Compile Data Set for Download or QSAR
maximum 50k data
Found 13 Enz. Inhib. hit(s) with all data for entry = 50029482
TargetMu-type opioid receptor(CALF)
TBA

Curated by ChEMBL
LigandPNGBDBM50030143(CHEMBL41098 | bis-(1N-[10-hydroxy-4-methyl-14-oxo-...)
Affinity DataIC50:  0.400nMAssay Description:Inhibitory activity of the compound against Opioid receptor mu 1 binding to bovine striatal membraneMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(CALF)
TBA

Curated by ChEMBL
LigandPNGBDBM50421363(CHEMBL2304424)
Affinity DataIC50:  1.40nMAssay Description:Inhibitory activity of the compound against Opioid receptor mu 1 binding to bovine striatal membraneMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(CALF)
TBA

Curated by ChEMBL
LigandPNGBDBM50284914(CHEMBL297605 | MET-TAMO and N-CPM-MET-TAMO analogu...)
Affinity DataIC50:  2.90nMAssay Description:Inhibitory activity of the compound against Opioid receptor mu 1 binding to bovine striatal membraneMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(CALF)
TBA

Curated by ChEMBL
LigandPNGBDBM50030145(CHEMBL290701 | bis-(1N-[4-cyclopropylmethyl-10-hyd...)
Affinity DataIC50:  3.90nMAssay Description:Inhibitory activity of the compound against Opioid receptor mu 1 binding to bovine striatal membraneMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDelta-type opioid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50421363(CHEMBL2304424)
Affinity DataIC50:  5.30nMAssay Description:Inhibitory activity of the compound against Opioid receptor delta 1 binding to bovine striatal membraneMore data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50421363(CHEMBL2304424)
Affinity DataIC50:  7.70nMAssay Description:Inhibitory activity of the compound against Opioid receptor kappa1 binding to bovine striatal membraneMore data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50030145(CHEMBL290701 | bis-(1N-[4-cyclopropylmethyl-10-hyd...)
Affinity DataIC50:  10nMAssay Description:Inhibitory activity of the compound against Opioid receptor kappa1 binding to bovine striatal membraneMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDelta-type opioid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50030143(CHEMBL41098 | bis-(1N-[10-hydroxy-4-methyl-14-oxo-...)
Affinity DataIC50:  11nMAssay Description:Inhibitory activity of the compound against Opioid receptor delta 1 binding to bovine striatal membraneMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDelta-type opioid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50030145(CHEMBL290701 | bis-(1N-[4-cyclopropylmethyl-10-hyd...)
Affinity DataIC50:  24nMAssay Description:Inhibitory activity of the compound against Opioid receptor delta 1 binding to bovine striatal membraneMore data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50030143(CHEMBL41098 | bis-(1N-[10-hydroxy-4-methyl-14-oxo-...)
Affinity DataIC50:  41nMAssay Description:Inhibitory activity of the compound against Opioid receptor kappa1 binding to bovine striatal membraneMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDelta-type opioid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284914(CHEMBL297605 | MET-TAMO and N-CPM-MET-TAMO analogu...)
Affinity DataIC50:  52nMAssay Description:Inhibitory activity of the compound against Opioid receptor delta 1 binding to bovine striatal membraneMore data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284914(CHEMBL297605 | MET-TAMO and N-CPM-MET-TAMO analogu...)
Affinity DataIC50:  89nMAssay Description:Inhibitory activity of the compound against Opioid receptor kappa1 binding to bovine striatal membraneMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(CALF)
TBA

Curated by ChEMBL
LigandPNGBDBM50421363(CHEMBL2304424)
Affinity DataKd:  0.400nMAssay Description:Binding affinity towards Opioid receptor mu 1 using [3H]DAMGO expressed as KdMore data for this Ligand-Target Pair
In DepthDetails Article