Compile Data Set for Download or QSAR
maximum 50k data
Found 36 Enz. Inhib. hit(s) with all data for entry = 50027007
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50264364(CHEMBL491229 | trans-4-[5-(4-Fluoro-phenyl)-1H-ben...)
Affinity DataIC50:  1.70nMAssay Description:Displacement of [125I]PYY from human recombinant NPYY5 receptor expressed in mouse LMtk cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50264493(CHEMBL489608 | trans-4-[5-(5-Trifluoromethyl-[1,2,...)
Affinity DataIC50:  2.10nMAssay Description:Displacement of [125I]PYY from human recombinant NPYY5 receptor expressed in mouse LMtk cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50264441(CHEMBL491239 | trans-6-Chloro-2-(3'-oxo-3'H-spiro[...)
Affinity DataIC50:  2.20nMAssay Description:Displacement of [125I]PYY from human recombinant NPYY5 receptor expressed in mouse LMtk cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50264395(CHEMBL490824 | trans-4-(5-Chloro-6-phenyl-1H-benzo...)
Affinity DataIC50:  2.20nMAssay Description:Displacement of [125I]PYY from human recombinant NPYY5 receptor expressed in mouse LMtk cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50264328(CHEMBL489587 | trans-4-(5-Phenyl-1H-benzoimidazol-...)
Affinity DataIC50:  2.30nMAssay Description:Displacement of [125I]PYY from human recombinant NPYY5 receptor expressed in mouse LMtk cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50264366(CHEMBL491427 | trans-4-(5-Pyridin-2-yl-1H-benzoimi...)
Affinity DataIC50:  2.40nMAssay Description:Displacement of [125I]PYY from human recombinant NPYY5 receptor expressed in mouse LMtk cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50264365(CHEMBL491230 | trans-4-(5-Benzoyl-1H-benzoimidazol...)
Affinity DataIC50:  2.40nMAssay Description:Displacement of [125I]PYY from human recombinant NPYY5 receptor expressed in mouse LMtk cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50264394(CHEMBL455815 | trans-4-(5-Chloro-6-trifluoromethyl...)
Affinity DataIC50:  2.60nMAssay Description:Displacement of [125I]PYY from human recombinant NPYY5 receptor expressed in mouse LMtk cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50264367(CHEMBL521959 | trans-4-(5-Pyridin-3-yl-1H-benzoimi...)
Affinity DataIC50:  3.10nMAssay Description:Displacement of [125I]PYY from human recombinant NPYY5 receptor expressed in mouse LMtk cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50264444(CHEMBL490427 | trans-4-[5-(5-Methyl-[1,3,4]oxadiaz...)
Affinity DataIC50:  3.30nMAssay Description:Displacement of [125I]PYY from human recombinant NPYY5 receptor expressed in mouse LMtk cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50264442(CHEMBL491436 | trans-4-Chloro-2-(3'-oxo-3'H-spiro[...)
Affinity DataIC50:  4.5nMAssay Description:Displacement of [125I]PYY from human recombinant NPYY5 receptor expressed in mouse LMtk cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50264492(CHEMBL522589 | trans-4-[5-(5-Methyl-[1,2,4]oxadiaz...)
Affinity DataIC50:  5.10nMAssay Description:Displacement of [125I]PYY from human recombinant NPYY5 receptor expressed in mouse LMtk cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50264444(CHEMBL490427 | trans-4-[5-(5-Methyl-[1,3,4]oxadiaz...)
Affinity DataIC50:  5.5nMAssay Description:Antagonist activity at human recombinant NPYY5 receptor expressed in mouse LMtk cells assessed as inhibition of NPY-induced calcium increaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50264494(CHEMBL521750 | trans-4-[5-(2-Methyl-2H-tetrazol-5-...)
Affinity DataIC50:  5.90nMAssay Description:Displacement of [125I]PYY from human recombinant NPYY5 receptor expressed in mouse LMtk cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50264492(CHEMBL522589 | trans-4-[5-(5-Methyl-[1,2,4]oxadiaz...)
Affinity DataIC50:  7nMAssay Description:Antagonist activity at human recombinant NPYY5 receptor expressed in mouse LMtk cells assessed as inhibition of NPY-induced calcium increaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50264494(CHEMBL521750 | trans-4-[5-(2-Methyl-2H-tetrazol-5-...)
Affinity DataIC50:  7.20nMAssay Description:Antagonist activity at human recombinant NPYY5 receptor expressed in mouse LMtk cells assessed as inhibition of NPY-induced calcium increaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50264397(CHEMBL522768 | trans-2-(3'-Oxo-3'H-spiro[cyclohex-...)
Affinity DataIC50:  7.70nMAssay Description:Displacement of [125I]PYY from human recombinant NPYY5 receptor expressed in mouse LMtk cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50264393(CHEMBL522788 | trans-4-(5,6-Dichloro-1H-benzoimida...)
Affinity DataIC50:  8nMAssay Description:Displacement of [125I]PYY from human recombinant NPYY5 receptor expressed in mouse LMtk cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50264443(CHEMBL522609 | trans-4-(5-[1,3,4]Oxadiazol-2-yl-1H...)
Affinity DataIC50:  15nMAssay Description:Displacement of [125I]PYY from human recombinant NPYY5 receptor expressed in mouse LMtk cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50264324(CHEMBL490608 | trans-2-(3'-Oxo-3'H-spiro[cyclohex-...)
Affinity DataIC50:  20nMAssay Description:Displacement of [125I]PYY from human recombinant NPYY5 receptor expressed in mouse LMtk cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50264325(CHEMBL523964 | trans-4-(5-Chloro-1H-benzoimidazol-...)
Affinity DataIC50:  39nMAssay Description:Displacement of [125I]PYY from human recombinant NPYY5 receptor expressed in mouse LMtk cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50264327(CHEMBL523943 | trans-4-(5-Bromo-1H-benzoimidazol-2...)
Affinity DataIC50:  45nMAssay Description:Displacement of [125I]PYY from human recombinant NPYY5 receptor expressed in mouse LMtk cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50264326(CHEMBL452726 | trans-4-(5-Trifluoromethyl-1H-benzo...)
Affinity DataIC50:  47nMAssay Description:Displacement of [125I]PYY from human recombinant NPYY5 receptor expressed in mouse LMtk cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50264295(CHEMBL491020 | trans-4-(1H-Benzoimidazol-2-yl)-spi...)
Affinity DataIC50:  91nMAssay Description:Displacement of [125I]PYY from human recombinant NPYY5 receptor expressed in mouse LMtk cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50264396(CHEMBL489806 | trans-4-(5,6-Dichloro-1-methyl-1H-b...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [125I]PYY from human recombinant NPYY5 receptor expressed in mouse LMtk cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50264495(CHEMBL489609 | cis-6-Chloro-2-(3'-oxo-3'H-spiro[cy...)
Affinity DataIC50:  1.00E+3nMAssay Description:Displacement of [125I]PYY from human recombinant NPYY5 receptor expressed in mouse LMtk cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50264528(CHEMBL483239 | cis-4-[5-(5-Methyl-[1,3,4]oxadiazol...)
Affinity DataIC50:  1.00E+3nMAssay Description:Displacement of [125I]PYY from human recombinant NPYY5 receptor expressed in mouse LMtk cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50264494(CHEMBL521750 | trans-4-[5-(2-Methyl-2H-tetrazol-5-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of NPYY2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50264492(CHEMBL522589 | trans-4-[5-(5-Methyl-[1,2,4]oxadiaz...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of NPYY2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 4(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50264494(CHEMBL521750 | trans-4-[5-(2-Methyl-2H-tetrazol-5-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of NPYY4 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 4(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50264492(CHEMBL522589 | trans-4-[5-(5-Methyl-[1,2,4]oxadiaz...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of NPYY4 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50264494(CHEMBL521750 | trans-4-[5-(2-Methyl-2H-tetrazol-5-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of NPYY1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 4(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50264444(CHEMBL490427 | trans-4-[5-(5-Methyl-[1,3,4]oxadiaz...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of NPYY4 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50264444(CHEMBL490427 | trans-4-[5-(5-Methyl-[1,3,4]oxadiaz...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of NPYY2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50264444(CHEMBL490427 | trans-4-[5-(5-Methyl-[1,3,4]oxadiaz...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of NPYY1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50264492(CHEMBL522589 | trans-4-[5-(5-Methyl-[1,2,4]oxadiaz...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of NPYY1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed