Compile Data Set for Download or QSAR
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Found 22 Enz. Inhib. hit(s) with all data for entry = 50048624
LigandPNGBDBM50223637(Alphacemethadone | Alphacetylmethadol)
Affinity DataKi:  1.20nMAssay Description:Inhibition of [3H]- naloxone binding to Opioid receptors in rat brain membrane in the absence of NaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50223633(Levomethadone)
Affinity DataKi:  2nMAssay Description:Inhibition of [3H]- naloxone binding to Opioid receptors in rat brain membrane in the absence of NaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50223637(Alphacemethadone | Alphacetylmethadol)
Affinity DataKi:  3.40nMAssay Description:Compound was evaluated for the inhibition of [3H]- naloxone binding to Opioid receptors in rat brain membrane in the presence of NaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  6nMAssay Description:Inhibition of [3H]- naloxone binding to Opioid receptors in rat brain membrane in the absence of NaMore data for this Ligand-Target Pair
LigandPNGBDBM50223631(Betacetylmethadol)
Affinity DataKi:  15nMAssay Description:Inhibition of [3H]- naloxone binding to Opioid receptors in rat brain membrane in the absence of NaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50223633(Levomethadone)
Affinity DataKi:  77nMAssay Description:Compound was evaluated for the inhibition of [3H]- naloxone binding to Opioid receptors in rat brain membrane in the presence of NaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50223640((S)-Methadone | CHEMBL350719)
Affinity DataKi:  110nMAssay Description:Inhibition of [3H]- naloxone binding to Opioid receptors in rat brain membrane in the absence of NaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50223639(CHEMBL171118)
Affinity DataKi:  150nMAssay Description:Inhibition of [3H]- naloxone binding to Opioid receptors in rat brain membrane in the absence of NaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  190nMAssay Description:Compound was evaluated for the inhibition of [3H]- naloxone binding to Opioid receptors in rat brain membrane in the presence of NaMore data for this Ligand-Target Pair
LigandPNGBDBM50223632(Alphamethadol)
Affinity DataKi:  230nMAssay Description:Compound was evaluated for the inhibition of [3H]- naloxone opiate receptor binding using rat brain membrane in the absence of NaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50223632(Alphamethadol)
Affinity DataKi:  230nMAssay Description:Inhibition of [3H]- naloxone binding to Opioid receptors in rat brain membrane in the absence of NaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50223631(Betacetylmethadol)
Affinity DataKi:  450nMAssay Description:Compound was evaluated for the inhibition of [3H]- naloxone binding to Opioid receptors in rat brain membrane in the presence of NaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50223635(CHEMBL355396)
Affinity DataKi:  600nMAssay Description:Inhibition of [3H]- naloxone binding to Opioid receptors in rat brain membrane in the absence of NaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50223636(CHEMBL173964)
Affinity DataKi:  900nMAssay Description:Compound was evaluated for the inhibition of [3H]- naloxone Opioid receptors binding using rat brain membrane in the absence of NaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50223634(CHEMBL1325)
Affinity DataKi:  1.10E+3nMAssay Description:Inhibition of [3H]- naloxone binding to Opioid receptors in rat brain membrane in the absence of NaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50223638(CHEMBL367330)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition of [3H]- naloxone binding to Opioid receptors in rat brain membrane in the absence of NaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50223639(CHEMBL171118)
Affinity DataKi:  2.00E+3nMAssay Description:Compound was evaluated for the inhibition of [3H]- naloxone binding to Opioid receptors in rat brain membrane in the presence of NaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50223640((S)-Methadone | CHEMBL350719)
Affinity DataKi:  3.20E+3nMAssay Description:Compound was evaluated for the inhibition of [3H]- naloxone binding to Opioid receptors in rat brain membrane in the presence of NaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50223635(CHEMBL355396)
Affinity DataKi:  5.00E+3nMAssay Description:Compound was evaluated for the inhibition of [3H]- naloxone binding to Opioid receptors in rat brain membrane in the presence of NaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50223634(CHEMBL1325)
Affinity DataKi:  6.80E+3nMAssay Description:Compound was evaluated for the inhibition of [3H]- naloxone binding to Opioid receptors in rat brain membrane in the presence of NaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50223636(CHEMBL173964)
Affinity DataKi:  1.00E+4nMAssay Description:Compound was evaluated for the inhibition of [3H]- naloxone Opioid receptors binding using rat brain membrane in the presence of 100 mM NaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50223638(CHEMBL367330)
Affinity DataKi:  3.00E+4nMAssay Description:Compound was evaluated for the inhibition of [3H]- naloxone binding to Opioid receptors in rat brain membrane in the presence of NaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed