PDB Entry - 5EM7

(Status - Released)

Summary information:

Title: EGFR kinase domain mutant ""TMLR"" with pyridone compound 13: 4-[(2-methoxyphenyl)amino]-~{N}-[4-(4-methylpiperazin-1-yl)phenyl]-2-oxidanylidene-1~{H}-pyridine-3-carboxamide

PDB DOI: https://doi.org/10.2210/pdb5em7/pdb

Primary publication DOI: https://doi.org/10.1021/acsmedchemlett.5b00428

Entry authors: Eigenbrot, C., Yu, C.

Initial deposition on: 5 November 2015

Initial release on: 30 December 2015

Latest revision on: 6 March 2024

Downloads:

Structure coordinates (PDBx/mmCIF)

Structure coordinates (PDBML)

Structure coordinates (PDB)

X-ray diffraction data (PDBx/mmCIF)

Validation report (XML)

Validation report (PDF)

Links to more resources for 5EM7 at: