolagus cuniculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50471821(CHEMBL121732)
Affinity DataIC50:  96nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium/hydrogen exchanger 3(Oryctolagus cuniculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50471810(CHEMBL445376)
Affinity DataIC50:  96nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium/hydrogen exchanger 3(Oryctolagus cuniculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50471806(CHEMBL125951)
Affinity DataIC50:  116nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium/hydrogen exchanger 3(Oryctolagus cuniculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50471793(CHEMBL121787)
Affinity DataIC50:  130nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium/hydrogen exchanger 3(Oryctolagus cuniculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50471798(CHEMBL122238)
Affinity DataIC50:  360nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium/hydrogen exchanger 3(Oryctolagus cuniculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50471824(CHEMBL124987)
Affinity DataIC50:  700nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium/hydrogen exchanger 3(Oryctolagus cuniculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50471822(CHEMBL124826)
Affinity DataIC50:  790nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium/hydrogen exchanger 3(Oryctolagus cuniculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50471800(CHEMBL333112)
Affinity DataIC50:  1.50E+3nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium/hydrogen exchanger 3(Oryctolagus cuniculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50471789(CHEMBL419609)
Affinity DataIC50:  2.20E+3nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed