Compile Data Set for Download or QSAR
maximum 50k data
Found 86 Enz. Inhib. hit(s) with all data for entry = 50021157
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50176050(8-(3,4-dimethoxystyryl)-1,3-diethyl-7-methyl-1H-pu...)
Affinity DataKi:  5.01nMAssay Description:Displacement of [3H]MSX2 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50221683(9-(4-hydroxyphenethyl)-1,3-dimethyl-6,7,8,9-tetrah...)
Affinity DataKi:  230nMAssay Description:Displacement of [3H]MSX2 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50176050(8-(3,4-dimethoxystyryl)-1,3-diethyl-7-methyl-1H-pu...)
Affinity DataKi:  230nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50221697(1,3-dimethyl-9-phenethyl-6,7,8,9-tetrahydropyrimid...)
Affinity DataKi:  320nMAssay Description:Displacement of [3H]MSX2 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50221691(9-(2-(1H-indol-3-yl)ethyl)-1,3-dimethyl-6,7,8,9-te...)
Affinity DataKi:  330nMAssay Description:Displacement of [3H]MSX2 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50221703(9-(4-methoxyphenethyl)-1,3-dimethyl-6,7,8,9-tetrah...)
Affinity DataKi:  370nMAssay Description:Displacement of [3H]MSX2 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50221681(9-(4-chlorophenethyl)-1,3-dimethyl-6,7,8,9-tetrahy...)
Affinity DataKi:  480nMAssay Description:Displacement of [3H]MSX2 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50221694(9-phenethyl-1,3-dipropyl-6,7,8,9-tetrahydropyrimid...)
Affinity DataKi:  590nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50221694(9-phenethyl-1,3-dipropyl-6,7,8,9-tetrahydropyrimid...)
Affinity DataKi:  620nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50221683(9-(4-hydroxyphenethyl)-1,3-dimethyl-6,7,8,9-tetrah...)
Affinity DataKi:  630nMAssay Description:Displacement of [3H]MSX2 from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50221701(9-(3,4-dimethoxyphenethyl)-1,3-dipropyl-6,7,8,9-te...)
Affinity DataKi:  820nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50221694(9-phenethyl-1,3-dipropyl-6,7,8,9-tetrahydropyrimid...)
Affinity DataKi:  860nMAssay Description:Displacement of [3H]MSX2 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50221680(9-(2-(1H-indol-3-yl)ethyl)-1,3-dipropyl-6,7,8,9-te...)
Affinity DataKi:  900nMAssay Description:Displacement of [3H]MSX2 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50221698(9-(2-(benzyloxy)ethyl)-1,3-dimethyl-6,7,8,9-tetrah...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]PSB11 from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50221701(9-(3,4-dimethoxyphenethyl)-1,3-dipropyl-6,7,8,9-te...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]PSB11 from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50221680(9-(2-(1H-indol-3-yl)ethyl)-1,3-dipropyl-6,7,8,9-te...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]PSB11 from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50221693(1,3-dimethyl-9-(2-(p-tolyloxy)ethyl)-6,7,8,9-tetra...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]PSB11 from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50221690((E)-9-(2-(cinnamyloxy)ethyl)-1,3-dimethyl-6,7,8,9-...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]PSB11 from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50221684(CHEMBL239444 | N-(4-(2-(1,3-dimethyl-2,4-dioxo-1,2...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]PSB11 from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50221685(9-(2-(4-fluorobenzyloxy)ethyl)-1,3-dimethyl-6,7,8,...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]PSB11 from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50221687(2-(1,3-dimethyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyr...)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]MSX2 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50221702(9-(2-(2,4-dichlorophenoxy)ethyl)-1,3-dimethyl-6,7,...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]PSB11 from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50221702(9-(2-(2,4-dichlorophenoxy)ethyl)-1,3-dimethyl-6,7,...)
Affinity DataKi:  1.09E+3nMAssay Description:Displacement of [3H]MSX2 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50221682(1,3-dimethyl-9-(3-phenylpropyl)-6,7,8,9-tetrahydro...)
Affinity DataKi:  1.10E+3nMAssay Description:Displacement of [3H]MSX2 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50221695(9-(2-hydroxy-2-phenylethyl)-1,3-dimethyl-6,7,8,9-t...)
Affinity DataKi:  1.11E+3nMAssay Description:Displacement of [3H]MSX2 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50221704(9-(3,4-dimethoxyphenethyl)-1,3-dimethyl-6,7,8,9-te...)
Affinity DataKi:  1.21E+3nMAssay Description:Displacement of [3H]MSX2 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50221689(2-(1,3-dimethyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyr...)
Affinity DataKi:  1.22E+3nMAssay Description:Displacement of [3H]MSX2 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50221701(9-(3,4-dimethoxyphenethyl)-1,3-dipropyl-6,7,8,9-te...)
Affinity DataKi:  1.33E+3nMAssay Description:Displacement of [3H]MSX2 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50221705(9-(2-(4-chlorobenzyloxy)ethyl)-1,3-dimethyl-6,7,8,...)
Affinity DataKi:  1.33E+3nMAssay Description:Displacement of [3H]MSX2 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50221680(9-(2-(1H-indol-3-yl)ethyl)-1,3-dipropyl-6,7,8,9-te...)
Affinity DataKi:  1.79E+3nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50221682(1,3-dimethyl-9-(3-phenylpropyl)-6,7,8,9-tetrahydro...)
Affinity DataKi:  1.99E+3nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50221684(CHEMBL239444 | N-(4-(2-(1,3-dimethyl-2,4-dioxo-1,2...)
Affinity DataKi:  2.02E+3nMAssay Description:Displacement of [3H]MSX2 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50221700(9-(1-hydroxy-1-phenylpropan-2-yl)-1,3-dimethyl-6,7...)
Affinity DataKi:  2.16E+3nMAssay Description:Displacement of [3H]MSX2 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50221706(9-(2-(4-fluorobenzylamino)ethyl)-1,3-dimethyl-6,7,...)
Affinity DataKi:  2.63E+3nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50221697(1,3-dimethyl-9-phenethyl-6,7,8,9-tetrahydropyrimid...)
Affinity DataKi:  2.89E+3nMAssay Description:Displacement of [3H]MSX2 from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50221685(9-(2-(4-fluorobenzyloxy)ethyl)-1,3-dimethyl-6,7,8,...)
Affinity DataKi:  3.05E+3nMAssay Description:Displacement of [3H]MSX2 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50221698(9-(2-(benzyloxy)ethyl)-1,3-dimethyl-6,7,8,9-tetrah...)
Affinity DataKi:  3.16E+3nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50221689(2-(1,3-dimethyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyr...)
Affinity DataKi:  3.40E+3nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50221702(9-(2-(2,4-dichlorophenoxy)ethyl)-1,3-dimethyl-6,7,...)
Affinity DataKi:  3.50E+3nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50221685(9-(2-(4-fluorobenzyloxy)ethyl)-1,3-dimethyl-6,7,8,...)
Affinity DataKi:  3.68E+3nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50221698(9-(2-(benzyloxy)ethyl)-1,3-dimethyl-6,7,8,9-tetrah...)
Affinity DataKi:  3.69E+3nMAssay Description:Displacement of [3H]MSX2 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50221703(9-(4-methoxyphenethyl)-1,3-dimethyl-6,7,8,9-tetrah...)
Affinity DataKi:  3.85E+3nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50221686(9-(2-(4-chlorophenoxy)ethyl)-1,3-dimethyl-6,7,8,9-...)
Affinity DataKi:  4.22E+3nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50221690((E)-9-(2-(cinnamyloxy)ethyl)-1,3-dimethyl-6,7,8,9-...)
Affinity DataKi:  4.29E+3nMAssay Description:Displacement of [3H]MSX2 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50221691(9-(2-(1H-indol-3-yl)ethyl)-1,3-dimethyl-6,7,8,9-te...)
Affinity DataKi:  4.56E+3nMAssay Description:Displacement of [3H]MSX2 from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50221693(1,3-dimethyl-9-(2-(p-tolyloxy)ethyl)-6,7,8,9-tetra...)
Affinity DataKi:  4.60E+3nMAssay Description:Displacement of [3H]MSX2 from adenosine A2A receptor in rat brain striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50221681(9-(4-chlorophenethyl)-1,3-dimethyl-6,7,8,9-tetrahy...)
Affinity DataKi:  6.47E+3nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50221683(9-(4-hydroxyphenethyl)-1,3-dimethyl-6,7,8,9-tetrah...)
Affinity DataKi:  7.20E+3nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50221696(9-(2-(benzylamino)ethyl)-1,3-dimethyl-6,7,8,9-tetr...)
Affinity DataKi:  7.55E+3nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50221679(2-(1,3-dimethyl-2,4-dioxo-1,2,3,4,7,8-hexahydropyr...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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