Compile Data Set for Download or QSAR
maximum 50k data
Found 38 Enz. Inhib. hit(s) with all data for entry = 50030753
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50300884((E)-3-(2,4-Dimethoxy-phenyl)-N-(4-[5-(4-fluoro-phe...)
Affinity DataIC50:  4nMAssay Description:Inhibition of recombinant CK1delta kinase domain by Cherenkov countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50300884((E)-3-(2,4-Dimethoxy-phenyl)-N-(4-[5-(4-fluoro-phe...)
Affinity DataIC50:  5nMAssay Description:Inhibition of GST-fused rat CK1delta by Cherenkov counting in presence of 20 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50300893((E)-3-(2,4-Dimethoxy-phenyl)-N-(4-[5-(4-fluoro-phe...)
Affinity DataIC50:  5nMAssay Description:Inhibition of recombinant CK1delta kinase domain by Cherenkov countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50300888((S)-4-(3-(4-fluorophenyl)-5-isopropylisoxazol-4-yl...)
Affinity DataIC50:  6nMAssay Description:Inhibition of p38alpha by Cherenkov countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50300893((E)-3-(2,4-Dimethoxy-phenyl)-N-(4-[5-(4-fluoro-phe...)
Affinity DataIC50:  11nMAssay Description:Inhibition of GST-fused rat CK1delta by Cherenkov counting in presence of 20 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50300884((E)-3-(2,4-Dimethoxy-phenyl)-N-(4-[5-(4-fluoro-phe...)
Affinity DataIC50:  19nMAssay Description:Inhibition of p38alpha by Cherenkov countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50300885(CHEMBL569551 | N-sec-butyl-4-(3-(4-fluorophenyl)-5...)
Affinity DataIC50:  30nMAssay Description:Inhibition of p38alpha by Cherenkov countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50300892((E)-3-(2,4-dimethoxyphenyl)-N-(4-(3-(4-fluoropheny...)
Affinity DataIC50:  33nMAssay Description:Inhibition of recombinant CK1delta kinase domain by Cherenkov countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM13336(4-[4-(4-fluorophenyl)-2-(4-methanesulfinylphenyl)-...)
Affinity DataIC50:  40nMAssay Description:Inhibition of p38alpha by Cherenkov countingMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50300893((E)-3-(2,4-Dimethoxy-phenyl)-N-(4-[5-(4-fluoro-phe...)
Affinity DataIC50:  41nMAssay Description:Inhibition of p38alpha by Cherenkov countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50300892((E)-3-(2,4-dimethoxyphenyl)-N-(4-(3-(4-fluoropheny...)
Affinity DataIC50:  47nMAssay Description:Inhibition of GST-fused rat CK1delta by Cherenkov counting in presence of 20 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM13531(4-(4-Fluorophenyl)-2-(4-hydroxyphenyl)-5-(4-pyridy...)
Affinity DataIC50:  50nMAssay Description:Inhibition of p38alpha by Cherenkov countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50300886(4-(3-(4-fluorophenyl)-5-isopropylisoxazol-4-yl)-N-...)
Affinity DataIC50:  60nMAssay Description:Inhibition of p38alpha by Cherenkov countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50300884((E)-3-(2,4-Dimethoxy-phenyl)-N-(4-[5-(4-fluoro-phe...)
Affinity DataIC50:  73nMAssay Description:Inhibition of recombinant CK1epsilon by Cherenkov counting in presence of 20 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50300890(2-(4-fluorophenyl)-N-(4-(3-(4-fluorophenyl)-5-isop...)
Affinity DataIC50:  90nMAssay Description:Inhibition of GST-fused rat CK1delta by Cherenkov counting in presence of 20 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50300890(2-(4-fluorophenyl)-N-(4-(3-(4-fluorophenyl)-5-isop...)
Affinity DataIC50:  110nMAssay Description:Inhibition of recombinant CK1delta kinase domain by Cherenkov countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM13336(4-[4-(4-fluorophenyl)-2-(4-methanesulfinylphenyl)-...)
Affinity DataIC50:  120nMAssay Description:Inhibition of CK1delta by Cherenkov counting in presence of 20 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50206421(3-(4-fluorophenyl)-5-isopropyl-4-(pyridin-4-yl)iso...)
Affinity DataIC50:  230nMAssay Description:Inhibition of CK1delta by Cherenkov counting in presence of 20 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50206421(3-(4-fluorophenyl)-5-isopropyl-4-(pyridin-4-yl)iso...)
Affinity DataIC50:  230nMAssay Description:Inhibition of GST-fused rat CK1delta by Cherenkov counting in presence of 20 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50229971(4-(4-(2,3-Dihydrobenzo[1,4]dioxin-6-yl)-5-pyridin-...)
Affinity DataIC50:  300nMAssay Description:Inhibition of GST-fused rat CK1delta expressed in Escherichia coli using phosphorylated peptide TFRPRTSpSNASTIS as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50300889(CHEMBL585533 | N-(4-(3-(4-fluorophenyl)-5-isopropy...)
Affinity DataIC50:  300nMAssay Description:Inhibition of p38alpha by Cherenkov countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50300889(CHEMBL585533 | N-(4-(3-(4-fluorophenyl)-5-isopropy...)
Affinity DataIC50:  330nMAssay Description:Inhibition of GST-fused rat CK1delta by Cherenkov counting in presence of 20 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50300891((rac)-N-(4-(3-(4-fluorophenyl)-5-isopropylisoxazol...)
Affinity DataIC50:  340nMAssay Description:Inhibition of GST-fused rat CK1delta by Cherenkov counting in presence of 20 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50300893((E)-3-(2,4-Dimethoxy-phenyl)-N-(4-[5-(4-fluoro-phe...)
Affinity DataIC50:  447nMAssay Description:Inhibition of recombinant CK1epsilon by Cherenkov counting in presence of 20 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50300887((R)-4-(3-(4-fluorophenyl)-5-isopropylisoxazol-4-yl...)
Affinity DataIC50:  450nMAssay Description:Inhibition of p38alpha by Cherenkov countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50206421(3-(4-fluorophenyl)-5-isopropyl-4-(pyridin-4-yl)iso...)
Affinity DataIC50:  450nMAssay Description:Inhibition of p38alpha by Cherenkov countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50206421(3-(4-fluorophenyl)-5-isopropyl-4-(pyridin-4-yl)iso...)
Affinity DataIC50:  540nMAssay Description:Inhibition of JNK3 by Cherenkov counting in presence of 20 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50300889(CHEMBL585533 | N-(4-(3-(4-fluorophenyl)-5-isopropy...)
Affinity DataIC50:  700nMAssay Description:Inhibition of recombinant CK1delta kinase domain by Cherenkov countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50300891((rac)-N-(4-(3-(4-fluorophenyl)-5-isopropylisoxazol...)
Affinity DataIC50:  820nMAssay Description:Inhibition of recombinant CK1delta kinase domain by Cherenkov countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50300891((rac)-N-(4-(3-(4-fluorophenyl)-5-isopropylisoxazol...)
Affinity DataIC50:  890nMAssay Description:Inhibition of p38alpha by Cherenkov countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50263829(3-(2,4,6-Trimethoxybenzylidene)indolin-2-one | 3-[...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of human CK1deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50206421(3-(4-fluorophenyl)-5-isopropyl-4-(pyridin-4-yl)iso...)
Affinity DataIC50:  1.28E+3nMAssay Description:Inhibition of JNK2 by Cherenkov counting in presence of 20 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50300890(2-(4-fluorophenyl)-N-(4-(3-(4-fluorophenyl)-5-isop...)
Affinity DataIC50:  1.56E+3nMAssay Description:Inhibition of p38alpha by Cherenkov countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50300888((S)-4-(3-(4-fluorophenyl)-5-isopropylisoxazol-4-yl...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of recombinant CK1delta kinase domain by Cherenkov countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50206423(4-(5-(4-fluorophenyl)-3-isopropylisoxazol-4-yl)pyr...)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of p38alpha by Cherenkov countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50300886(4-(3-(4-fluorophenyl)-5-isopropylisoxazol-4-yl)-N-...)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of recombinant CK1delta kinase domain by Cherenkov countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50300892((E)-3-(2,4-dimethoxyphenyl)-N-(4-(3-(4-fluoropheny...)
Affinity DataIC50:  2.52E+3nMAssay Description:Inhibition of p38alpha by Cherenkov countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls University

Curated by ChEMBL
LigandPNGBDBM50229971(4-(4-(2,3-Dihydrobenzo[1,4]dioxin-6-yl)-5-pyridin-...)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of GST-fused human p38alpha expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed