Compile Data Set for Download or QSAR
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Found 49 Enz. Inhib. hit(s) with all data for entry = 50045143
LigandPNGBDBM50362741(CHEMBL1939826)
Affinity DataIC50:  19nMAssay Description:Antagonist activity at rat TRPA1 assessed as inhibition of AITC-induced calcium uptake by [45Ca2+] fluorimetry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50362741(CHEMBL1939826)
Affinity DataIC50:  26nMAssay Description:Antagonist activity at human TRPA1 assessed as inhibition of AITC-induced calcium uptake by [45Ca2+] fluorimetry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50046740(CHEMBL1939972 | US9186360, 90)
Affinity DataIC50:  28nMAssay Description:Antagonist activity at rat TRPA1 assessed as inhibition of AITC-induced calcium uptake by [45Ca2+] fluorimetry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50046740(CHEMBL1939972 | US9186360, 90)
Affinity DataIC50:  30nMAssay Description:Antagonist activity at human TRPA1 assessed as inhibition of AITC-induced calcium uptake by [45Ca2+] fluorimetry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50046742(CHEMBL3314489)
Affinity DataIC50:  45nMAssay Description:Antagonist activity at rat TRPA1 assessed as inhibition of AITC-induced calcium uptake by [45Ca2+] fluorimetry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50046743(CHEMBL3314488)
Affinity DataIC50:  140nMAssay Description:Antagonist activity at rat TRPA1 assessed as inhibition of AITC-induced calcium uptake by [45Ca2+] fluorimetry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50046742(CHEMBL3314489)
Affinity DataIC50:  170nMAssay Description:Antagonist activity at human TRPA1 assessed as inhibition of AITC-induced calcium uptake by [45Ca2+] fluorimetry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50046743(CHEMBL3314488)
Affinity DataIC50:  200nMAssay Description:Antagonist activity at human TRPA1 assessed as inhibition of AITC-induced calcium uptake by [45Ca2+] fluorimetry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50046744(CHEMBL3314487)
Affinity DataIC50:  230nMAssay Description:Antagonist activity at rat TRPA1 assessed as inhibition of AITC-induced calcium uptake by [45Ca2+] fluorimetry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50046745(CHEMBL3314486)
Affinity DataIC50:  230nMAssay Description:Antagonist activity at rat TRPA1 assessed as inhibition of AITC-induced calcium uptake by [45Ca2+] fluorimetry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50046745(CHEMBL3314486)
Affinity DataIC50:  300nMAssay Description:Antagonist activity at human TRPA1 assessed as inhibition of AITC-induced calcium uptake by [45Ca2+] fluorimetry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50046746(CHEMBL3314485)
Affinity DataIC50:  360nMAssay Description:Antagonist activity at rat TRPA1 assessed as inhibition of AITC-induced calcium uptake by [45Ca2+] fluorimetry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50046738(CHEMBL3314482)
Affinity DataIC50:  530nMAssay Description:Antagonist activity at rat TRPA1 assessed as inhibition of AITC-induced calcium uptake by [45Ca2+] fluorimetry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50046744(CHEMBL3314487)
Affinity DataIC50:  590nMAssay Description:Antagonist activity at human TRPA1 assessed as inhibition of AITC-induced calcium uptake by [45Ca2+] fluorimetry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50046746(CHEMBL3314485)
Affinity DataIC50:  710nMAssay Description:Antagonist activity at human TRPA1 assessed as inhibition of AITC-induced calcium uptake by [45Ca2+] fluorimetry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50046741(CHEMBL3314490)
Affinity DataIC50:  940nMAssay Description:Antagonist activity at human TRPA1 assessed as inhibition of AITC-induced calcium uptake by [45Ca2+] fluorimetry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50046749(CHEMBL3314484)
Affinity DataIC50:  970nMAssay Description:Antagonist activity at human TRPA1 assessed as inhibition of AITC-induced calcium uptake by [45Ca2+] fluorimetry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50046749(CHEMBL3314484)
Affinity DataIC50:  1.00E+3nMAssay Description:Antagonist activity at rat TRPA1 assessed as inhibition of AITC-induced calcium uptake by [45Ca2+] fluorimetry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50046738(CHEMBL3314482)
Affinity DataIC50:  1.20E+3nMAssay Description:Antagonist activity at human TRPA1 assessed as inhibition of AITC-induced calcium uptake by [45Ca2+] fluorimetry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50046741(CHEMBL3314490)
Affinity DataIC50:  1.30E+3nMAssay Description:Antagonist activity at rat TRPA1 assessed as inhibition of AITC-induced calcium uptake by [45Ca2+] fluorimetry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50046739(CHEMBL3314481)
Affinity DataIC50: >2.00E+3nMAssay Description:Antagonist activity at rat TRPA1 assessed as inhibition of AITC-induced calcium uptake by [45Ca2+] fluorimetry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50046739(CHEMBL3314481)
Affinity DataIC50: >2.00E+3nMAssay Description:Antagonist activity at human TRPA1 assessed as inhibition of AITC-induced calcium uptake by [45Ca2+] fluorimetry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50046731(CHEMBL3314483)
Affinity DataIC50: >4.00E+4nMAssay Description:Antagonist activity at human TRPA1 assessed as inhibition of AITC-induced calcium uptake by [45Ca2+] fluorimetry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50046731(CHEMBL3314483)
Affinity DataIC50: >4.00E+4nMAssay Description:Antagonist activity at rat TRPA1 assessed as inhibition of AITC-induced calcium uptake by [45Ca2+] fluorimetry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50046750(CHEMBL3314491)
Affinity DataIC50: >4.00E+7nMAssay Description:Antagonist activity at human TRPA1 assessed as inhibition of AITC-induced calcium uptake by [45Ca2+] fluorimetry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50046741(CHEMBL3314490)
Affinity DataEC50: >4.00E+4nMAssay Description:Agonist activity at human TRPA1 by [45Ca2+] fluorimetry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50046742(CHEMBL3314489)
Affinity DataEC50: >4.00E+4nMAssay Description:Agonist activity at human TRPA1 by [45Ca2+] fluorimetry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50046743(CHEMBL3314488)
Affinity DataEC50: >4.00E+4nMAssay Description:Agonist activity at human TRPA1 by [45Ca2+] fluorimetry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50046744(CHEMBL3314487)
Affinity DataEC50: >4.00E+4nMAssay Description:Agonist activity at human TRPA1 by [45Ca2+] fluorimetry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50046745(CHEMBL3314486)
Affinity DataEC50: >4.00E+4nMAssay Description:Agonist activity at human TRPA1 by [45Ca2+] fluorimetry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50046746(CHEMBL3314485)
Affinity DataEC50: >4.00E+4nMAssay Description:Agonist activity at human TRPA1 by [45Ca2+] fluorimetry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50046749(CHEMBL3314484)
Affinity DataEC50: >4.00E+4nMAssay Description:Agonist activity at human TRPA1 by [45Ca2+] fluorimetry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50046740(CHEMBL1939972 | US9186360, 90)
Affinity DataEC50: >4.00E+4nMAssay Description:Agonist activity at rat TRPA1 by [45Ca2+] fluorimetry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50046739(CHEMBL3314481)
Affinity DataEC50: >4.00E+4nMAssay Description:Agonist activity at rat TRPA1 by [45Ca2+] fluorimetry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50046738(CHEMBL3314482)
Affinity DataEC50: >4.00E+4nMAssay Description:Agonist activity at rat TRPA1 by [45Ca2+] fluorimetry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50046731(CHEMBL3314483)
Affinity DataEC50: >4.00E+4nMAssay Description:Agonist activity at rat TRPA1 by [45Ca2+] fluorimetry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50046749(CHEMBL3314484)
Affinity DataEC50: >4.00E+4nMAssay Description:Agonist activity at rat TRPA1 by [45Ca2+] fluorimetry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50046746(CHEMBL3314485)
Affinity DataEC50: >4.00E+4nMAssay Description:Agonist activity at rat TRPA1 by [45Ca2+] fluorimetry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50046745(CHEMBL3314486)
Affinity DataEC50: >4.00E+4nMAssay Description:Agonist activity at rat TRPA1 by [45Ca2+] fluorimetry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50046744(CHEMBL3314487)
Affinity DataEC50: >4.00E+4nMAssay Description:Agonist activity at rat TRPA1 by [45Ca2+] fluorimetry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50046743(CHEMBL3314488)
Affinity DataEC50: >4.00E+4nMAssay Description:Agonist activity at rat TRPA1 by [45Ca2+] fluorimetry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50046742(CHEMBL3314489)
Affinity DataEC50: >4.00E+4nMAssay Description:Agonist activity at rat TRPA1 by [45Ca2+] fluorimetry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50046741(CHEMBL3314490)
Affinity DataEC50: >4.00E+4nMAssay Description:Agonist activity at rat TRPA1 by [45Ca2+] fluorimetry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50362741(CHEMBL1939826)
Affinity DataEC50: >4.00E+4nMAssay Description:Agonist activity at rat TRPA1 by [45Ca2+] fluorimetry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50046740(CHEMBL1939972 | US9186360, 90)
Affinity DataEC50: >4.00E+4nMAssay Description:Agonist activity at human TRPA1 by [45Ca2+] fluorimetry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50046739(CHEMBL3314481)
Affinity DataEC50: >4.00E+4nMAssay Description:Agonist activity at human TRPA1 by [45Ca2+] fluorimetry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50362741(CHEMBL1939826)
Affinity DataEC50: >4.00E+4nMAssay Description:Agonist activity at human TRPA1 by [45Ca2+] fluorimetry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50046731(CHEMBL3314483)
Affinity DataEC50: >4.00E+4nMAssay Description:Agonist activity at human TRPA1 by [45Ca2+] fluorimetry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50046738(CHEMBL3314482)
Affinity DataEC50: >4.00E+4nMAssay Description:Agonist activity at human TRPA1 by [45Ca2+] fluorimetry assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed