Compile Data Set for Download or QSAR
maximum 50k data
Found 4 Enz. Inhib. hit(s) with all data for entry = 50005813
TargetSterol O-acyltransferase 1(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50041289((S)-2-Hexylsulfanyl-decanoic acid (6-methyl-2,4-bi...)
Affinity DataIC50:  22nMAssay Description:In vitro potency was determined using Acyl coenzyme A:cholesterol acyltransferase in liver microsomes from ratsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50041290((S)-2-Hexylsulfanyl-decanoic acid (6-methylsulfany...)
Affinity DataIC50:  135nMAssay Description:In vitro potency was determined using Acyl coenzyme A:cholesterol acyltransferase in liver microsomes from ratsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50453642(CHEMBL2093028)
Affinity DataIC50:  160nMAssay Description:In vitro potency was determined using Acyl coenzyme A:cholesterol acyltransferase in liver microsomes from ratsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50453641(CHEMBL2093029)
Affinity DataIC50:  750nMAssay Description:In vitro potency was determined using Acyl coenzyme A:cholesterol acyltransferase in liver microsomes from ratsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed