Compile Data Set for Download or QSAR
maximum 50k data
Found 146 Enz. Inhib. hit(s) with all data for entry = 50003024
TargetD(4) dopamine receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50465908(CHEMBL4291048)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D4 receptor by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50465911(CHEMBL1644980)
Affinity DataKi:  38nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D2 receptor expressed in stable fibroblast cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50465911(CHEMBL1644980)
Affinity DataKi:  58nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D4 receptor by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50465911(CHEMBL1644980)
Affinity DataKi:  62nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D3 receptor expressed in HEK293T cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50465911(CHEMBL1644980)
Affinity DataKi:  70nMAssay Description:Displacement of [3H]DAMGO from human MOR expressed in HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50465909(CHEMBL1644978)
Affinity DataKi:  77nMAssay Description:Displacement of [3H]Nisoxetine from human NET expressed in HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50465911(CHEMBL1644980)
Affinity DataKi:  121nMAssay Description:Displacement of [3H]WIN35428 from human DAT expressed in HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50465911(CHEMBL1644980)
Affinity DataKi:  121nMAssay Description:Displacement of [3H]SCH23390 from human dopamine D5 receptor expressed in HEK293T cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50026066(1-(4,4-bis(4-fluorophenyl)butyl)-4-(4-chloro-3-(tr...)
Affinity DataKi:  125nMAssay Description:Displacement of [3H]SCH23390 from human dopamine D5 receptor expressed in HEK293T cells by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50465907(CHEMBL4282702)
Affinity DataKi:  132nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D4 receptor by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50465911(CHEMBL1644980)
Affinity DataKi:  135nMAssay Description:Displacement of [3H]SCH23390 from human dopamine D1 receptor expressed in HEK293T cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50026066(1-(4,4-bis(4-fluorophenyl)butyl)-4-(4-chloro-3-(tr...)
Affinity DataKi:  136nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D3 receptor expressed in HEK293T cells by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50026066(1-(4,4-bis(4-fluorophenyl)butyl)-4-(4-chloro-3-(tr...)
Affinity DataKi:  147nMAssay Description:Displacement of [3H]SCH23390 from human dopamine D1 receptor expressed in HEK293T cells by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50465908(CHEMBL4291048)
Affinity DataKi:  148nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D2 receptor expressed in stable fibroblast cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50026066(1-(4,4-bis(4-fluorophenyl)butyl)-4-(4-chloro-3-(tr...)
Affinity DataKi:  159nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D2 receptor expressed in stable fibroblast cells by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50465908(CHEMBL4291048)
Affinity DataKi:  164nMAssay Description:Displacement of [3H]Ketanserin from 5-HT2A receptor (unknown origin) by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50465908(CHEMBL4291048)
Affinity DataKi:  177nMAssay Description:Displacement of [3H]LSD from human 5-HT2B receptor expressed in HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50026066(1-(4,4-bis(4-fluorophenyl)butyl)-4-(4-chloro-3-(tr...)
Affinity DataKi:  184nMAssay Description:Displacement of [3H]LSD from human 5-HT2B receptor expressed in HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50465909(CHEMBL1644978)
Affinity DataKi:  194nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D2 receptor expressed in stable fibroblast cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50465909(CHEMBL1644978)
Affinity DataKi:  209nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D3 receptor expressed in HEK293T cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50465908(CHEMBL4291048)
Affinity DataKi:  252nMAssay Description:Displacement of [3H]Cimetidine from human H2 receptor expressed in HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50465911(CHEMBL1644980)
Affinity DataKi:  278nMAssay Description:Displacement of [3H]Cimetidine from human H2 receptor expressed in HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50026066(1-(4,4-bis(4-fluorophenyl)butyl)-4-(4-chloro-3-(tr...)
Affinity DataKi:  280nMAssay Description:Displacement of [3H]LSD from human 5-HT7A receptor expressed in HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50465908(CHEMBL4291048)
Affinity DataKi:  300nMAssay Description:Displacement of [3H]SCH23390 from human dopamine D1 receptor expressed in HEK293T cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50465912(CHEMBL4287623)
Affinity DataKi:  317nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D2 receptor expressed in stable fibroblast cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50465911(CHEMBL1644980)
Affinity DataKi:  326nMAssay Description:Displacement of [3H]LSD from human 5-HT7A receptor expressed in HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50465912(CHEMBL4287623)
Affinity DataKi:  328nMAssay Description:Displacement of [3H]DAMGO from human MOR expressed in HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50465909(CHEMBL1644978)
Affinity DataKi:  356nMAssay Description:Displacement of [3H]DAMGO from human MOR expressed in HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50026066(1-(4,4-bis(4-fluorophenyl)butyl)-4-(4-chloro-3-(tr...)
Affinity DataKi:  356nMAssay Description:Displacement of [3H]-Way100635 from human 5HT1A receptor expressed in stable CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50026066(1-(4,4-bis(4-fluorophenyl)butyl)-4-(4-chloro-3-(tr...)
Affinity DataKi:  361nMAssay Description:Displacement of [3H]Ketanserin from 5-HT2A receptor (unknown origin) by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50465911(CHEMBL1644980)
Affinity DataKi:  374nMAssay Description:Displacement of [3H]LSD from human 5-HT2B receptor expressed in HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50465909(CHEMBL1644978)
Affinity DataKi:  385nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D4 receptor by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50026066(1-(4,4-bis(4-fluorophenyl)butyl)-4-(4-chloro-3-(tr...)
Affinity DataKi:  401nMAssay Description:Displacement of [3H]Rauwolscine from human alpha 2B adrenergic receptor expressed in HEK293T cells by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50465907(CHEMBL4282702)
Affinity DataKi:  401nMAssay Description:Displacement of [3H]Cimetidine from human H2 receptor expressed in HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50465908(CHEMBL4291048)
Affinity DataKi:  402nMAssay Description:Displacement of [3H]Mesulergine from human 5-HT2C receptor expressed in HEK293FlpIN cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50465906(CHEMBL4293307)
Affinity DataKi:  417nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D2 receptor expressed in stable fibroblast cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50465909(CHEMBL1644978)
Affinity DataKi:  423nMAssay Description:Displacement of [3H]LSD from human 5-HT2B receptor expressed in HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50465909(CHEMBL1644978)
Affinity DataKi:  428nMAssay Description:Displacement of [3H]Citalopram from human SERT expressed in HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50465908(CHEMBL4291048)
Affinity DataKi:  437nMAssay Description:Displacement of [3H]SCH23390 from human dopamine D5 receptor expressed in HEK293T cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50465906(CHEMBL4293307)
Affinity DataKi:  437nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D3 receptor expressed in HEK293T cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50026066(1-(4,4-bis(4-fluorophenyl)butyl)-4-(4-chloro-3-(tr...)
Affinity DataKi:  445nMAssay Description:Displacement of [3H]Rauwolscine from human alpha 2C adrenergic receptor expressed in MDCK cells by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50465910(CHEMBL4278465)
Affinity DataKi:  458nMAssay Description:Displacement of [3H]Nisoxetine from human NET expressed in HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50465906(CHEMBL4293307)
Affinity DataKi:  459nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D4 receptor by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50465907(CHEMBL4282702)
Affinity DataKi:  460nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D2 receptor expressed in stable fibroblast cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50465908(CHEMBL4291048)
Affinity DataKi:  474nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D3 receptor expressed in HEK293T cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50465911(CHEMBL1644980)
Affinity DataKi:  481nMAssay Description:Displacement of [3H]-Way100635 from human 5HT1A receptor expressed in stable CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50465910(CHEMBL4278465)
Affinity DataKi:  509nMAssay Description:Displacement of [3H]LSD from human 5-HT2B receptor expressed in HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50026066(1-(4,4-bis(4-fluorophenyl)butyl)-4-(4-chloro-3-(tr...)
Affinity DataKi:  515nMAssay Description:Displacement of [3H]CGP12177 from human beta 3 adrenergic receptor expressed in HEK293FlpIN cells by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50465911(CHEMBL1644980)
Affinity DataKi:  518nMAssay Description:Displacement of [3H]Nisoxetine from human NET expressed in HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))
Texas Tech University Health Sciences Center

Curated by ChEMBL
LigandPNGBDBM50465912(CHEMBL4287623)
Affinity DataKi:  526nMAssay Description:Displacement of [3H]Cimetidine from human H2 receptor expressed in HEK cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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