Compile Data Set for Download or QSAR
maximum 50k data
Found 42 Enz. Inhib. hit(s) with all data for entry = 50000284
TargetAdenosine receptor A1(GUINEA PIG)
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50421971(CHEMBL611917)
Affinity DataEC50:  2.57E+4nMAssay Description:In vitro prolonging of the stimulus-QRS interval in guinea pig heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50421971(CHEMBL611917)
Affinity DataEC50:  7.40nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(GUINEA PIG)
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50421973(CHEMBL610727)
Affinity DataEC50:  2.51E+4nMAssay Description:In vitro prolonging of the stimulus-QRS interval in guinea pig heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(GUINEA PIG)
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50421974(CHEMBL607873)
Affinity DataEC50:  3.63E+3nMAssay Description:In vitro prolonging of the stimulus-QRS interval in guinea pig heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(GUINEA PIG)
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50421975(CHEMBL611607)
Affinity DataEC50:  7.24E+3nMAssay Description:In vitro prolonging of the stimulus-QRS interval in guinea pig heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(GUINEA PIG)
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50421976(CHEMBL607796)
Affinity DataEC50:  1.74E+4nMAssay Description:In vitro prolonging of the stimulus-QRS interval in guinea pig heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(GUINEA PIG)
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50009509((CGS 22,492) 2-[6-Amino-2-(2-cyclohexyl-ethylamino...)
Affinity DataEC50:  1.23E+4nMAssay Description:In vitro prolonging of the stimulus-QRS interval in guinea pig heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(GUINEA PIG)
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50421977(CHEMBL609231)
Affinity DataEC50:  1.35E+4nMAssay Description:In vitro prolonging of the stimulus-QRS interval in guinea pig heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(GUINEA PIG)
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50421978(CHEMBL611314)
Affinity DataEC50:  1.10E+4nMAssay Description:In vitro prolonging of the stimulus-QRS interval in guinea pig heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(GUINEA PIG)
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50421979(CHEMBL607585)
Affinity DataEC50:  1.15E+4nMAssay Description:In vitro prolonging of the stimulus-QRS interval in guinea pig heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(GUINEA PIG)
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50421980(CHEMBL2113592)
Affinity DataEC50:  2.09E+4nMAssay Description:In vitro prolonging of the stimulus-QRS interval in guinea pig heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(GUINEA PIG)
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50421981(CHEMBL607877)
Affinity DataEC50:  1.20E+4nMAssay Description:In vitro prolonging of the stimulus-QRS interval in guinea pig heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(GUINEA PIG)
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50009535((CGS 22,989) 2-[6-Amino-2-(2-cyclohex-1-enyl-ethyl...)
Affinity DataEC50:  2.29E+4nMAssay Description:In vitro prolonging of the stimulus-QRS interval in guinea pig heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(GUINEA PIG)
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50421982(CHEMBL608663)
Affinity DataEC50:  9.77E+3nMAssay Description:In vitro prolonging of the stimulus-QRS interval in guinea pig heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(GUINEA PIG)
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50421983(CHEMBL608966)
Affinity DataEC50:  6.61E+4nMAssay Description:In vitro prolonging of the stimulus-QRS interval in guinea pig heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(GUINEA PIG)
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50421984(CHEMBL607599)
Affinity DataEC50:  1.26E+4nMAssay Description:In vitro prolonging of the stimulus-QRS interval in guinea pig heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(GUINEA PIG)
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50421985(CHEMBL611916)
Affinity DataEC50:  2.51E+4nMAssay Description:In vitro prolonging of the stimulus-QRS interval in guinea pig heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(GUINEA PIG)
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50421986(CHEMBL610443)
Affinity DataEC50:  2.04E+4nMAssay Description:In vitro prolonging of the stimulus-QRS interval in guinea pig heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(GUINEA PIG)
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50368478(CHEMBL610444)
Affinity DataEC50:  2.00E+4nMAssay Description:In vitro prolonging of the stimulus-QRS interval in guinea pig heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(GUINEA PIG)
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50421987(CHEMBL611919)
Affinity DataEC50:  8.91E+3nMAssay Description:In vitro prolonging of the stimulus-QRS interval in guinea pig heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50009509((CGS 22,492) 2-[6-Amino-2-(2-cyclohexyl-ethylamino...)
Affinity DataEC50:  1.90nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50230152(Binodenoson | Corvue | MRE0470 | WRC-0470)
Affinity DataEC50:  0.257nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50421987(CHEMBL611919)
Affinity DataEC50:  178nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50421976(CHEMBL607796)
Affinity DataEC50:  3.5nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50421980(CHEMBL2113592)
Affinity DataEC50:  0.468nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50421972(CHEMBL611921)
Affinity DataEC50:  2nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50421982(CHEMBL608663)
Affinity DataEC50:  0.692nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50421983(CHEMBL608966)
Affinity DataEC50:  1.80nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50421975(CHEMBL611607)
Affinity DataEC50:  0.324nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50009535((CGS 22,989) 2-[6-Amino-2-(2-cyclohex-1-enyl-ethyl...)
Affinity DataEC50:  2.20nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(GUINEA PIG)
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50230152(Binodenoson | Corvue | MRE0470 | WRC-0470)
Affinity DataEC50:  3.55E+3nMAssay Description:In vitro prolonging of the stimulus-QRS interval in guinea pig heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50368478(CHEMBL610444)
Affinity DataEC50:  79nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50421985(CHEMBL611916)
Affinity DataEC50:  1nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50421986(CHEMBL610443)
Affinity DataEC50:  3.30nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50421984(CHEMBL607599)
Affinity DataEC50:  7.40nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50421977(CHEMBL609231)
Affinity DataEC50:  13nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50421973(CHEMBL610727)
Affinity DataEC50:  35nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50421979(CHEMBL607585)
Affinity DataEC50:  2.90nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50421981(CHEMBL607877)
Affinity DataEC50:  50nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50421978(CHEMBL611314)
Affinity DataEC50:  5.80nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50421974(CHEMBL607873)
Affinity DataEC50:  76nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(GUINEA PIG)
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50421972(CHEMBL611921)
Affinity DataEC50:  1.66E+4nMAssay Description:In vitro prolonging of the stimulus-QRS interval in guinea pig heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed