TargetD(4) dopamine receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataKi: 25nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D4 receptor by radioligand binding assayMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataKi: 38nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D2 receptor expressed in stable fibroblast cells by radioligand binding assayMore data for this Ligand-Target Pair
TargetD(4) dopamine receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataKi: 58nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D4 receptor by radioligand binding assayMore data for this Ligand-Target Pair
TargetD(3) dopamine receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataKi: 62nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D3 receptor expressed in HEK293T cells by radioligand binding assayMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataKi: 70nMAssay Description:Displacement of [3H]DAMGO from human MOR expressed in HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataKi: 77nMAssay Description:Displacement of [3H]Nisoxetine from human NET expressed in HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataKi: 121nMAssay Description:Displacement of [3H]WIN35428 from human DAT expressed in HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataKi: 121nMAssay Description:Displacement of [3H]SCH23390 from human dopamine D5 receptor expressed in HEK293T cells by radioligand binding assayMore data for this Ligand-Target Pair
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataKi: 125nMAssay Description:Displacement of [3H]SCH23390 from human dopamine D5 receptor expressed in HEK293T cells by radioligand binding assayMore data for this Ligand-Target Pair
TargetD(4) dopamine receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataKi: 132nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D4 receptor by radioligand binding assayMore data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataKi: 135nMAssay Description:Displacement of [3H]SCH23390 from human dopamine D1 receptor expressed in HEK293T cells by radioligand binding assayMore data for this Ligand-Target Pair
TargetD(3) dopamine receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataKi: 136nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D3 receptor expressed in HEK293T cells by radioligand binding assayMore data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataKi: 147nMAssay Description:Displacement of [3H]SCH23390 from human dopamine D1 receptor expressed in HEK293T cells by radioligand binding assayMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataKi: 148nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D2 receptor expressed in stable fibroblast cells by radioligand binding assayMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataKi: 159nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D2 receptor expressed in stable fibroblast cells by radioligand binding assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataKi: 164nMAssay Description:Displacement of [3H]Ketanserin from 5-HT2A receptor (unknown origin) by radioligand binding assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataKi: 177nMAssay Description:Displacement of [3H]LSD from human 5-HT2B receptor expressed in HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataKi: 184nMAssay Description:Displacement of [3H]LSD from human 5-HT2B receptor expressed in HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataKi: 194nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D2 receptor expressed in stable fibroblast cells by radioligand binding assayMore data for this Ligand-Target Pair
TargetD(3) dopamine receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataKi: 209nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D3 receptor expressed in HEK293T cells by radioligand binding assayMore data for this Ligand-Target Pair
TargetHistamine H2 receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataKi: 252nMAssay Description:Displacement of [3H]Cimetidine from human H2 receptor expressed in HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
TargetHistamine H2 receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataKi: 278nMAssay Description:Displacement of [3H]Cimetidine from human H2 receptor expressed in HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataKi: 280nMAssay Description:Displacement of [3H]LSD from human 5-HT7A receptor expressed in HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataKi: 300nMAssay Description:Displacement of [3H]SCH23390 from human dopamine D1 receptor expressed in HEK293T cells by radioligand binding assayMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataKi: 317nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D2 receptor expressed in stable fibroblast cells by radioligand binding assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataKi: 326nMAssay Description:Displacement of [3H]LSD from human 5-HT7A receptor expressed in HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataKi: 328nMAssay Description:Displacement of [3H]DAMGO from human MOR expressed in HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataKi: 356nMAssay Description:Displacement of [3H]DAMGO from human MOR expressed in HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataKi: 356nMAssay Description:Displacement of [3H]-Way100635 from human 5HT1A receptor expressed in stable CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataKi: 361nMAssay Description:Displacement of [3H]Ketanserin from 5-HT2A receptor (unknown origin) by radioligand binding assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataKi: 374nMAssay Description:Displacement of [3H]LSD from human 5-HT2B receptor expressed in HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
TargetD(4) dopamine receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataKi: 385nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D4 receptor by radioligand binding assayMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataKi: 401nMAssay Description:Displacement of [3H]Rauwolscine from human alpha 2B adrenergic receptor expressed in HEK293T cells by radioligand binding assayMore data for this Ligand-Target Pair
TargetHistamine H2 receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataKi: 401nMAssay Description:Displacement of [3H]Cimetidine from human H2 receptor expressed in HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataKi: 402nMAssay Description:Displacement of [3H]Mesulergine from human 5-HT2C receptor expressed in HEK293FlpIN cells by radioligand binding assayMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataKi: 417nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D2 receptor expressed in stable fibroblast cells by radioligand binding assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataKi: 423nMAssay Description:Displacement of [3H]LSD from human 5-HT2B receptor expressed in HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataKi: 428nMAssay Description:Displacement of [3H]Citalopram from human SERT expressed in HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataKi: 437nMAssay Description:Displacement of [3H]SCH23390 from human dopamine D5 receptor expressed in HEK293T cells by radioligand binding assayMore data for this Ligand-Target Pair
TargetD(3) dopamine receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataKi: 437nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D3 receptor expressed in HEK293T cells by radioligand binding assayMore data for this Ligand-Target Pair
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataKi: 445nMAssay Description:Displacement of [3H]Rauwolscine from human alpha 2C adrenergic receptor expressed in MDCK cells by radioligand binding assayMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataKi: 458nMAssay Description:Displacement of [3H]Nisoxetine from human NET expressed in HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
TargetD(4) dopamine receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataKi: 459nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D4 receptor by radioligand binding assayMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataKi: 460nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D2 receptor expressed in stable fibroblast cells by radioligand binding assayMore data for this Ligand-Target Pair
TargetD(3) dopamine receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataKi: 474nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D3 receptor expressed in HEK293T cells by radioligand binding assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataKi: 481nMAssay Description:Displacement of [3H]-Way100635 from human 5HT1A receptor expressed in stable CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataKi: 509nMAssay Description:Displacement of [3H]LSD from human 5-HT2B receptor expressed in HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataKi: 515nMAssay Description:Displacement of [3H]CGP12177 from human beta 3 adrenergic receptor expressed in HEK293FlpIN cells by radioligand binding assayMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataKi: 518nMAssay Description:Displacement of [3H]Nisoxetine from human NET expressed in HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
TargetHistamine H2 receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center
Curated by ChEMBL
Texas Tech University Health Sciences Center
Curated by ChEMBL
Affinity DataKi: 526nMAssay Description:Displacement of [3H]Cimetidine from human H2 receptor expressed in HEK cells by radioligand binding assayMore data for this Ligand-Target Pair