Compile Data Set for Download or QSAR
maximum 50k data
Found 42 Enz. Inhib. hit(s) with all data for entry = 50035536
TargetAminopeptidase N(Sus scrofa (Pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50017478(Amastatin | CHEMBL28650 | Leu[1psi,CHOHCONH]ValVal...)
Affinity DataKi:  20nMAssay Description:Effect of inhibitor structure on the slow binding inhibition of Aminopeptidase M from porcine kidney was determined and Ki was reported which is obta...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50017478(Amastatin | CHEMBL28650 | Leu[1psi,CHOHCONH]ValVal...)
Affinity DataKi:  20nMAssay Description:Effect of inhibitor structure on the slow binding inhibition of aminopeptidase M was determined and Ki* was reported which is obtained by the equatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50027041(2-(3-Amino-2-hydroxy-5-methyl-hexanoylamino)-4-met...)
Affinity DataKi:  120nMAssay Description:Compound was evaluated for the inhibition of Leucine aminopeptidase and the inhibition constant was determined after preincubating the enzyme and inh...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50027042(3-Amino-2-hydroxy-5-methyl-hexanoic acid {2-methyl...)
Affinity DataKi:  180nMAssay Description:Compound was evaluated for the inhibition of Aminopeptidase M (AP-M) and the inhibition constant was determined after preincubating the enzyme and in...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50017478(Amastatin | CHEMBL28650 | Leu[1psi,CHOHCONH]ValVal...)
Affinity DataKi:  200nMAssay Description:Effect of inhibitor structure on the slow binding inhibition of Leucine aminopeptidase was determined and the Ki was reported which is = k2/k1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

TargetCytosol aminopeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50017478(Amastatin | CHEMBL28650 | Leu[1psi,CHOHCONH]ValVal...)
Affinity DataKi:  220nMAssay Description:Effect of inhibitor structure on the slow binding inhibition of aminopeptidase M was determined and Ki* was reported which is obtained by the equatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

TargetCytosol aminopeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50027043(3-Amino-2-hydroxy-N-(3-methyl-butyl)-4-phenyl-buty...)
Affinity DataKi:  500nMAssay Description:Compound was evaluated for the inhibition of Leucine aminopeptidase from porcine kidney and the inhibition constant was determined after preincubatin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50027042(3-Amino-2-hydroxy-5-methyl-hexanoic acid {2-methyl...)
Affinity DataKi:  890nMAssay Description:Compound was evaluated for the inhibition of Leucine aminopeptidase and the inhibition constant was determined after preincubating the enzyme and in...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50027046(2-[2-(3-Amino-2-hydroxy-5-methyl-hexanoylamino)-3-...)
Affinity DataKi:  900nMAssay Description:Effect of inhibitor structure on the slow binding inhibition of aminopeptidase M was determined and Ki* was reported which is obtained by the equatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50027046(2-[2-(3-Amino-2-hydroxy-5-methyl-hexanoylamino)-3-...)
Affinity DataKi:  940nMAssay Description:Compound was evaluated for the inhibitory activity against aminopeptidase MMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50027046(2-[2-(3-Amino-2-hydroxy-5-methyl-hexanoylamino)-3-...)
Affinity DataKi:  1.24E+3nMAssay Description:Compound was evaluated for the inhibition of Leucine aminopeptidase and the inhibition constant was determined after preincubating the enzyme and inh...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50017478(Amastatin | CHEMBL28650 | Leu[1psi,CHOHCONH]ValVal...)
Affinity DataKi:  2.00E+3nMAssay Description:Effect of inhibitor structure on the slow binding inhibition of aminopeptidase M was determined and the Ki was reported which is = k2/k1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50367209(BESTATIN HYDROCHLORIDE | Ubenimex)
Affinity DataKi:  4.10E+3nMAssay Description:Effect of inhibitor structure on the slow binding inhibition of aminopeptidase M was determined and Ki* was reported which is obtained by the equatio...More data for this Ligand-Target Pair
TargetAminopeptidase N(Sus scrofa (Pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50367209(BESTATIN HYDROCHLORIDE | Ubenimex)
Affinity DataKi:  4.10E+3nMAssay Description:Compound was evaluated for the inhibition of Aminopeptidase M (AP-M) and the inhibition constant was determined after preincubating the enzyme and in...More data for this Ligand-Target Pair
TargetAminopeptidase N(Sus scrofa (Pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50367209(BESTATIN HYDROCHLORIDE | Ubenimex)
Affinity DataKi:  7.00E+3nMAssay Description:Effect of inhibitor structure on the slow binding inhibition of aminopeptidase M was determined and the Ki was reported which is = k2/k1More data for this Ligand-Target Pair
TargetAminopeptidase N(Sus scrofa (Pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50027041(2-(3-Amino-2-hydroxy-5-methyl-hexanoylamino)-4-met...)
Affinity DataKi:  1.18E+4nMAssay Description:Compound was evaluated for the inhibition of Aminopeptidase M (AP-M) and the inhibition constant was determined after preincubating the enzyme and in...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50027043(3-Amino-2-hydroxy-N-(3-methyl-butyl)-4-phenyl-buty...)
Affinity DataKi:  1.60E+4nMAssay Description:Effect of inhibitor structure on the slow binding inhibition of aminopeptidase M was determined and Ki* was reported which is obtained by the equatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50027043(3-Amino-2-hydroxy-N-(3-methyl-butyl)-4-phenyl-buty...)
Affinity DataKi:  1.60E+4nMAssay Description:Compound was evaluated for the inhibition of Aminopeptidase M (AP-M) from porcine kidney and the inhibition constant was determined after preincubati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50027043(3-Amino-2-hydroxy-N-(3-methyl-butyl)-4-phenyl-buty...)
Affinity DataKi:  1.63E+4nMAssay Description:Compound was evaluated for the inhibition of Aminopeptidase M (AP-M) and the inhibition constant was determined after preincubating the enzyme and in...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50046325((S)-2-((2S,3S)-3-Amino-2-hydroxy-4-phenyl-butyryla...)
Affinity DataKi:  1.70E+4nMAssay Description:Compound was evaluated for the inhibition of Leucine aminopeptidase and the inhibition constant was determined after preincubating the enzyme and inh...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50017478(Amastatin | CHEMBL28650 | Leu[1psi,CHOHCONH]ValVal...)
Affinity DataKi:  2.00E+4nMAssay Description:Effect of inhibitor structure on the slow binding inhibition of aminopeptidase M was determined and the Ki was reported which is = k2/k1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

TargetCytosol aminopeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50367209(BESTATIN HYDROCHLORIDE | Ubenimex)
Affinity DataKi:  2.00E+4nMAssay Description:Compound was evaluated for the inhibition of Leucine aminopeptidase and the inhibition constant was determined after preincubating the enzyme and inh...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50027045(2-{2-[2-(3-Amino-2-hydroxy-5-methyl-hexanoylamino)...)
Affinity DataKi:  2.00E+4nMAssay Description:Effect of inhibitor structure on the slow binding inhibition of aminopeptidase M was determined and the Ki was reported which is = k2/k1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50027045(2-{2-[2-(3-Amino-2-hydroxy-5-methyl-hexanoylamino)...)
Affinity DataKi:  2.00E+4nMAssay Description:Effect of inhibitor structure on the slow binding inhibition of Aminopeptidase M from porcine kidney was determined and the Ki was reported which is ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50027045(2-{2-[2-(3-Amino-2-hydroxy-5-methyl-hexanoylamino)...)
Affinity DataKi: <2.30E+4nMAssay Description:Compound was evaluated for the inhibition of Aminopeptidase M (AP-M) and the inhibition constant was determined after preincubating the enzyme and in...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50027040(2-{2-[2-(3-Amino-5-methyl-hexanoylamino)-3-methyl-...)
Affinity DataKi:  2.50E+4nMAssay Description:Compound was evaluated for the inhibition of Aminopeptidase M (AP-M) and the inhibition constant was determined after preincubating the enzyme and in...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50027045(2-{2-[2-(3-Amino-2-hydroxy-5-methyl-hexanoylamino)...)
Affinity DataKi:  2.60E+4nMAssay Description:Compound was evaluated for the inhibitory activity against aminopeptidase MMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50027046(2-[2-(3-Amino-2-hydroxy-5-methyl-hexanoylamino)-3-...)
Affinity DataKi:  4.00E+4nMAssay Description:Effect of inhibitor structure on the slow binding inhibition of aminopeptidase M was determined and the Ki was reported which is = k2/k1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50027045(2-{2-[2-(3-Amino-2-hydroxy-5-methyl-hexanoylamino)...)
Affinity DataKi:  2.00E+5nMAssay Description:Effect of inhibitor structure on the slow binding inhibition of Leucine aminopeptidase was determined and the Ki was reported which is = k2/k1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50046325((S)-2-((2S,3S)-3-Amino-2-hydroxy-4-phenyl-butyryla...)
Affinity DataKi:  2.00E+5nMAssay Description:Effect of inhibitor structure on the slow binding inhibition of aminopeptidase M was determined and Ki* was reported which is obtained by the equatio...More data for this Ligand-Target Pair
TargetAminopeptidase N(Sus scrofa (Pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50046325((S)-2-((2S,3S)-3-Amino-2-hydroxy-4-phenyl-butyryla...)
Affinity DataKi:  5.00E+5nMAssay Description:Effect of inhibitor structure on the slow binding inhibition of aminopeptidase M was determined and the Ki was reported which is = k2/k1More data for this Ligand-Target Pair
TargetCytosol aminopeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50027040(2-{2-[2-(3-Amino-5-methyl-hexanoylamino)-3-methyl-...)
Affinity DataKi:  6.81E+5nMAssay Description:Compound was evaluated for the inhibition of Leucine aminopeptidase and the inhibition constant was determined after preincubating the enzyme and inh...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50027044(2-{2-[2-(2-Hydroxy-5-methyl-hexanoylamino)-3-methy...)
Affinity DataKi:  7.00E+5nMAssay Description:Compound was evaluated for the inhibition of Aminopeptidase M (AP-M) from porcine kidney and the inhibition constant was determined after preincubati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50027044(2-{2-[2-(2-Hydroxy-5-methyl-hexanoylamino)-3-methy...)
Affinity DataKi:  7.40E+5nMAssay Description:Compound was evaluated for the inhibition of Leucine aminopeptidase from porcine kidney and the inhibition constant was determined after preincubatin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50027047(4-Amino-3-hydroxy-6-methyl-heptanoic acid {2-methy...)
Affinity DataKi:  1.00E+6nMAssay Description:Compound was evaluated for the inhibition of Leucine aminopeptidase from porcine kidney and the inhibition constant was determined after preincubatin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50027047(4-Amino-3-hydroxy-6-methyl-heptanoic acid {2-methy...)
Affinity DataKi:  1.00E+6nMAssay Description:Compound was evaluated for the inhibition of Aminopeptidase M (AP-M) from porcine kidney and the inhibition constant was determined after preincubati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50027050(2-[2-(2-tert-Butoxycarbonylamino-3-methyl-butyryla...)
Affinity DataKi:  1.40E+6nMAssay Description:Compound was evaluated for the inhibition of Leucine aminopeptidase from porcine kidney and the inhibition constant was determined after preincubatin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50027045(2-{2-[2-(3-Amino-2-hydroxy-5-methyl-hexanoylamino)...)
Affinity DataKi:  2.00E+6nMAssay Description:Compound was evaluated for the inhibition of Aminopeptidase M (AP-M) and the inhibition constant was determined after preincubating the enzyme and in...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50027049(2-(3-Amino-2-methyl-4-phenyl-butyrylamino)-4-methy...)
Affinity DataKi:  3.78E+6nMAssay Description:Compound was evaluated for the inhibition of Leucine aminopeptidase and the inhibition constant was determined after preincubating the enzyme and inh...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50017478(Amastatin | CHEMBL28650 | Leu[1psi,CHOHCONH]ValVal...)
Affinity DataIC50:  1.10E+3nMAssay Description:Effect of inhibitor structure on the slow binding inhibition of Leucine aminopeptidase was determined and Ki* was reported which is obtained by the e...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Sus scrofa (Pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50367209(BESTATIN HYDROCHLORIDE | Ubenimex)
Affinity DataIC50:  3.03E+3nMAssay Description:Compound was evaluated for the inhibitory activity against aminopeptidase MMore data for this Ligand-Target Pair
TargetAminopeptidase N(Sus scrofa (Pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50027045(2-{2-[2-(3-Amino-2-hydroxy-5-methyl-hexanoylamino)...)
Affinity DataIC50: >5.00E+5nMAssay Description:Effect of inhibitor structure on the slow binding inhibition of aminopeptidase M was determined and the Ki was reported which is = k2/k1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed