Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with all data for entry = 50033666
TargetCannabinoid receptor 2(Homo sapiens (Human))
Imir K.U. Leuven

Curated by ChEMBL
LigandPNGBDBM50349311(CHEMBL1807841)
Affinity DataKi:  27nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cells after 1 hrs by beta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Imir K.U. Leuven

Curated by ChEMBL
LigandPNGBDBM50349311(CHEMBL1807841)
Affinity DataKi:  1.00E+4nMAssay Description:Displacement of [3H]-SR141716A from human CB1 receptor expressed in CHO cells after 1 hrs by beta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Imir K.U. Leuven

Curated by ChEMBL
LigandPNGBDBM50349311(CHEMBL1807841)
Affinity DataEC50:  17.9nMAssay Description:Inverse agonist activity at human CB2 receptor expressed in CHO cells assessed as effect on [35S]-GTPgammaS binding after 1 hrs by beta countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed