Found 63 Enz. Inhib. hit(s) with all data for entry = 50033219 
Affinity DataIC50: 200nMAssay Description:Inverse agonist activity at SF-1More data for this Ligand-Target Pair
Affinity DataIC50: 7.30E+3nMAssay Description:Inverse agonist activity at SF-1More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 5 group A member 2(Homo sapiens (Human))
University Of Southampton
Curated by ChEMBL
University Of Southampton
Curated by ChEMBL
Affinity DataEC50: 3.16E+3nMAssay Description:Agonist activity at human LRH-1 receptor assessed as TIF2 737-757 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 5 group A member 2(Homo sapiens (Human))
University Of Southampton
Curated by ChEMBL
University Of Southampton
Curated by ChEMBL
Affinity DataEC50: 5.01E+3nMAssay Description:Agonist activity at human LRH-1 receptor assessed as TIF2 737-757 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
Affinity DataEC50: 31.6nMAssay Description:Agonist activity at human SF-1 assessed as DAX1 1-23 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 5 group A member 2(Homo sapiens (Human))
University Of Southampton
Curated by ChEMBL
University Of Southampton
Curated by ChEMBL
Affinity DataEC50: 31.6nMAssay Description:Agonist activity at human LRH-1 receptor assessed as TIF2 737-757 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
Affinity DataEC50: 39.8nMAssay Description:Agonist activity at human SF-1 assessed as DAX1 1-23 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
Affinity DataEC50: 39.8nMAssay Description:Agonist activity at human SF-1 assessed as DAX1 1-23 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
Affinity DataEC50: 63.1nMAssay Description:Agonist activity at human SF-1 assessed as DAX1 1-23 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
Affinity DataEC50: 63.1nMAssay Description:Agonist activity at human SF-1 assessed as DAX1 1-23 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
Affinity DataEC50: 63.1nMAssay Description:Agonist activity at human SF-1 assessed as DAX1 1-23 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
Affinity DataEC50: 63.1nMAssay Description:Agonist activity at human SF-1 assessed as DAX1 1-23 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
Affinity DataEC50: 63.1nMAssay Description:Agonist activity at human SF-1 assessed as DAX1 1-23 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
Affinity DataEC50: 79.4nMAssay Description:Agonist activity at human SF-1 assessed as DAX1 1-23 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
Affinity DataEC50: 79.4nMAssay Description:Agonist activity at human SF-1 assessed as DAX1 1-23 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 5 group A member 2(Homo sapiens (Human))
University Of Southampton
Curated by ChEMBL
University Of Southampton
Curated by ChEMBL
Affinity DataEC50: 100nMAssay Description:Agonist activity at human LRH-1 receptor assessed as TIF2 737-757 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
Affinity DataEC50: 126nMAssay Description:Agonist activity at human SF-1 assessed as DAX1 1-23 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
Affinity DataEC50: 158nMAssay Description:Agonist activity at human SF-1 assessed as DAX1 1-23 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
Affinity DataEC50: 158nMAssay Description:Agonist activity at human SF-1 assessed as DAX1 1-23 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
Affinity DataEC50: 158nMAssay Description:Agonist activity at human SF-1 assessed as DAX1 1-23 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
Affinity DataEC50: 158nMAssay Description:Agonist activity at human SF-1 assessed as DAX1 1-23 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 5 group A member 2(Homo sapiens (Human))
University Of Southampton
Curated by ChEMBL
University Of Southampton
Curated by ChEMBL
Affinity DataEC50: 158nMAssay Description:Agonist activity at human LRH-1 receptor assessed as TIF2 737-757 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
Affinity DataEC50: 200nMAssay Description:Agonist activity at human SF-1 assessed as DAX1 1-23 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
Affinity DataEC50: 200nMAssay Description:Agonist activity at human SF-1 assessed as DAX1 1-23 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
Affinity DataEC50: 200nMAssay Description:Agonist activity at human SF-1 assessed as DAX1 1-23 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
Affinity DataEC50: 200nMAssay Description:Agonist activity at human SF-1 assessed as DAX1 1-23 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
Affinity DataEC50: 200nMAssay Description:Agonist activity at human SF-1 assessed as DAX1 1-23 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 5 group A member 2(Homo sapiens (Human))
University Of Southampton
Curated by ChEMBL
University Of Southampton
Curated by ChEMBL
Affinity DataEC50: 200nMAssay Description:Agonist activity at human LRH-1 receptor assessed as TIF2 737-757 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
Affinity DataEC50: 251nMAssay Description:Agonist activity at human SF-1 assessed as DAX1 1-23 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 5 group A member 2(Homo sapiens (Human))
University Of Southampton
Curated by ChEMBL
University Of Southampton
Curated by ChEMBL
Affinity DataEC50: 2.51E+3nMAssay Description:Agonist activity at human LRH-1 receptor assessed as TIF2 737-757 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
Affinity DataEC50: 251nMAssay Description:Agonist activity at human SF-1 assessed as DAX1 1-23 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 5 group A member 2(Homo sapiens (Human))
University Of Southampton
Curated by ChEMBL
University Of Southampton
Curated by ChEMBL
Affinity DataEC50: 251nMAssay Description:Agonist activity at human LRH-1 receptor assessed as TIF2 737-757 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 5 group A member 2(Homo sapiens (Human))
University Of Southampton
Curated by ChEMBL
University Of Southampton
Curated by ChEMBL
Affinity DataEC50: 251nMAssay Description:Agonist activity at human LRH-1 receptor assessed as TIF2 737-757 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
3D Structure (crystal)TargetNuclear receptor subfamily 5 group A member 2(Homo sapiens (Human))
University Of Southampton
Curated by ChEMBL
University Of Southampton
Curated by ChEMBL
Affinity DataEC50: 251nMAssay Description:Agonist activity at human LRH-1 receptor assessed as TIF2 737-757 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 5 group A member 2(Homo sapiens (Human))
University Of Southampton
Curated by ChEMBL
University Of Southampton
Curated by ChEMBL
Affinity DataEC50: 251nMAssay Description:Agonist activity at human LRH-1 receptor assessed as TIF2 737-757 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 5 group A member 2(Homo sapiens (Human))
University Of Southampton
Curated by ChEMBL
University Of Southampton
Curated by ChEMBL
Affinity DataEC50: 251nMAssay Description:Agonist activity at human LRH-1 receptor assessed as TIF2 737-757 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
Affinity DataEC50: 316nMAssay Description:Agonist activity at human SF-1 assessed as DAX1 1-23 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
Affinity DataEC50: 316nMAssay Description:Agonist activity at human SF-1 assessed as DAX1 1-23 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 5 group A member 2(Homo sapiens (Human))
University Of Southampton
Curated by ChEMBL
University Of Southampton
Curated by ChEMBL
Affinity DataEC50: 316nMAssay Description:Agonist activity at human LRH-1 receptor assessed as TIF2 737-757 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 5 group A member 2(Homo sapiens (Human))
University Of Southampton
Curated by ChEMBL
University Of Southampton
Curated by ChEMBL
Affinity DataEC50: 316nMAssay Description:Agonist activity at human LRH-1 receptor assessed as TIF2 737-757 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
Affinity DataEC50: 398nMAssay Description:Agonist activity at human SF-1 assessed as DAX1 1-23 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
Affinity DataEC50: 398nMAssay Description:Agonist activity at human SF-1 assessed as DAX1 1-23 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
Affinity DataEC50: 398nMAssay Description:Agonist activity at human SF-1 assessed as DAX1 1-23 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
Affinity DataEC50: 398nMAssay Description:Agonist activity at human SF-1 assessed as DAX1 1-23 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 5 group A member 2(Homo sapiens (Human))
University Of Southampton
Curated by ChEMBL
University Of Southampton
Curated by ChEMBL
Affinity DataEC50: 398nMAssay Description:Agonist activity at human LRH-1 receptor assessed as TIF2 737-757 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 5 group A member 2(Homo sapiens (Human))
University Of Southampton
Curated by ChEMBL
University Of Southampton
Curated by ChEMBL
Affinity DataEC50: 398nMAssay Description:Agonist activity at human LRH-1 receptor assessed as TIF2 737-757 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
Affinity DataEC50: 501nMAssay Description:Agonist activity at human SF-1 assessed as DAX1 1-23 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 5 group A member 2(Homo sapiens (Human))
University Of Southampton
Curated by ChEMBL
University Of Southampton
Curated by ChEMBL
Affinity DataEC50: 501nMAssay Description:Agonist activity at human LRH-1 receptor assessed as TIF2 737-757 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 5 group A member 2(Homo sapiens (Human))
University Of Southampton
Curated by ChEMBL
University Of Southampton
Curated by ChEMBL
Affinity DataEC50: 631nMAssay Description:Agonist activity at human LRH-1 receptor assessed as TIF2 737-757 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 5 group A member 2(Homo sapiens (Human))
University Of Southampton
Curated by ChEMBL
University Of Southampton
Curated by ChEMBL
Affinity DataEC50: 794nMAssay Description:Agonist activity at human LRH-1 receptor assessed as TIF2 737-757 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
