PDB Entry - 5K7K

(Status - Released)

Summary information:

Title: Design and Optimization of Biaryl Ether Aryl Sulfonamides as Selective Inhibitors of NaV1.7: Discovery of Clinical Candidate PF-05089771

PDB DOI: https://doi.org/10.2210/pdb5k7k/pdb

Primary publication DOI: https://doi.org/10.1021/acs.jmedchem.7b00598

Entry authors: Swain, N., Chrencik, J.

Initial deposition on: 26 May 2016

Initial release on: 7 June 2017

Latest revision on: 27 September 2023

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Structure coordinates (PDB)

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Validation report (mmCIF)

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