Compile Data Set for Download or QSAR
maximum 50k data
Found 7 Enz. Inhib. hit(s) with all data for entry = 50034554
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50364112(CHEMBL1950962)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of HMT-G9a using S-adenosylmethionine and biotinylated H3 peptide after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50364111(CHEMBL1950961)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of HMT-G9a using S-adenosylmethionine and biotinylated H3 peptide after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50134315(7-hydroxy-11-hydroxymethyl-12-methyl-14,15-dithia-...)
Affinity DataIC50:  6.40E+3nMAssay Description:Inhibition of HMT-G9a using S-adenosylmethionine and biotinylated H3 peptide after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50364109(CHEMBL1950960)
Affinity DataIC50:  5.50E+4nMAssay Description:Inhibition of HMT-G9a using S-adenosylmethionine and biotinylated H3 peptide after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50364110(CHEMBL1088849)
Affinity DataIC50:  5.80E+4nMAssay Description:Inhibition of HMT-G9a using S-adenosylmethionine and biotinylated H3 peptide after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50364108(CHEMBL1950959)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of HMT-G9a using S-adenosylmethionine and biotinylated H3 peptide after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50315535(CHEMBL1088981 | bis(methylthio)gliotoxin)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of HMT-G9a using S-adenosylmethionine and biotinylated H3 peptide after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed