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Found 54 Enz. Inhib. hit(s) with all data for entry = 50042390
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50425256(CHEMBL2315179)
Affinity DataIC50:  1nMAssay Description:Inhibition of rat SCD1 by rat microsomal assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50425259(CHEMBL2315473)
Affinity DataIC50:  3nMAssay Description:Inhibition of rat SCD1 by rat microsomal assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50425258(CHEMBL2315181)
Affinity DataIC50:  3nMAssay Description:Inhibition of rat SCD1 by rat microsomal assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50425257(CHEMBL2315472)
Affinity DataIC50:  4nMAssay Description:Inhibition of rat SCD1 by rat microsomal assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50425266(CHEMBL2315480)
Affinity DataIC50:  4nMAssay Description:Inhibition of rat SCD1 by rat microsomal assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50425255(CHEMBL2315180)
Affinity DataIC50:  8nMAssay Description:Inhibition of rat SCD1 by rat microsomal assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50425261(CHEMBL2315475)
Affinity DataIC50:  10nMAssay Description:Inhibition of rat SCD1 by rat microsomal assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50425265(CHEMBL2315479)
Affinity DataIC50:  12nMAssay Description:Inhibition of rat SCD1 by rat microsomal assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50425283(CHEMBL2315498)
Affinity DataIC50:  17nMAssay Description:Inhibition of rat SCD1 by rat microsomal assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50425277(CHEMBL2315490)
Affinity DataIC50:  19nMAssay Description:Inhibition of rat SCD1 by rat microsomal assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50425289(CHEMBL2315503)
Affinity DataIC50:  32nMAssay Description:Inhibition of rat SCD1 by rat microsomal assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50425267(CHEMBL2315481)
Affinity DataIC50:  40nMAssay Description:Inhibition of rat SCD1 by rat microsomal assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50425284(CHEMBL2315497)
Affinity DataIC50:  42nMAssay Description:Inhibition of rat SCD1 by rat microsomal assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50425285(CHEMBL2315496)
Affinity DataIC50:  57nMAssay Description:Inhibition of rat SCD1 by rat microsomal assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50425262(CHEMBL2315476)
Affinity DataIC50:  130nMAssay Description:Inhibition of rat SCD1 by rat microsomal assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50425275(CHEMBL2315488)
Affinity DataIC50:  140nMAssay Description:Inhibition of rat SCD1 by rat microsomal assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50425272(CHEMBL2315486)
Affinity DataIC50:  180nMAssay Description:Inhibition of rat SCD1 by rat microsomal assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50425280(CHEMBL2315493)
Affinity DataIC50:  350nMAssay Description:Inhibition of rat SCD1 by rat microsomal assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50425276(CHEMBL2315491)
Affinity DataIC50:  380nMAssay Description:Inhibition of rat SCD1 by rat microsomal assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50425295(CHEMBL2315509)
Affinity DataIC50:  430nMAssay Description:Inhibition of rat SCD1 by rat microsomal assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50425269(CHEMBL2315483)
Affinity DataIC50:  440nMAssay Description:Inhibition of rat SCD1 by rat microsomal assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50425288(CHEMBL2315504)
Affinity DataIC50:  460nMAssay Description:Inhibition of rat SCD1 by rat microsomal assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50425290(CHEMBL2315502)
Affinity DataIC50:  680nMAssay Description:Inhibition of rat SCD1 by rat microsomal assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50425292(CHEMBL2315500)
Affinity DataIC50:  830nMAssay Description:Inhibition of rat SCD1 by rat microsomal assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50425263(CHEMBL2315477)
Affinity DataIC50:  930nMAssay Description:Inhibition of rat SCD1 by rat microsomal assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50425286(CHEMBL2315495)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of rat SCD1 by rat microsomal assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50425303(CHEMBL2315513)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of rat SCD1 by rat microsomal assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50425297(CHEMBL2315507)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of rat SCD1 by rat microsomal assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50425296(CHEMBL2315508)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of rat SCD1 by rat microsomal assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50425278(CHEMBL2315489)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of rat SCD1 by rat microsomal assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50425299(CHEMBL2315517)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of rat SCD1 by rat microsomal assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50425291(CHEMBL2315501)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of rat SCD1 by rat microsomal assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50330381(5-Fluoro-1'-{6-[5-(pyridin-3-ylmethyl)-1,3,4-oxadi...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of rat SCD1 by rat microsomal assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50425264(CHEMBL2315478)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of rat SCD1 by rat microsomal assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50425271(CHEMBL2315485)
Affinity DataIC50:  2.45E+3nMAssay Description:Inhibition of rat SCD1 by rat microsomal assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50425279(CHEMBL2315494)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of rat SCD1 by rat microsomal assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50425294(CHEMBL2315510)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of rat SCD1 by rat microsomal assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50425253(CHEMBL2315519)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of rat SCD1 by rat microsomal assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50425268(CHEMBL2315482)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibition of rat SCD1 by rat microsomal assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50425260(CHEMBL2315474)
Affinity DataIC50:  4.70E+3nMAssay Description:Inhibition of rat SCD1 by rat microsomal assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50425270(CHEMBL2315484)
Affinity DataIC50:  5.90E+3nMAssay Description:Inhibition of rat SCD1 by rat microsomal assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50425273(CHEMBL2315512)
Affinity DataIC50:  6.40E+3nMAssay Description:Inhibition of mouse SCD1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50425274(CHEMBL2315487)
Affinity DataIC50:  8.20E+3nMAssay Description:Inhibition of rat SCD1 by rat microsomal assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50425300(CHEMBL2315516)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of rat SCD1 by rat microsomal assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50425298(CHEMBL2315506)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of rat SCD1 by rat microsomal assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50425293(CHEMBL2315511)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of rat SCD1 by rat microsomal assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50425287(CHEMBL2315505)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of rat SCD1 by rat microsomal assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50425282(CHEMBL2315499)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of rat SCD1 by rat microsomal assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50425281(CHEMBL2315492)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of rat SCD1 by rat microsomal assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50425301(CHEMBL2315515)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of rat SCD1 by rat microsomal assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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