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Synthesis and AMPA-receptor modulating activity of benzodioxanecarboxylic and piperonylic acid derivatives

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A series of amides of benzodioxane-6-carboxylic and piperonylic acids have been synthesized. Biological studies showed that some of the synthesized compounds influence the central nervous system (in particular, AMPA receptors).

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Correspondence to M. I. Lavrov.

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Translated from Khimiko-Farmatsevticheskii Zhurnal, Vol. 46, No. 2, pp. 27 – 30, February, 2012.

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Lavrov, M.I., Lapteva, V.L., Grigor’ev, V.V. et al. Synthesis and AMPA-receptor modulating activity of benzodioxanecarboxylic and piperonylic acid derivatives. Pharm Chem J 46, 92–95 (2012). https://doi.org/10.1007/s11094-012-0740-1

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  • DOI: https://doi.org/10.1007/s11094-012-0740-1

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