Affinity DataIC50: 85nMAssay Description:In vitro 5-lipoxygenase inhibitory activity against A-23,187-stimulated conversion of [14C]-AA to 5-HETE in guinea pig peritoneal polymorphonuclear l...More data for this Ligand-Target Pair
Affinity DataIC50: 97nMAssay Description:In vitro 5-lipoxygenaseinhibitory activity against A-23,187-stimulated conversion of [14C]-AA to LTB4 in guinea pig peritoneal polymorphonuclear leuk...More data for this Ligand-Target Pair
Affinity DataIC50: 98nMAssay Description:In vitro 5-lipoxygenase inhibitory activity against A-23,187-stimulated conversion of [14C]-AA to 5-HETE in guinea pig peritoneal polymorphonuclear l...More data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:In vitro 5-lipoxygenase inhibitory activity against A-23,187-stimulated conversion of [14C]-AA to 5-HETE in guinea pig peritoneal polymorphonuclear l...More data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:In vitro 5-lipoxygenase inhibitory activity against A-23,187-stimulated conversion of [14C]-AA to LTB4 in guinea pig peritoneal polymorphonuclear leu...More data for this Ligand-Target Pair
Affinity DataIC50: 120nMAssay Description:In vitro 5-lipoxygenase inhibitory activity against A-23,187-stimulated conversion of [14C]-AA to 5-HETE in guinea pig peritoneal polymorphonuclear l...More data for this Ligand-Target Pair
Affinity DataIC50: 120nMAssay Description:In vitro 5-lipoxygenase inhibitory activity against A-23,187-stimulated conversion of [14C]-AA to LTB4 in guinea pig peritoneal polymorphonuclear leu...More data for this Ligand-Target Pair
Affinity DataIC50: 140nMAssay Description:In vitro 5-lipoxygenase inhibitory activity against A-23,187-stimulated conversion of [14C]-AA to LTB4 in guinea pig peritoneal polymorphonuclear leu...More data for this Ligand-Target Pair
Affinity DataIC50: 170nMAssay Description:In vitro 5-lipoxygenase inhibitory activity against A-23,187-stimulated conversion of [14C]-AA to LTB4 in guinea pig peritoneal polymorphonuclear leu...More data for this Ligand-Target Pair
Affinity DataIC50: 180nMAssay Description:In vitro 5-lipoxygenase inhibitory activity against A-23,187-stimulated conversion of [14C]-AA to 5-HETE in guinea pig peritoneal polymorphonuclear l...More data for this Ligand-Target Pair
Affinity DataIC50: 390nMAssay Description:Ex vivo inhibition of 5-lipoxygenase was determined by the measurement of A-23,187-stimulated LTB4 production in dog blood at 12 h, following intrave...More data for this Ligand-Target Pair
Affinity DataIC50: 420nMAssay Description:In vitro 5-lipoxygenase inhibitory activity against A-23,187-stimulated conversion of [14C]-AA to LTB4 in guinea pig peritoneal polymorphonuclear leu...More data for this Ligand-Target Pair
Affinity DataIC50: 450nMAssay Description:In vitro 5-lipoxygenase inhibitory activity against A-23,187-stimulated conversion of [14C]-AA to LTB4 in guinea pig peritoneal polymorphonuclear leu...More data for this Ligand-Target Pair
Affinity DataIC50: 480nMAssay Description:In vitro 5-lipoxygenase inhibitory activity against A-23,187-stimulated conversion of [14C]-AA to 5-HETE in guinea pig peritoneal polymorphonuclear l...More data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+3nMAssay Description:In vitro 5-lipoxygenase inhibitory activity against A-23,187-stimulated conversion of [14C]-AA to 5-HETE in guinea pig peritoneal polymorphonuclear l...More data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+3nMAssay Description:In vitro 5-lipoxygenase inhibitory activity against A-23,187-stimulated conversion of [14C]-AA to LTB4 in guinea pig peritoneal polymorphonuclear leu...More data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+3nMAssay Description:In vitro 5-lipoxygenase inhibitory activity against A-23,187-stimulated conversion of [14C]-AA to 5-HETE in guinea pig peritoneal polymorphonuclear l...More data for this Ligand-Target Pair
Affinity DataIC50: 2.20E+3nMAssay Description:In vitro 5-lipoxygenase inhibitory activity against A-23,187-stimulated conversion of [14C]-AA to LTB4 in guinea pig peritoneal polymorphonuclear leu...More data for this Ligand-Target Pair
Affinity DataIC50: 2.70E+3nMAssay Description:In vitro 5-lipoxygenase inhibitory activity against A-23,187-stimulated conversion of [14C]-AA to 5-HETE in guinea pig peritoneal polymorphonuclear l...More data for this Ligand-Target Pair
Affinity DataIC50: 2.90E+3nMAssay Description:In vitro 5-lipoxygenase inhibitory activity against A-23,187-stimulated conversion of [14C]-AA to LTB4 in guinea pig peritoneal polymorphonuclear leu...More data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+3nMAssay Description:In vitro 5-lipoxygenase inhibitory activity against A-23,187-stimulated conversion of [14C]-AA to 5-HETE in guinea pig peritoneal polymorphonuclear l...More data for this Ligand-Target Pair
Affinity DataIC50: 6.00E+3nMAssay Description:In vitro 5-lipoxygenase inhibitory activity against A-23,187-stimulated conversion of [14C]-AA to LTB4 in guinea pig peritoneal polymorphonuclear leu...More data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+4nMAssay Description:In vitro 5-lipoxygenase inhibitory activity against A-23,187-stimulated conversion of [14C]-AA to LTB4 in guinea pig peritoneal polymorphonuclear leu...More data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+4nMAssay Description:In vitro 5-lipoxygenase inhibitory activity against A-23,187-stimulated conversion of [14C]-AA to 5-HETE in guinea pig peritoneal polymorphonuclear l...More data for this Ligand-Target Pair