Skip to main content
SpringerLink
Log in

A New Binding Mode of Competitive Antagonists to Metabotropic Glutamate Receptors Exemplified by the mGluR1-Receptor Antagonist AIDA (RS-Aminoindan-1,5-Dicarboxylic Acid)

  • Published:
Doklady Biochemistry and Biophysics Aims and scope Submit manuscript

This is a preview of subscription content, log in via an institution to check access.

Access this article

Log in via an institution

Price excludes VAT (USA)
Tax calculation will be finalised during checkout.

Instant access to the full article PDF.

Institutional subscriptions

REFERENCES

  1. Kunishima, N., Shimada, Y., Tsuji, Y., et al., Nature, 2000, vol. 407, no.6807, pp. 971–977.

    PubMed  Google Scholar 

  2. Costantino, G., Macchiarulo, A., and Pellicciari, R., J. Med. Chem., 1999, vol. 42, no.26, pp. 5390–5401.

    PubMed  Google Scholar 

  3. Pellicciari, R., Costantino, G., and Macchiarulo, A., Pharm. Acta Helv., 2000, vol. 74, nos.2- 3, pp. 231–237.

    Google Scholar 

  4. Brauner-Osborne, H., Egebjerg, J., Nielsen, E., et al., J. Med. Chem., 2000, vol. 43, no.14, pp. 2609–2645.

    PubMed  Google Scholar 

  5. Pellicciari, R., Costantino, G., Giovagnoni, E., et al., Bioorg. Med. Chem. Lett., 1998, vol. 8, no.12, pp. 1569–1574.

    PubMed  Google Scholar 

  6. Belenikin, M.S., Baskin, I.I., Palyulin, V.A., and Zefirov, N.S., Dokl. Akad. Nauk, 2002, vol. 383, no.5.

  7. Kumar, S. and Nussinov, R., J. Mol. Biol., 1999, vol. 293, no.5, pp. 1241–1255.

    PubMed  Google Scholar 

  8. Moroni, F., Lombardi, G., Thomsen, C., et al., J.Pharmacol. Exp. Ther., 1997, vol. 281, no.2, pp. 721–729.

    PubMed  Google Scholar 

  9. Schoepp, D.D., Jane, D.E., and Monn, J.A., Neuropharmacology, 1999, vol. 38, no.10, pp. 1431–1476.

    PubMed  Google Scholar 

  10. Sybyl 6.6. Tripos, Inc. 1699 South Hanley Road, St. Louis, (Mo.) 63144. http://www.tripos.com.

  11. Marelius, J., Kolmodin, K., Feierberg, I., et al., J. Mol. Graphics Mod., 1998, vol. 16, pp. 213–225.

    Google Scholar 

  12. Morris, G.M., Goodsell, D.S., Halliday, R.S., et al., J. Comput. Chem., 1998, vol. 19, pp. 1639–1662.

    Google Scholar 

Download references

Author information

Authors and Affiliations

  1. Moscow State University, Vorob'evy gory, Moscow, 119992, Russia

    M. S. Belenikin, I. I. Baskin, V. A. Palyulin & N. S. Zefirov

Authors
  1. M. S. Belenikin
    View author publications

    You can also search for this author in PubMed Google Scholar

  2. I. I. Baskin
    View author publications

    You can also search for this author in PubMed Google Scholar

  3. V. A. Palyulin
    View author publications

    You can also search for this author in PubMed Google Scholar

  4. N. S. Zefirov
    View author publications

    You can also search for this author in PubMed Google Scholar

Rights and permissions

Reprints and permissions

About this article

Cite this article

Belenikin, M.S., Baskin, I.I., Palyulin, V.A. et al. A New Binding Mode of Competitive Antagonists to Metabotropic Glutamate Receptors Exemplified by the mGluR1-Receptor Antagonist AIDA (RS-Aminoindan-1,5-Dicarboxylic Acid). Doklady Biochemistry and Biophysics 384, 131–135 (2002). https://doi.org/10.1023/A:1016076028063

Download citation

  • Issue Date:

  • DOI: https://doi.org/10.1023/A:1016076028063

Keywords

Search

Navigation