Compile Data Set for Download or QSAR
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Found 28 Enz. Inhib. hit(s) with all data for entry = 50012675
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Albert-Ludwigs-Universit£T Freiburg

Curated by ChEMBL
LigandPNGBDBM50559306(CHEMBL4762202)
Affinity DataKd:  420nMAssay Description:Binding affinity to BRD4 BD1 (unknown origin) at 25 degree C by ITC analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Albert-Ludwigs-Universit£T Freiburg

Curated by ChEMBL
LigandPNGBDBM50559312(CHEMBL4747940)
Affinity DataKd:  170nMAssay Description:Binding affinity to BRD4 BD1 (unknown origin) at 37 degree C by ITC analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Albert-Ludwigs-Universit£T Freiburg

Curated by ChEMBL
LigandPNGBDBM50559308(CHEMBL4776447)
Affinity DataKd:  260nMAssay Description:Binding affinity to BRD4 BD1 (unknown origin) at 25 degree C by ITC analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Albert-Ludwigs-Universit£T Freiburg

Curated by ChEMBL
LigandPNGBDBM50559309(CHEMBL4762147)
Affinity DataKd:  80nMAssay Description:Binding affinity to BRD4 BD1 (unknown origin) at 25 degree C by ITC analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Albert-Ludwigs-Universit£T Freiburg

Curated by ChEMBL
LigandPNGBDBM50559310(CHEMBL4778822)
Affinity DataKd:  180nMAssay Description:Binding affinity to BRD4 BD1 (unknown origin) at 25 degree C by ITC analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Albert-Ludwigs-Universit£T Freiburg

Curated by ChEMBL
LigandPNGBDBM50559311(CHEMBL4780011)
Affinity DataKd:  140nMAssay Description:Binding affinity to BRD4 BD1 (unknown origin) at 25 degree C by ITC analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Albert-Ludwigs-Universit£T Freiburg

Curated by ChEMBL
LigandPNGBDBM50559312(CHEMBL4747940)
Affinity DataKd:  70nMAssay Description:Binding affinity to BRD4 BD1 (unknown origin) at 25 degree C by ITC analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Albert-Ludwigs-Universit£T Freiburg

Curated by ChEMBL
LigandPNGBDBM50559313(CHEMBL4783790)
Affinity DataKd:  6.41E+3nMAssay Description:Binding affinity to BRD4 BD1 (unknown origin) at 25 degree C by ITC analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Albert-Ludwigs-Universit£T Freiburg

Curated by ChEMBL
LigandPNGBDBM50559314(CHEMBL4741587)
Affinity DataKd: >4.00E+3nMAssay Description:Binding affinity to human BRD4 BD1 (N44 to E168 aa residues) by bromoKdELECT Discover assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Albert-Ludwigs-Universit£T Freiburg

Curated by ChEMBL
LigandPNGBDBM50151663(CHEMBL3774655)
Affinity DataKd:  5.60E+3nMAssay Description:Binding affinity to human BRD4 BD1 (N44 to E168 aa residues) by bromoKdELECT Discover assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Albert-Ludwigs-Universit£T Freiburg

Curated by ChEMBL
LigandPNGBDBM50266968(CHEMBL4065619 | US11773085, Compound B27)
Affinity DataKd: >990nMAssay Description:Binding affinity to human BRD4 BD1 (N44 to E168 aa residues) by bromoKdELECT Discover assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Albert-Ludwigs-Universit£T Freiburg

Curated by ChEMBL
LigandPNGBDBM50365262((+)-JQ1 | (S)-JQ1 (1) | CHEMBL1957266 | JQ1 | US10...)
Affinity DataKd:  13nMAssay Description:Binding affinity to human BRD4 BD1 (N44 to E168 aa residues) by bromoKdELECT Discover assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Albert-Ludwigs-Universit£T Freiburg

Curated by ChEMBL
LigandPNGBDBM50559306(CHEMBL4762202)
Affinity DataKd:  300nMAssay Description:Binding affinity to human BRD4 BD1 (N44 to E168 aa residues) by bromoKdELECT Discover assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Albert-Ludwigs-Universit£T Freiburg

Curated by ChEMBL
LigandPNGBDBM50559307(CHEMBL4787841)
Affinity DataKd:  82nMAssay Description:Binding affinity to human BRD4 BD1 (N44 to E168 aa residues) by bromoKdELECT Discover assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Albert-Ludwigs-Universit£T Freiburg

Curated by ChEMBL
LigandPNGBDBM50559308(CHEMBL4776447)
Affinity DataKd:  150nMAssay Description:Binding affinity to human BRD4 BD1 (N44 to E168 aa residues) by bromoKdELECT Discover assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Albert-Ludwigs-Universit£T Freiburg

Curated by ChEMBL
LigandPNGBDBM50559309(CHEMBL4762147)
Affinity DataKd:  60nMAssay Description:Binding affinity to human BRD4 BD1 (N44 to E168 aa residues) by bromoKdELECT Discover assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Albert-Ludwigs-Universit£T Freiburg

Curated by ChEMBL
LigandPNGBDBM50559310(CHEMBL4778822)
Affinity DataKd:  170nMAssay Description:Binding affinity to human BRD4 BD1 (N44 to E168 aa residues) by bromoKdELECT Discover assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Albert-Ludwigs-Universit£T Freiburg

Curated by ChEMBL
LigandPNGBDBM50559311(CHEMBL4780011)
Affinity DataKd:  85nMAssay Description:Binding affinity to human BRD4 BD1 (N44 to E168 aa residues) by bromoKdELECT Discover assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetBromodomain-containing protein 9(Homo sapiens (Human))
Albert-Ludwigs-Universit£T Freiburg

Curated by ChEMBL
LigandPNGBDBM50559314(CHEMBL4741587)
Affinity DataKd:  2.90E+3nMAssay Description:Binding affinity to human partial length BRD9 (R130 to V259 residues) by bromoKdELECT Discover assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))
Albert-Ludwigs-Universit£T Freiburg

Curated by ChEMBL
LigandPNGBDBM50157607(CHEMBL3753082 | US11773085, Compound B24)
Affinity DataKd:  99nMAssay Description:Binding affinity to human partial length BRD9 (R130 to V259 residues) by bromoKdELECT Discover assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 9(Homo sapiens (Human))
Albert-Ludwigs-Universit£T Freiburg

Curated by ChEMBL
LigandPNGBDBM50559306(CHEMBL4762202)
Affinity DataKd:  68nMAssay Description:Binding affinity to human partial length BRD9 (R130 to V259 residues) by bromoKdELECT Discover assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))
Albert-Ludwigs-Universit£T Freiburg

Curated by ChEMBL
LigandPNGBDBM50559307(CHEMBL4787841)
Affinity DataKd:  300nMAssay Description:Binding affinity to human partial length BRD9 (R130 to V259 residues) by bromoKdELECT Discover assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))
Albert-Ludwigs-Universit£T Freiburg

Curated by ChEMBL
LigandPNGBDBM50559308(CHEMBL4776447)
Affinity DataKd:  4.30nMAssay Description:Binding affinity to human partial length BRD9 (R130 to V259 residues) by bromoKdELECT Discover assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))
Albert-Ludwigs-Universit£T Freiburg

Curated by ChEMBL
LigandPNGBDBM50559309(CHEMBL4762147)
Affinity DataKd:  67nMAssay Description:Binding affinity to human partial length BRD9 (R130 to V259 residues) by bromoKdELECT Discover assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))
Albert-Ludwigs-Universit£T Freiburg

Curated by ChEMBL
LigandPNGBDBM50559310(CHEMBL4778822)
Affinity DataKd:  530nMAssay Description:Binding affinity to human partial length BRD9 (R130 to V259 residues) by bromoKdELECT Discover assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))
Albert-Ludwigs-Universit£T Freiburg

Curated by ChEMBL
LigandPNGBDBM50559311(CHEMBL4780011)
Affinity DataKd:  160nMAssay Description:Binding affinity to human partial length BRD9 (R130 to V259 residues) by bromoKdELECT Discover assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Albert-Ludwigs-Universit£T Freiburg

Curated by ChEMBL
LigandPNGBDBM50559312(CHEMBL4747940)
Affinity DataKd: <10nMAssay Description:Binding affinity to BRD4 BD1 (unknown origin) at 15 degree C by ITC analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Albert-Ludwigs-Universit£T Freiburg

Curated by ChEMBL
LigandPNGBDBM50559307(CHEMBL4787841)
Affinity DataKd:  50nMAssay Description:Binding affinity to BRD4 BD1 (unknown origin) at 25 degree C by ITC analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB