Issue 8, 2014
From the journal:

RSC Advances

A one-pot process for palladium catalyzed direct C–H acylation of anilines in water using a removable ortho directing group†

Fruzsina Szabó,a   Dániel Simkóa  and  Zoltán Novák*a  

* Corresponding authors

a MTA-ELTE “Lendület” Catalysis and Organic Synthesis Research Group, Institute of Chemistry, Eötvös University, Pázmány Péter stny. 1/a, H-1117 Budapest, Hungary
E-mail: novakz@elte.hu
Fax: +36-1-372-2592
Tel: +36-1-372-2500#1610

Abstract

A new mild, practical method for the synthesis of aminobenzophenone derivatives through a three step one-pot reaction sequence involving acylation of anilines, palladium catalyzed cross-dehydrogenative coupling of the formed anilides and the hydrolytic cleavage is reported. The full reaction sequence was performed under aqueous conditions.

Graphical abstract: A one-pot process for palladium catalyzed direct C–H acylation of anilines in water using a removable ortho directing group

About
Cited by
Related
Download options Please wait...

Supplementary files

Article information

DOI
https://doi.org/10.1039/C3RA45160G
Article type
Communication
Submitted
16 Sep 2013
Accepted
04 Dec 2013
First published
05 Dec 2013

RSC Adv., 2014,4, 3883-3886

Permissions

Request permissions

A one-pot process for palladium catalyzed direct C–H acylation of anilines in water using a removable ortho directing group

F. Szabó, D. Simkó and Z. Novák, RSC Adv., 2014, 4, 3883 DOI: 10.1039/C3RA45160G

To request permission to reproduce material from this article, please go to the Copyright Clearance Center request page.

If you are an author contributing to an RSC publication, you do not need to request permission provided correct acknowledgement is given.

If you are the author of this article, you do not need to request permission to reproduce figures and diagrams provided correct acknowledgement is given. If you want to reproduce the whole article in a third-party publication (excluding your thesis/dissertation for which permission is not required) please go to the Copyright Clearance Center request page.

Read more about how to correctly acknowledge RSC content.

Social activity

Spotlight

Advertisements