Compile Data Set for Download or QSAR
maximum 50k data
Found 47 Enz. Inhib. hit(s) with all data for entry = 50005774
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040815(2-Methylsulfanyl-6,11-dihydro-dibenzo[b,e]oxepine-...)
Affinity DataIC50:  7nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040830(2-Bromo-6,11-dihydro-dibenzo[b,e]oxepine-11-carbox...)
Affinity DataIC50:  23nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040849(5H-Dibenzo[a,d]cycloheptene-5-carboxylic acid (2,6...)
Affinity DataIC50:  25nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040854(11-(2,6-Diisopropyl-phenylcarbamoyl)-2-methyl-6,11...)
Affinity DataIC50:  27nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040828(2-Iodo-6,11-dihydro-dibenzo[b,e]oxepine-11-carboxy...)
Affinity DataIC50:  35nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040831(3-Bromo-10,11-dihydro-5H-dibenzo[a,d]cycloheptene-...)
Affinity DataIC50:  39nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040826(10,11-Dihydro-5H-dibenzo[a,d]cycloheptene-5-carbox...)
Affinity DataIC50:  40nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040855(2-Methyl-6,11-dihydro-dibenzo[b,e]oxepine-11-carbo...)
Affinity DataIC50:  50nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040851(3-Methyl-10,11-dihydro-5H-dibenzo[a,d]cycloheptene...)
Affinity DataIC50:  55nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040841(2,9-Dibromo-6,11-dihydro-dibenzo[b,e]oxepine-11-ca...)
Affinity DataIC50:  58nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040848(2,3-Dimethyl-6,11-dihydro-dibenzo[b,e]oxepine-11-c...)
Affinity DataIC50:  64nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040843(2-Bromo-6,11-dihydro-dibenzo[b,e]oxepine-11-carbox...)
Affinity DataIC50:  74nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040840(7-Bromo-5,11-dihydro-10-oxa-1-aza-dibenzo[a,d]cycl...)
Affinity DataIC50:  78nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040824(6,11-Dihydro-dibenzo[b,e]oxepine-11-carboxylic aci...)
Affinity DataIC50:  94nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040822(4-Bromo-2-methyl-6,11-dihydro-dibenzo[b,e]oxepine-...)
Affinity DataIC50:  100nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040829(2-Methyl-6,11-dihydro-dibenzo[b,e]oxepine-11-carbo...)
Affinity DataIC50:  110nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040817(9-Bromo-2-methyl-6,11-dihydro-dibenzo[b,e]oxepine-...)
Affinity DataIC50:  120nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040814(2-Ethyl-6,11-dihydro-dibenzo[b,e]oxepine-11-carbox...)
Affinity DataIC50:  130nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040837(2-Methoxy-6,11-dihydro-dibenzo[b,e]oxepine-11-carb...)
Affinity DataIC50:  140nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040818(2-Chloro-6,11-dihydro-dibenzo[b,e]oxepine-11-carbo...)
Affinity DataIC50:  150nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040813(7-Bromo-5,11-dihydro-10-thia-dibenzo[a,d]cyclohept...)
Affinity DataIC50:  150nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040833(2-Trifluoromethyl-6,11-dihydro-dibenzo[b,e]oxepine...)
Affinity DataIC50:  160nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040812(3-Bromo-6,11-dihydro-dibenzo[b,e]oxepine-11-carbox...)
Affinity DataIC50:  180nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040823(11-(2,6-Diisopropyl-phenylcarbamoyl)-6,11-dihydro-...)
Affinity DataIC50:  180nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040847(9-Bromo-6,11-dihydro-dibenzo[b,e]oxepine-11-carbox...)
Affinity DataIC50:  190nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040845(2-Methyl-6,11-dihydro-dibenzo[b,e]oxepine-11-carbo...)
Affinity DataIC50:  190nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040844(2-Methyl-6,11-dihydro-dibenzo[b,e]oxepine-11-carbo...)
Affinity DataIC50:  190nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040810(2-Fluoro-6,11-dihydro-dibenzo[b,e]oxepine-11-carbo...)
Affinity DataIC50:  210nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040821(2-Bromo-5-methyl-6-oxo-6,11-dihydro-5H-dibenzo[b,e...)
Affinity DataIC50:  240nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040811(2-Nitro-6,11-dihydro-dibenzo[b,e]oxepine-11-carbox...)
Affinity DataIC50:  240nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040827(2-Bromo-6,11-dihydro-dibenzo[b,e]oxepine-11-carbox...)
Affinity DataIC50:  250nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040852(2-Methyl-6,11-dihydro-dibenzo[b,e]oxepine-11-carbo...)
Affinity DataIC50:  260nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040838(2-Methyl-6,11-dihydro-dibenzo[b,e]oxepine-11-carbo...)
Affinity DataIC50:  270nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50022279(3-(2,4-Difluoro-phenyl)-1-[4-(2,2-dimethyl-propyl)...)
Affinity DataIC50:  320nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040839(2-Methyl-6,11-dihydro-dibenzo[b,e]oxepine-11-carbo...)
Affinity DataIC50:  350nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040836(2-Isopropyl-6,11-dihydro-dibenzo[b,e]oxepine-11-ca...)
Affinity DataIC50:  360nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040816(6,11-Dihydro-dibenzo[b,e]oxepine-2,11-dicarboxylic...)
Affinity DataIC50:  400nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040819(2-tert-Butyl-6,11-dihydro-dibenzo[b,e]oxepine-11-c...)
Affinity DataIC50:  420nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040835(2-Cyano-6,11-dihydro-dibenzo[b,e]oxepine-11-carbox...)
Affinity DataIC50:  490nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040825(2-Isopropyl-6,11-dihydro-dibenzo[b,e]oxepine-11-ca...)
Affinity DataIC50:  500nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040846(2-tert-Butyl-6,11-dihydro-dibenzo[b,e]oxepine-11-c...)
Affinity DataIC50:  500nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040820(2-Bromo-6,11-dihydro-dibenzo[b,e]oxepine-11-carbox...)
Affinity DataIC50:  580nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040842(2-Methyl-6,11-dihydro-dibenzo[b,e]oxepine-11-carbo...)
Affinity DataIC50:  580nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040832(2-Hydroxymethyl-6,11-dihydro-dibenzo[b,e]oxepine-1...)
Affinity DataIC50:  580nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040853(5,11-Dihydro-10-oxa-1-aza-dibenzo[a,d]cycloheptene...)
Affinity DataIC50:  640nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040850(2-Methyl-6,11-dihydro-dibenzo[b,e]oxepine-11-carbo...)
Affinity DataIC50:  730nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50040834(3-Bromo-6,11-dihydro-dibenzo[b,e]oxepine-11-carbox...)
Affinity DataIC50:  940nMAssay Description:In vitro inhibitory activity against acyl coenzyme A:cholesterol acyltransferase in liver microsomes isolated from cholesterol-fed rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed