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Found 16 Enz. Inhib. hit(s) with all data for entry = 50043203
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50437341(WITHANOLIDE E)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of TNFalpha-induced IkappaBalpha (unknown origin) phosphorylation expressed in human HeLa cells pretreated 30 mins before TNFalpha additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50437352(CHEMBL2408033)
Affinity DataIC50:  2.62E+4nMAssay Description:Inhibition of TNFalpha-induced IkappaBalpha (unknown origin) phosphorylation expressed in human HeLa cells pretreated 30 mins before TNFalpha additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50378033(PHYSALIN F)
Affinity DataIC50:  2.71E+4nMAssay Description:Inhibition of TNFalpha-induced IkappaBalpha (unknown origin) phosphorylation expressed in human HeLa cells pretreated 30 mins before TNFalpha additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50437349(25-HYDROXY PHYSALIN F)
Affinity DataIC50:  3.01E+4nMAssay Description:Inhibition of TNFalpha-induced IkappaBalpha (unknown origin) phosphorylation expressed in human HeLa cells pretreated 30 mins before TNFalpha additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50378034(CHEMBL504404 | NSC-287088 | PHYSALIN B)
Affinity DataIC50:  3.75E+4nMAssay Description:Inhibition of TNFalpha-induced IkappaBalpha (unknown origin) phosphorylation expressed in human HeLa cells pretreated 30 mins before TNFalpha additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50437346(CHEMBL2408037)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of TNFalpha-induced IkappaBalpha (unknown origin) phosphorylation expressed in human HeLa cells pretreated 30 mins before TNFalpha additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50437347(PHYSALIN J)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of TNFalpha-induced IkappaBalpha (unknown origin) phosphorylation expressed in human HeLa cells pretreated 30 mins before TNFalpha additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50437348(25-HYDROXY PHYSALIN J)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of TNFalpha-induced IkappaBalpha (unknown origin) phosphorylation expressed in human HeLa cells pretreated 30 mins before TNFalpha additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50437350(CHEMBL2408034)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of TNFalpha-induced IkappaBalpha (unknown origin) phosphorylation expressed in human HeLa cells pretreated 30 mins before TNFalpha additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50437351(PHYSALIN A)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of TNFalpha-induced IkappaBalpha (unknown origin) phosphorylation expressed in human HeLa cells pretreated 30 mins before TNFalpha additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50437345(PHYSALIN O)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of TNFalpha-induced IkappaBalpha (unknown origin) phosphorylation expressed in human HeLa cells pretreated 30 mins before TNFalpha additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50437344(WITHANOLIDE F)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of TNFalpha-induced IkappaBalpha (unknown origin) phosphorylation expressed in human HeLa cells pretreated 30 mins before TNFalpha additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50437343(CHEMBL2333678)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of TNFalpha-induced IkappaBalpha (unknown origin) phosphorylation expressed in human HeLa cells pretreated 30 mins before TNFalpha additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50437342(CHEMBL2333675)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of TNFalpha-induced IkappaBalpha (unknown origin) phosphorylation expressed in human HeLa cells pretreated 30 mins before TNFalpha additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50437339(CHEMBL2408039)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of TNFalpha-induced IkappaBalpha (unknown origin) phosphorylation expressed in human HeLa cells pretreated 30 mins before TNFalpha additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNF-kappa-B inhibitor alpha(Homo sapiens (Human))
Riken

Curated by ChEMBL
LigandPNGBDBM50437340(CHEMBL2408038)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of TNFalpha-induced IkappaBalpha (unknown origin) phosphorylation expressed in human HeLa cells pretreated 30 mins before TNFalpha additio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed