Compile Data Set for Download or QSAR
maximum 50k data
Found 27 Enz. Inhib. hit(s) with all data for entry = 50012799
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50560404(CHEMBL4750820)
Affinity DataEC50:  5.51E+3nMAssay Description:Agonist activity at Rev-Erb alpha (unknown origin) by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50560414(CHEMBL4763333)
Affinity DataEC50:  150nMAssay Description:Inverse agonist activity at Rev-Erb alpha LBD (unknown origin) by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50560406(CHEMBL4757143)
Affinity DataEC50: <1.00E+3nMAssay Description:Agonist activity at Rev-Erb alpha (unknown origin) by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50383676(CHEMBL2030075)
Affinity DataEC50:  140nMAssay Description:Agonist activity at Rev-Erb alpha (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50383670(CHEMBL2030069)
Affinity DataEC50: >3.00E+3nMAssay Description:Agonist activity at Rev-Erb alpha (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50383661(CHEMBL2030064)
Affinity DataEC50:  650nMAssay Description:Agonist activity at Rev-Erb alpha (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50434037(CHEMBL2381208)
Affinity DataEC50:  200nMAssay Description:Agonist activity at Rev-Erb alpha (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50434030(CHEMBL2381202)
Affinity DataEC50:  160nMAssay Description:Agonist activity at Rev-Erb alpha (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50366239(CHEMBL1961797)
Affinity DataEC50:  710nMAssay Description:Agonist activity at Rev-Erb alpha (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50366238(CHEMBL1961796)
Affinity DataEC50:  620nMAssay Description:Agonist activity at Rev-Erb alpha (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50560407(CHEMBL4795406)
Affinity DataEC50:  520nMAssay Description:Agonist activity at Rev-Erb alpha (unknown origin) by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50560408(CHEMBL4744123)
Affinity DataEC50: <5.00E+3nMAssay Description:Agonist activity at Rev-Erb alpha (unknown origin) by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50383675(CHEMBL2030074)
Affinity DataEC50:  77nMAssay Description:Agonist activity at Rev-Erb alpha (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50560409(CHEMBL4781178)
Affinity DataEC50:  68nMAssay Description:Agonist activity at Rev-Erb alpha (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50434039(CHEMBL2381193)
Affinity DataEC50:  200nMAssay Description:Agonist activity at Rev-Erb alpha (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50560410(CHEMBL4761268)
Affinity DataEC50:  50nMAssay Description:Agonist activity at Rev-Erb alpha (unknown origin) by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50383684(CHEMBL1961795)
Affinity DataEC50:  2.30E+3nMAssay Description:Agonist activity at Rev-Erb alpha (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50383676(CHEMBL2030075)
Affinity DataEC50:  140nMAssay Description:Agonist activity at Rev-Erb alpha (unknown origin) by BMAL1-luciferase reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50383675(CHEMBL2030074)
Affinity DataEC50:  77nMAssay Description:Agonist activity at Rev-Erb alpha (unknown origin) by BMAL1-luciferase reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50383670(CHEMBL2030069)
Affinity DataEC50:  3.00E+3nMAssay Description:Agonist activity at Rev-Erb alpha (unknown origin) by BMAL1-luciferase reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50383661(CHEMBL2030064)
Affinity DataEC50:  650nMAssay Description:Agonist activity at Rev-Erb alpha (unknown origin) by BMAL1-luciferase reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50560411(CHEMBL4739959)
Affinity DataEC50:  1.30E+3nMAssay Description:Antagonist activity at Rev-Erb alpha (unknown origin) by BMAL1-luciferase reporter assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50560412(CHEMBL4799119)
Affinity DataEC50:  1.30E+3nMAssay Description:Antagonist activity at Rev-Erb alpha (unknown origin) by BMAL1-luciferase reporter assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50560413(CHEMBL4754504)
Affinity DataEC50:  470nMAssay Description:Antagonist activity at Rev-Erb alpha (unknown origin) by BMAL1-luciferase reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50560410(CHEMBL4761268)
Affinity DataEC50:  2.05E+3nMAssay Description:Antagonist activity at Rev-Erb alpha (unknown origin) by BMAL1-luciferase reporter assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50095836(CHEMBL3590544)
Affinity DataEC50:  3.00E+4nMAssay Description:Antagonist activity at Rev-Erb alpha (unknown origin) by RORE-luciferase reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50560405(CHEMBL4747677)
Affinity DataEC50:  1.13E+3nMAssay Description:Agonist activity at Rev-Erb alpha (unknown origin) by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed